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Report error Found 255 Enz. Inhib. hit(s) with Target = 'Papain'
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409589(CHEMBL2028920)
Affinity DataKi:  0.100nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409598(CHEMBL2028910)
Affinity DataKi:  0.120nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50284944(((S)-1-(S)-Oxiranyl-2-phenyl-ethyl)-carbamic acid ...)
Affinity DataKi:  0.208nMAssay Description:Kinetic parameter (Ki 1/min) was evaluated for the inactivation of papainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409597(CHEMBL2028912)
Affinity DataKi:  0.280nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409590(CHEMBL2028909)
Affinity DataKi:  0.560nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409583(CHEMBL2028921)
Affinity DataKi:  0.580nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409586(CHEMBL2028907)
Affinity DataKi:  0.770nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409592(CHEMBL2028908)
Affinity DataKi:  0.780nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409587(CHEMBL2028911)
Affinity DataKi:  0.950nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409588(CHEMBL2028919)
Affinity DataKi:  1.35nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50157741(CHEMBL374508 | E-64 | E64)
Affinity DataIC50: 2nMAssay Description:Inhibition of papaya papain using Z-Leu-Leu-Arg-AMC as substrate after 30 mins by spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50213272(CHEBI:6426 | Leupeptin)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of papaya papain using cbzFRamc substrate preincubated for 10 mins followed by addition of substrate and measured every 30 sec for 60 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50553988(Antipain)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of papaya papain using cbzFRamc substrate preincubated for 10 mins followed by addition of substrate and measured every 30 sec for 60 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50304793((S)-benzyl 1-(2-cyano-1,2-dimethylhydrazinyl)-1-ox...)
Affinity DataKi:  3.90nMAssay Description:Inhibition of Carica papaya papain by microtiter plate spectrofluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50553989(CHEMBL4764505)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of papaya papain using cbzFRamc substrate preincubated for 10 mins followed by addition of substrate and measured every 30 sec for 60 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50304796((S)-benzyl 1-(2-cyano-1-methyl-2-phenethylhydrazin...)
Affinity DataKi:  6.30nMAssay Description:Inhibition of Carica papaya papain by microtiter plate spectrofluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50118425(Z-leu-Val-Agly-Val-OBzl | CHEMBL263061)
Affinity DataKi:  6.70nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50157741(CHEMBL374508 | E-64 | E64)
Affinity DataIC50: 7nMAssay Description:Inhibition of papaya papain using Z-Leu-Leu-Arg-AMC as substrate after 30 mins by fluorescence microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50304794((S)-benzyl 1-(2-cyano-1,2-dimethylhydrazinyl)-4-me...)
Affinity DataKi:  8.20nMAssay Description:Inhibition of Carica papaya papain by microtiter plate spectrofluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50304797((S)-benzyl 1-(2-cyano-1-methyl-2-pentylhydrazinyl)...)
Affinity DataKi:  10nMAssay Description:Inhibition of Carica papaya papain by microtiter plate spectrofluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50094931(Oxirane-2,3-dicarboxylic acid monoethyl ester | CH...)
Affinity DataIC50: 11nMAssay Description:The compound was evaluated for inhibition of papain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM20124(tert-butyl N-[(1S)-1-[(2-oxoethyl)carbamoyl]-2-phe...)
Affinity DataKi:  15nMAssay Description:Enzyme activities were calculated from kinetic measurements performed by spectrophotometric detection of the product p-nitroaniline (pNA) at waveleng...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2008
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM20114(tert-butyl N-[(1S)-1-[(cyanomethyl)carbamoyl]-2-(4...)
Affinity DataKi:  16nMAssay Description:Enzyme activities were calculated from kinetic measurements performed by spectrophotometric detection of the product p-nitroaniline (pNA) at waveleng...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2008
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM20120((2S)-N-(cyanomethyl)-3-phenyl-2-[(4-phenylphenyl)f...)
Affinity DataKi:  16nMAssay Description:Enzyme activities were calculated from kinetic measurements performed by spectrophotometric detection of the product p-nitroaniline (pNA) at waveleng...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2008
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409584(CHEMBL2028906)
Affinity DataKi:  17nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50553990(CHEMBL4788595)
Affinity DataIC50: 18nMAssay Description:Inhibition of papaya papain using cbzFRamc substrate preincubated for 10 mins followed by addition of substrate and measured every 30 sec for 60 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409599(CHEMBL2028925)
Affinity DataKi:  20nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM20113(tert-butyl N-[(1S)-1-[(cyanomethyl)carbamoyl]-2-(n...)
Affinity DataKi:  21nMAssay Description:Enzyme activities were calculated from kinetic measurements performed by spectrophotometric detection of the product p-nitroaniline (pNA) at waveleng...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2008
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409594(CHEMBL2028924)
Affinity DataKi:  21nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50364010(CHEMBL1950263)
Affinity DataKi:  23nMAssay Description:Inhibition of papaya papainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50118412(Boc-Agly-Val-Agly-OEt | CHEMBL135413)
Affinity DataKi:  24nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409596(CHEMBL2028923)
Affinity DataKi:  28nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM20107(tert-butyl N-[(1S)-2-(4-bromophenyl)-1-[(cyanometh...)
Affinity DataKi:  29nM ΔG°:  -43.0kJ/molepH: 6.5 T: 2°CAssay Description:Enzyme activities were calculated from kinetic measurements performed by spectrophotometric detection of the product p-nitroaniline (pNA) at waveleng...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2008
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409591(CHEMBL2028922)
Affinity DataKi:  30nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409582(CHEMBL2028926)
Affinity DataKi:  32nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50303441(9-(3,5-Difluorophenyl)-6-(ethylamino)-9H-purine-2-...)
Affinity DataIC50: 33.1nMAssay Description:Inhibition of papaya papainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50304795((S)-benzyl 1-(2-benzyl-2-cyano-1-methylhydrazinyl)...)
Affinity DataKi:  42nMAssay Description:Inhibition of Carica papaya papain by microtiter plate spectrofluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50303420(6-(3,5-Difluorophenylamino)-9-ethyl-9H-purine-2-ca...)
Affinity DataIC50: 44.7nMAssay Description:Inhibition of papaya papainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50157741(CHEMBL374508 | E-64 | E64)
Affinity DataIC50: 47nMAssay Description:Inhibition of Carica papaya papain by spectrofluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409585(CHEMBL2028918)
Affinity DataKi:  59nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409595(CHEMBL2028917)
Affinity DataKi:  61nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM20119((2S)-N-(cyanomethyl)-3-phenyl-2-(phenylformamido)p...)
Affinity DataKi:  62nMAssay Description:Enzyme activities were calculated from kinetic measurements performed by spectrophotometric detection of the product p-nitroaniline (pNA) at waveleng...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2008
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50366497(CHEMBL1790164)
Affinity DataIC50: 70nMAssay Description:Ability to inhibit papain was evaluated by amidolytic method using fluorogenic or chromogenic substratesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50229129(4-methyl-N-((S)-1-oxo-3-phenyl-1-((S)-5-phenyl-1-(...)
Affinity DataIC50: 81nMAssay Description:Inhibition of papaya papain assessed as reduction in p-nitoaniline release using Nalpha-benzoyl-L-arginine 4-nitroanilide hydrochloride as substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50409593(CHEMBL2028913)
Affinity DataKi:  100nMAssay Description:In vitro inhibition of papain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50546078(CHEMBL4750628)
Affinity DataIC50: 106nMAssay Description:Inhibition of papaya papain assessed as reduction in p-nitoaniline release using Nalpha-benzoyl-L-arginine 4-nitroanilide hydrochloride as substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50546076(CHEMBL4744708)
Affinity DataIC50: 124nMAssay Description:Inhibition of papaya papain assessed as reduction in p-nitoaniline release using Nalpha-benzoyl-L-arginine 4-nitroanilide hydrochloride as substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50546077(CHEMBL4742162)
Affinity DataIC50: 129nMAssay Description:Inhibition of papaya papain assessed as reduction in p-nitoaniline release using Nalpha-benzoyl-L-arginine 4-nitroanilide hydrochloride as substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50070495([(S)-1-((S)-1-Formyl-4-guanidino-butylcarbamoyl)-2...)
Affinity DataIC50: 130nMAssay Description:Ability to inhibit papain was evaluated by amidolytic method using fluorogenic or chromogenic substratesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetPapain(Papaya)
University of Gda£?Sk

Curated by ChEMBL
LigandPNGBDBM50546071(CHEMBL4762654)
Affinity DataIC50: 148nMAssay Description:Inhibition of papaya papain assessed as reduction in p-nitoaniline release using Nalpha-benzoyl-L-arginine 4-nitroanilide hydrochloride as substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
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