Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with Target = 'Proteasome subunit alpha type-1'
TargetProteasome subunit alpha type-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50652793(CHEMBL5653589)
Affinity DataKd:  9.78E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetProteasome subunit alpha type-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50652792(CHEMBL3752910)
Affinity DataKd:  1.04E+4nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetProteasome subunit alpha type-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50577134(CHEMBL4877708)
Affinity DataIC50: 3.80nMAssay Description:Inhibition of caspase-like activity of human proteasome beta-1c subunit using SUC-LLE-AMC as flurogenic substrate preincubated for 15 mins followed b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteasome subunit alpha type-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50577116(CHEMBL4872258)
Affinity DataIC50: 4.36E+3nMAssay Description:Inhibition of caspase-like activity of human proteasome beta-1c subunit using SUC-LLE-AMC as flurogenic substrate preincubated for 15 mins followed b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteasome subunit alpha type-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50007203(CHEMBL3237875)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of caspase-like activity of human proteasome beta-1c subunit using SUC-LLE-AMC as flurogenic substrate preincubated for 15 mins followed b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteasome subunit alpha type-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50577130(CHEMBL4846410)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of caspase-like activity of human proteasome beta-1c subunit using SUC-LLE-AMC as flurogenic substrate preincubated for 15 mins followed b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteasome subunit alpha type-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50577131(CHEMBL4855915)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of caspase-like activity of human proteasome beta-1c subunit using SUC-LLE-AMC as flurogenic substrate preincubated for 15 mins followed b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProteasome subunit alpha type-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50577133(CHEMBL4870115)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of caspase-like activity of human proteasome beta-1c subunit using SUC-LLE-AMC as flurogenic substrate preincubated for 15 mins followed b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed