Compile Data Set for Download or QSAR
Report error Found 1705 Enz. Inhib. hit(s) with Target = 'Platelet-activating factor receptor'
TargetPlatelet-activating factor receptor(Guinea pig)
Paris Diderot University

Curated by ChEMBL
LigandPNGBDBM50046991((1,4-bis(3,4,5-trimethoxybenzoyl)piperazin-2-yl)me...)
Affinity DataEC50:  680nMAssay Description:Inhibition of [3H]PAF binding to rabbit platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Paris Diderot University

Curated by ChEMBL
LigandPNGBDBM50046983(2,2-Dimethyl-propionic acid 1,4-bis-(3,4,5-trimeth...)
Affinity DataEC50:  300nMAssay Description:Inhibition of [3H]PAF binding to rabbit platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Paris Diderot University

Curated by ChEMBL
LigandPNGBDBM50251276(CHEMBL514432 | BN 52021 | ginkgolide B | Gingkolid...)
Affinity DataEC50:  180nMAssay Description:Inhibition of [3H]PAF binding to rabbit platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Paris Diderot University

Curated by ChEMBL
LigandPNGBDBM50046986(Acetic acid 1,4-bis-(3,4,5-trimethoxy-benzoyl)-pip...)
Affinity DataEC50:  400nMAssay Description:Inhibition of [3H]PAF binding to rabbit platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Paris Diderot University

Curated by ChEMBL
LigandPNGBDBM50046966(Butyl-carbamic acid 1,4-bis-(3,4,5-trimethoxy-benz...)
Affinity DataEC50:  700nMAssay Description:Inhibition of [3H]PAF binding to rabbit platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Paris Diderot University

Curated by ChEMBL
LigandPNGBDBM50046968(2-Chloro-benzoic acid 1,4-bis-(3,4,5-trimethoxy-be...)
Affinity DataEC50:  450nMAssay Description:Inhibition of [3H]PAF binding to rabbit platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Paris Diderot University

Curated by ChEMBL
LigandPNGBDBM50046976((1,2-Dimethyl-propyl)-carbamic acid 1,4-bis-(3,4,5...)
Affinity DataEC50:  70nMAssay Description:Inhibition of [3H]PAF binding to rabbit platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Paris Diderot University

Curated by ChEMBL
LigandPNGBDBM50046978((1,3-Dimethyl-butyl)-carbamic acid 1,4-bis-(3,4,5-...)
Affinity DataEC50:  180nMAssay Description:Inhibition of [3H]PAF binding to rabbit platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Paris Diderot University

Curated by ChEMBL
LigandPNGBDBM50046963(2-Ethyl-butyric acid 1,4-bis-(3,4,5-trimethoxy-ben...)
Affinity DataEC50:  90nMAssay Description:Inhibition of [3H]PAF binding to rabbit platelet membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Boehringer Ingelheim International

WIPO
LigandPNGBDBM552607(WO2022101377, Example 6)
Affinity DataAssay Description:USING AN ENDPOINT ASSAY HEK293 cells overexpressing human PAFR (produced in-house) are seeded into a Poly-D-Lysine coated 384 well white cell culture...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2022
Entry Details
WIPO WO2022101377

TargetPlatelet-activating factor receptor(Guinea pig)
Paris Diderot University

Curated by ChEMBL
LigandPNGBDBM50021572(CHEMBL287709 | (2S,3S)-2-(3,4-Dimethoxy-phenyl)-3-...)
Affinity DataIC50: 0nMAssay Description:Inhibitor concentration required to block 50% of the specific [3H]PAF binding to rabbit platelet membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Boehringer Ingelheim International

WIPO
LigandPNGBDBM50280478(N-((S)-1-Ethoxymethyl-3-methyl-butyl)-4-(2-methyl-...)
Affinity DataIC50: 0.0150nMAssay Description:Antagonistic activity for inhibition of [3H]PAF receptor binding to washed human platelet membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetPlatelet-activating factor receptor(Human)
Boehringer Ingelheim International

WIPO
LigandPNGBDBM50011635(CHEMBL277701 | 1-{3-[4-(2-Chloro-phenyl)-9-methyl-...)
Affinity DataIC50: 0.200nMAssay Description:PAF-antagonist activity determined in dog platelets by PAF-binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Boehringer Ingelheim International

WIPO
LigandPNGBDBM85035(bloodplatelet-activatingfactor | CAS_65154-06-5 | ...)
Affinity DataIC50: 0.280nMAssay Description:Displacement of [3H]PAF from platelet activating factor receptor in human platelets after 3 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPlatelet-activating factor receptor(Human)
Boehringer Ingelheim International

WIPO
LigandPNGBDBM50011650(CHEMBL20195 | 1-{3-[4-(2-Chloro-phenyl)-9-methyl-6...)
Affinity DataIC50: 0.300nMAssay Description:PAF-antagonist activity determined in dog platelets by PAF-binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Paris Diderot University

Curated by ChEMBL
LigandPNGBDBM50033236(8,9-Dichloro-2-methyl-5-[4-(2-methyl-imidazo[4,5-c...)
Affinity DataIC50: 0.300nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Paris Diderot University

Curated by ChEMBL
LigandPNGBDBM50033242(3-Cyclohexyl-6-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50: 0.400nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Boehringer Ingelheim International

WIPO
LigandPNGBDBM552615(WO2022101377, Example 14)
Affinity DataIC50: 0.400nMAssay Description:USING AN ENDPOINT ASSAY HEK293 cells overexpressing human PAFR (produced in-house) are seeded into a Poly-D-Lysine coated 384 well white cell culture...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2022
Entry Details
WIPO WO2022101377

TargetPlatelet-activating factor receptor(Human)
Boehringer Ingelheim International

WIPO
LigandPNGBDBM50617206(CHEMBL5439289)
Affinity DataIC50: 0.400nMAssay Description:Antagonist activity at human PAFR expressed in HEK293 cells assessed as inhibition of PAF C-16 ligand induced receptor activation preincubated for 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Paris Diderot University

Curated by ChEMBL
LigandPNGBDBM50033212(7,8-Dichloro-4-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50: 0.5nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Paris Diderot University

Curated by ChEMBL
LigandPNGBDBM50033213(7,8-Dichloro-1-methyl-4-[4-(2-methyl-imidazo[4,5-c...)
Affinity DataIC50: 0.5nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Paris Diderot University

Curated by ChEMBL
LigandPNGBDBM50033211(7,8-Dichloro-4-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50: 0.5nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Paris Diderot University

Curated by ChEMBL
LigandPNGBDBM50033257(1,8-Dimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50: 0.5nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Paris Diderot University

Curated by ChEMBL
LigandPNGBDBM50004622(CHEMBL106908 | 4-(2-Chloro-phenyl)-2-methyl-6-[4-(...)
Affinity DataIC50: 0.5nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Boehringer Ingelheim International

WIPO
LigandPNGBDBM552651(WO2022101377, Example 50)
Affinity DataIC50: 0.5nMAssay Description:USING AN ENDPOINT ASSAY HEK293 cells overexpressing human PAFR (produced in-house) are seeded into a Poly-D-Lysine coated 384 well white cell culture...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2022
Entry Details
WIPO WO2022101377

TargetPlatelet-activating factor receptor(Human)
Boehringer Ingelheim International

WIPO
LigandPNGBDBM552651(WO2022101377, Example 50)
Affinity DataIC50: 0.5nMAssay Description:Antagonist activity at human PAFR expressed in HEK293 cells assessed as inhibition of PAF C-16 ligand induced receptor activation preincubated for 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-activating factor receptor(Human)
Boehringer Ingelheim International

WIPO
LigandPNGBDBM50011611(CHEMBL19640 | 1-{3-[4-(2-Chloro-phenyl)-9-methyl-6...)
Affinity DataIC50: 0.600nMAssay Description:PAF-antagonist activity determined in dog platelets by PAF-binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Paris Diderot University

Curated by ChEMBL
LigandPNGBDBM50033223(7,8-Dimethyl-4-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50: 0.600nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Paris Diderot University

Curated by ChEMBL
LigandPNGBDBM50033240(1-Methyl-5-[4-(2-methyl-imidazo[4,5-c]pyridin-1-yl...)
Affinity DataIC50: 0.600nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Paris Diderot University

Curated by ChEMBL
LigandPNGBDBM50033238(3-(4-Chloro-phenyl)-1,8-dimethyl-5-[4-(2-methyl-im...)
Affinity DataIC50: 0.600nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Boehringer Ingelheim International

WIPO
LigandPNGBDBM50011623(CHEMBL20019 | 2a-{3-[4-(2-Chloro-phenyl)-9-methyl-...)
Affinity DataIC50: 0.700nMAssay Description:PAF-antagonist activity determined in dog platelets by PAF-binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Boehringer Ingelheim International

WIPO
LigandPNGBDBM50011634(CHEMBL19747 | 4-{3-[4-(2-Chloro-phenyl)-9-methyl-6...)
Affinity DataIC50: 0.700nMAssay Description:PAF-antagonist activity determined in dog platelets by PAF-binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Paris Diderot University

Curated by ChEMBL
LigandPNGBDBM50033214(7,8-Dimethyl-4-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50: 0.700nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Paris Diderot University

Curated by ChEMBL
LigandPNGBDBM50033264(3-Cyclohexyl-1,8-dimethyl-5-[4-(2-methyl-imidazo[4...)
Affinity DataIC50: 0.700nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Boehringer Ingelheim International

WIPO
LigandPNGBDBM552674(WO2022101377, Example 73)
Affinity DataIC50: 0.700nMAssay Description:USING AN ENDPOINT ASSAY HEK293 cells overexpressing human PAFR (produced in-house) are seeded into a Poly-D-Lysine coated 384 well white cell culture...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2022
Entry Details
WIPO WO2022101377

TargetPlatelet-activating factor receptor(Human)
Boehringer Ingelheim International

WIPO
LigandPNGBDBM552674(WO2022101377, Example 73)
Affinity DataIC50: 0.700nMAssay Description:Antagonist activity at human PAFR expressed in HEK293 cells assessed as inhibition of PAF C-16 ligand induced receptor activation preincubated for 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Paris Diderot University

Curated by ChEMBL
LigandPNGBDBM50033260(3-Isobutoxymethyl-1,8-dimethyl-5-[4-(2-methyl-imid...)
Affinity DataIC50: 0.800nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Paris Diderot University

Curated by ChEMBL
LigandPNGBDBM50033206(7,8-Dichloro-4-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50: 0.900nMAssay Description:Antagonistic activity was tested against Platelet-Activating Factor-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Boehringer Ingelheim International

WIPO
LigandPNGBDBM50280339(L-671284 | (S)-2-[4-(2-Benzenesulfonyl-ethoxy)-3-m...)
Affinity DataIC50: 1nMAssay Description:Compound was evaluated for inhibitory activity of binding of [3H]-C18 PAF to human platelet membrane Platelet activating factor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetPlatelet-activating factor receptor(Human)
Boehringer Ingelheim International

WIPO
LigandPNGBDBM50013923(CHEMBL99294 | 3-(1-Butyl-4-methoxy-naphthalen-2-yl...)
Affinity DataIC50: 1nMAssay Description:Inhibition of [3H]PAF binding to platelet activating factor receptor citrate-treated dog bloodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Boehringer Ingelheim International

WIPO
LigandPNGBDBM50011603(CHEMBL281779 | 1-{3-[4-(2-Chloro-phenyl)-9-methyl-...)
Affinity DataIC50: 1nMAssay Description:PAF-antagonist activity determined in dog platelets by PAF-binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Boehringer Ingelheim International

WIPO
LigandPNGBDBM50011640(CHEMBL283162 | 4-(2-Chloro-phenyl)-2-(3-indazol-1-...)
Affinity DataIC50: 1nMAssay Description:PAF-antagonist activity determined in dog platelets by PAF-binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Boehringer Ingelheim International

WIPO
LigandPNGBDBM50011653(CHEMBL282883 | 2-{3-[4-(2-Chloro-phenyl)-9-methyl-...)
Affinity DataIC50: 1nMAssay Description:PAF-antagonist activity determined in dog platelets by PAF-binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Paris Diderot University

Curated by ChEMBL
LigandPNGBDBM50033234(1,3-Dimethyl-7-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50: 1nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Boehringer Ingelheim International

WIPO
LigandPNGBDBM552632(WO2022101377, Example 31)
Affinity DataIC50: 1.10nMAssay Description:USING AN ENDPOINT ASSAY HEK293 cells overexpressing human PAFR (produced in-house) are seeded into a Poly-D-Lysine coated 384 well white cell culture...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2022
Entry Details
WIPO WO2022101377

TargetPlatelet-activating factor receptor(Human)
Boehringer Ingelheim International

WIPO
LigandPNGBDBM50617208(CHEMBL5411707)
Affinity DataIC50: 1.10nMAssay Description:Antagonist activity at human PAFR expressed in HEK293 cells assessed as inhibition of PAF C-16 ligand induced receptor activation preincubated for 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Paris Diderot University

Curated by ChEMBL
LigandPNGBDBM50033233(8,9-Dichloro-1-methyl-5-[4-(2-methyl-imidazo[4,5-c...)
Affinity DataIC50: 1.20nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Paris Diderot University

Curated by ChEMBL
LigandPNGBDBM50033229(8,9-Dimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50: 1.30nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Paris Diderot University

Curated by ChEMBL
LigandPNGBDBM50033249(5,7,9-Trimethyl-2-[4-(2-methyl-imidazo[4,5-c]pyrid...)
Affinity DataIC50: 1.30nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Paris Diderot University

Curated by ChEMBL
LigandPNGBDBM50004615(CHEMBL318172 | 4-(2-Chloro-phenyl)-2-methyl-6-[4-(...)
Affinity DataIC50: 1.30nMAssay Description:In vitro inhibition of PAF-induced aggregation of rabbit washed platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
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