Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with Target = 'Peptidyl-prolyl cis-trans isomerase NIMA-interacting 4'
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 4(Human)
Horizon Discovery

Curated by ChEMBL
LigandPNGBDBM50437711(CHEMBL2409076)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of Par14 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 4(Human)
Horizon Discovery

Curated by ChEMBL
LigandPNGBDBM50095936(CHEMBL3590367)
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of Pin4 (unknown origin) pre-incubated for 10 mins before addition of Suc-Ala-Glu-Pro-Phe-pNA substrate in presence of alpha-chymotrypsin ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 4(Human)
Horizon Discovery

Curated by ChEMBL
LigandPNGBDBM50080528(Cycloheximid | 3-((R)-2-((1S,3S,5S)-3,5-dimethyl-2...)
Affinity DataKi:  1.87E+5nMAssay Description:Inhibition constant(Ki) for inhibition of PPIase activity of Escherichia coli parvulin (Conc=4 nM) of Parvulins sfamilyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed