Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with Target = 'Penicillin-binding protein 4'
TargetPenicillin-binding protein 4(Bacillus subtilis (strain 168))
Wesleyan University

Curated by ChEMBL
LigandPNGBDBM50370584(Beepen-VK | Betapen-VK | Penapar-VK | Penicillin P...)
Affinity DataKoff:  1.90E+4s-1Assay Description:Inhibition of Bacillus subtilis 168 PBP4 after 30 mins by SDS-PAGEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetPenicillin-binding protein 4(Bacillus subtilis (strain 168))
Wesleyan University

Curated by ChEMBL
LigandPNGBDBM50495677(CHEMBL3114799)
Affinity DataKoff:  190s-1Assay Description:Inhibition of Bacillus subtilis 168 PBP4 after 30 mins by SDS-PAGEMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetPenicillin-binding protein 4(Staphylococcus aureus)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50483327(CEFTOBIPROLE MEDOCARIL)
Affinity DataIC50: 1.44E+3nMAssay Description:Inhibition of methicillin-susceptible Staphylococcus aureus ATCC 29213 PBP 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPenicillin-binding protein 4(Staphylococcus aureus)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50482776(CHEBI:70718 | Ceftaroline Fosamil | PPI-0903 | TAK...)
Affinity DataIC50: 1.46E+3nMAssay Description:Binding affinity to methicillin-susceptible Staphylococcus aureus PBP 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPenicillin-binding protein 4(Staphylococcus aureus)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50378857(Zeftera | Zevtera | CEFTOBIPROLE)
Affinity DataIC50: 1.87E+3nMAssay Description:Inhibition of bocillin FL binding to methicillin-susceptible Staphylococcus aureus ATCC 29213 penicillin-binding protein 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetPenicillin-binding protein 4(Staphylococcus aureus)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50053180(Sodium; (2S,3S,5R)-3-methyl-4,4,7-trioxo-3-((Z)-2-...)
Affinity DataIC50: 1.40E+4nMAssay Description:Compound was tested for inhibition of Penicillin-binding protein 4 from Staphylococcus aureus (Schoch).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2012
Entry Details Article
PubMed
TargetPenicillin-binding protein 4(Staphylococcus aureus)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50053179(Sodium; (2S,3S,5R)-3-methyl-4,4,7-trioxo-3-((Z)-2-...)
Affinity DataIC50: 1.50E+4nMAssay Description:Compound was tested for inhibition of Penicillin-binding protein 4 from Staphylococcus aureus (Schoch).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2012
Entry Details Article
PubMed
TargetPenicillin-binding protein 4(Staphylococcus aureus)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50053183(Trifluoro-methanesulfonate1-[(E)-3-((2S,3S,5R)-2-c...)
Affinity DataIC50: 1.50E+4nMAssay Description:Compound was tested for inhibition of Penicillin-binding protein 4 from Staphylococcus aureus (Schoch).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2012
Entry Details Article
PubMed
TargetPenicillin-binding protein 4(Staphylococcus aureus)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50076680(Sodium; (2S,3R,5R)-3-((Z)-2-cyano-vinyl)-3-methyl-...)
Affinity DataIC50: 1.70E+4nMAssay Description:Compound was tested for inhibition of Penicillin-binding protein 4 from Staphylococcus aureus (Schoch).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2012
Entry Details Article
PubMed
TargetPenicillin-binding protein 4(Staphylococcus aureus)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50103601(CHEBI:29007 | Ceftriaxone)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of bocillin FL binding to methicillin-susceptible Staphylococcus aureus ATCC 29213 penicillin-binding protein 4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetPenicillin-binding protein 4(Staphylococcus aureus)
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50053175((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-((E)-2-thiazol-...)
Affinity DataIC50: 1.43E+5nMAssay Description:Compound was tested for inhibition of Penicillin-binding protein 4 from Staphylococcus aureus (Schoch).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2012
Entry Details Article
PubMed