Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with Target = 'Potassium voltage-gated channel subfamily A member 6'
TargetPotassium voltage-gated channel subfamily A member 6(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50067880(4-methoxy-7H-furo[3,2-g]chromen-7-one | 5-methoxyp...)
Affinity DataKd:  1.87E+5nMAssay Description:Blockade of peak K+ currents against Kv1.6 geneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 6(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50279106(5-(4-phenoxybutoxy)psoralen | 4-(4-phenoxybutoxy)-...)
Affinity DataIC50: 130nMAssay Description:Inhibition of human Kv1.6 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 6(Rat)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456976(CHEMBL4207745)
Affinity DataIC50: 170nMAssay Description:Inhibition of rat Kv1.6 expressed in Xenopus laevis oocytes at -90 mV holding potential by two-electrode voltage clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 6(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50456976(CHEMBL4207745)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human Kv1.6 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 6(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50456974(CHEMBL3621636)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of human Kv1.6 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 6(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50220547(oroidin base | oroidin | 4,5-Dibromo-1H-pyrrole-2-...)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of human Kv1.6 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 6(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50456970(CHEMBL3261431)
Affinity DataIC50: 7.90E+3nMAssay Description:Inhibition of human Kv1.6 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 6(Rat)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456975(CHEMBL4213446)
Affinity DataIC50: 9.80E+3nMAssay Description:Inhibition of rat Kv1.6 expressed in Xenopus laevis oocytes at -90 mV holding potential by two-electrode voltage clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 6(Rat)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456982(CHEMBL4208517)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat Kv1.6 expressed in Xenopus laevis oocytes at -90 mV holding potential by two-electrode voltage clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 6(Rat)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50220547(oroidin base | oroidin | 4,5-Dibromo-1H-pyrrole-2-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat Kv1.6 expressed in Xenopus laevis oocytes at -90 mV holding potential by two-electrode voltage clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 6(Rat)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456969(CHEMBL4202870)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat Kv1.6 expressed in Xenopus laevis oocytes at -90 mV holding potential by two-electrode voltage clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 6(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50456975(CHEMBL4213446)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of human Kv1.6 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 6(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50456977(CHEMBL3261430)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of human Kv1.6 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 6(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50456969(CHEMBL4202870)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of human Kv1.6 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 6(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50456971(CHEMBL4210636)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of human Kv1.6 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 6(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50456982(CHEMBL4208517)
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of human Kv1.6 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 6(Human)
University of Kiel

Curated by ChEMBL
LigandPNGBDBM50456973(Clathrodin)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human Kv1.6 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed