Compile Data Set for Download or QSAR
Report error Found 144 Enz. Inhib. hit(s) with Target = 'Phospholipase A2, major isoenzyme'
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50055367([3-Aminooxalyl-1-(3-chloro-benzyl)-2-ethyl-1H-indo...)
Affinity DataIC50: 3nMAssay Description:Compound was tested for inhibition of porcine secreted pancreatic PLA2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50055384((3-Aminooxalyl-1-biphenyl-3-ylmethyl-2-methyl-1H-i...)
Affinity DataIC50: 7nMAssay Description:Compound was tested for inhibition of porcine secretory pancreatic Phospholipase A2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50055384((3-Aminooxalyl-1-biphenyl-3-ylmethyl-2-methyl-1H-i...)
Affinity DataIC50: 7nMAssay Description:Inhibition of pig group IB phospholipase A2 incubated for 1 hrs by scintillation counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50055383(2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-methyl-1Hind...)
Affinity DataIC50: 15nMAssay Description:Compound was tested for inhibition of porcine secretory pancreatic Phospholipase A2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50055383(2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-methyl-1Hind...)
Affinity DataIC50: 15nMAssay Description:Inhibition of pig group IB phospholipase A2 incubated for 1 hrs by scintillation counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50004495(CHEMBL101015 | Hexadecanoic acid 3-[hydroxy-(2-hyd...)
Affinity DataIC50: 30nMAssay Description:In vitro inhibition of porcine pancreatic phospholipase A2 evaluated by monomeric substrate assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50004502(CHEMBL101972 | Phosphoric acid 2-hexadecanoylamino...)
Affinity DataIC50: 30nMAssay Description:In vitro inhibition of porcine pancreatic phospholipase A2 evaluated by monomeric substrate assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50055366(Varespladib sodium | (3-Aminooxalyl-1-benzyl-2-eth...)
Affinity DataIC50: 48nMAssay Description:Compound was tested for inhibition of porcine secretory pancreatic PLA2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50055366(Varespladib sodium | (3-Aminooxalyl-1-benzyl-2-eth...)
Affinity DataIC50: 48nMAssay Description:Inhibition of pig group IB phospholipase A2 incubated for 1 hrs by scintillation counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50055371((3-aminooxalyl-1-biphenyl-2-ylmethyl-2-methyl-1H-i...)
Affinity DataIC50: 97nMAssay Description:Compound was tested for inhibition of porcine secretory pancreatic Phospholipase A2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50055371((3-aminooxalyl-1-biphenyl-2-ylmethyl-2-methyl-1H-i...)
Affinity DataIC50: 97nMAssay Description:Inhibition of pig group IB phospholipase A2 incubated for 1 hrs by scintillation counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50004499((R)-O-(2-Hexadecanamidoisohexyl) phosphocholine | ...)
Affinity DataIC50: 230nMAssay Description:In vitro inhibition of porcine pancreatic phospholipase A2 evaluated by monomeric substrate assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50269843(Bolinaquinone | CHEMBL477692)
Affinity DataIC50: 400nMAssay Description:Inhibition of pig pancreatic group 1 secretory phospholipase A2 by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50055287(4-(1-Benzyl-3-carbamoylmethyl-2-methyl-1H-indol-4-...)
Affinity DataIC50: 610nMAssay Description:Compound was tested for the inhibitory activity against porcine pancreatic PLA2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50031087(3-(4-Fluoro-phenyl)-2-(4-methanesulfonyl-phenyl)-5...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibitory activity rat polymorphonuclear leukocyte phospholipase-A2 (PMN-PLA2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50004504(CHEMBL102135 | (R)-O-(2-Hexadecanamidopropyl] phos...)
Affinity DataIC50: 1.40E+3nMAssay Description:In vitro inhibition of porcine pancreatic phospholipase A2 evaluated by monomeric substrate assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50206912((+/-)-3-O-[4-(4,5-dihydro-5-oxo-1,2,4-4H-oxadiazol...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of pig group IB PLA2 by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50004502(CHEMBL101972 | Phosphoric acid 2-hexadecanoylamino...)
Affinity DataIC50: 2.60E+3nMAssay Description:In vitro inhibition of porcine pancreatic phospholipase A2 evaluated by Deoxycholate-phospholipid mixed micelle assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50004495(CHEMBL101015 | Hexadecanoic acid 3-[hydroxy-(2-hyd...)
Affinity DataIC50: 3.50E+3nMAssay Description:In vitro inhibition of porcine pancreatic phospholipase A2 evaluated by Deoxycholate-phospholipid mixed micelle assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50316463(1-[4-(4,5-Dihydro-1,2,4-(4H)-5-oxo-oxadiazol-3-ylm...)
Affinity DataIC50: 3.58E+3nMAssay Description:Inhibition of porcine group 1B phospholipase A2 by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50055287(4-(1-Benzyl-3-carbamoylmethyl-2-methyl-1H-indol-4-...)
Affinity DataIC50: 3.66E+3nMAssay Description:Compound was tested for the inhibitory activity against human pancreatic PLA2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50004493(CHEMBL101890 | O-(2-hexadecanamidoethyl) phosphoch...)
Affinity DataIC50: 4.00E+3nMAssay Description:In vitro inhibition of porcine pancreatic phospholipase A2 evaluated by monomeric substrate assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50004505(CHEMBL101828 | (S)-O-(2-Hexadecanamidoisohexyl) ph...)
Affinity DataIC50: 4.50E+3nMAssay Description:In vitro inhibition of porcine pancreatic phospholipase A2 evaluated by monomeric substrate assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50004500(CHEMBL319067 | Phosphoric acid mono-(2-hexadecanoy...)
Affinity DataIC50: 5.00E+3nMAssay Description:In vitro inhibition of porcine pancreatic phospholipase A2 evaluated by monomeric substrate assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50316459(1-[4-(4,5-Dihydro-1,2,4-(4H)-5-oxo-oxadiazol-3-ylm...)
Affinity DataIC50: 5.33E+3nMAssay Description:Inhibition of porcine group 1B phospholipase A2 by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50280987(1N-[12-isopropyl-2,6-dimethyltricyclo[8.4.0.02,7]t...)
Affinity DataIC50: 5.40E+3nMAssay Description:Tested for its inhibitory activity against Phospholipase A2 (PLA2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50206913((+/-)-3-O-[4-(4,5-dihydro-5-oxo-1,2,4-4H-oxadiazol...)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of pig group IB PLA2 by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50004501(CHEMBL102090 | (E)-(R)-O-(2-Dec-3-enamidoisohexyl)...)
Affinity DataIC50: 6.00E+3nMAssay Description:In vitro inhibition of porcine pancreatic phospholipase A2 evaluated by monomeric substrate assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50316458(1-[4-(4,5-Dihydro-1,2,4-(4H)-5-oxo-oxadiazol-3-ylm...)
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of porcine group 1B phospholipase A2 by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50316456(1-[4-(4,5-Dihydro-1,2,4-(4H)-5-oxo-oxadiazol-3-ylm...)
Affinity DataIC50: 7.41E+3nMAssay Description:Inhibition of porcine group 1B phospholipase A2 by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM23771(CHEMBL146186 | (3-{[1-benzyl-3-(carbamoylmethyl)-2...)
Affinity DataIC50: 8.00E+3nMAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2008
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50004498(CHEMBL99161 | O-[2-(2-Naphthalenecarboxamido)ethyl...)
Affinity DataIC50: 8.00E+3nMAssay Description:In vitro inhibition of porcine pancreatic phospholipase A2 evaluated by monomeric substrate assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM23771(CHEMBL146186 | (3-{[1-benzyl-3-(carbamoylmethyl)-2...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of pig group IB PLA2 by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM23771(CHEMBL146186 | (3-{[1-benzyl-3-(carbamoylmethyl)-2...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of porcine group 1B phospholipase A2 by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50206908((+/-)-1-O-(4-cyanomethylphenyl)-3-O-[4-(4,5-dihydr...)
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibition of pig group IB PLA2 by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50004496(CHEMBL318193 | Phosphoric acid mono-(2-hexadecanoy...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of porcine pancreatic phospholipase A2 evaluated by monomeric substrate assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50316457(1-[4-(4,5-Dihydro-1,2,4-(4H)-5-oxo-oxadiazol-3-ylm...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of porcine group 1B phospholipase A2 by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50591711(CHEMBL5203236)
Affinity DataIC50: 1.07E+4nMAssay Description:Inhibition of porcine PLA2G1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50591712(CHEMBL5194852)
Affinity DataIC50: 1.24E+4nMAssay Description:Inhibition of porcine PLA2G1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50591713(CHEMBL5207115)
Affinity DataIC50: 1.36E+4nMAssay Description:Inhibition of porcine PLA2G1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50591715(CHEMBL5179709)
Affinity DataIC50: 1.45E+4nMAssay Description:Inhibition of porcine PLA2G1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50591714(CHEMBL5200953)
Affinity DataIC50: 1.48E+4nMAssay Description:Inhibition of porcine PLA2G1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50004497(CHEMBL330205 | Phosphoric acid 2-trimethylamino-et...)
Affinity DataIC50: 1.50E+4nMAssay Description:In vitro inhibition of porcine pancreatic phospholipase A2 evaluated by Deoxycholate-phospholipid mixed micelle assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50280984(C-((4aS,10aR)-7-Isopropyl-1,4a-dimethyl-1,2,3,4,4a...)
Affinity DataIC50: 2.10E+4nMAssay Description:Tested for its inhibitory activity against Phospholipase A2 (PLA2)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50316460(1-[4-(4,5-Dihydro-1,2,4-(4H)-5-oxo-oxadiazol-3-ylm...)
Affinity DataIC50: 2.16E+4nMAssay Description:Inhibition of porcine group 1B phospholipase A2 by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50316454(1-[4-(4,5-Dihydro-1,2,4-(4H)-5-oxo-oxadiazol-3-ylm...)
Affinity DataIC50: 2.45E+4nMAssay Description:Inhibition of porcine group 1B phospholipase A2 by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50031087(3-(4-Fluoro-phenyl)-2-(4-methanesulfonyl-phenyl)-5...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory activity porcine pancreatic phospholipase-A2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50206904((+/-)-1-O-benzyl-3-O-[4-(4,5-dihydro-5-oxo-1,2,4-4...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of pig group IB PLA2 by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50316462(1-[4-(4,5-Dihydro-1,2,4-(4H)-5-oxo-oxadiazol-3-ylm...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of porcine group 1B phospholipase A2 by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetPhospholipase A2, major isoenzyme(Pig)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50316444(1-[4-(4,5-Dihydro-1,2,4(4H)-5-oxo-oxadiazol-3-yl)b...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of porcine group 1B phospholipase A2 by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
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