Compile Data Set for Download or QSAR
Report error Found 674 Enz. Inhib. hit(s) with Target = 'PAS domain-containing serine/threonine-protein kinase'
TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 5.5nMAssay Description:Inhibition of human PASK using KKLNRTLSFAEPG as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 15.8nMAssay Description:Inhibition of human PASK using KKLNRTLSFAEPG as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50154943(CHEMBL3775576)
Affinity DataIC50: 260nMAssay Description:Inhibition of PASK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2017
Entry Details Article
PubMed
TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463442(3-(4-(4-Methoxyphenyl)piperidin-1-yl)-2-phenylquin...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified hPASK from insect cells (0.02 μg) is added to a 50 μL reaction mix containing 40 mM HEPES (pH 7.0), 100 mM KCl, 5 mM MgCl2, 1 mM D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463448(3-Morpholino-2-phenylquinoxaline-6-carboxylic acid...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified hPASK from insect cells (0.02 μg) is added to a 50 μL reaction mix containing 40 mM HEPES (pH 7.0), 100 mM KCl, 5 mM MgCl2, 1 mM D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463449(3-(4-Methyl-1,4-diazepan-1-yl)-2-phenylquinoxaline...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified hPASK from insect cells (0.02 μg) is added to a 50 μL reaction mix containing 40 mM HEPES (pH 7.0), 100 mM KCl, 5 mM MgCl2, 1 mM D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463450(3-(Isopropylamino)-2-phenylquinoxaline-6-carboxyli...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified hPASK from insect cells (0.02 μg) is added to a 50 μL reaction mix containing 40 mM HEPES (pH 7.0), 100 mM KCl, 5 mM MgCl2, 1 mM D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
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TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463451(2-Phenyl-3-(4-(pyrimidin-2-yl)piperazin-1-yl)quino...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified hPASK from insect cells (0.02 μg) is added to a 50 μL reaction mix containing 40 mM HEPES (pH 7.0), 100 mM KCl, 5 mM MgCl2, 1 mM D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463452(2-Phenyl-3-(4-(5-(trifluoromethyl)pyridin-2-yl)pip...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified hPASK from insect cells (0.02 μg) is added to a 50 μL reaction mix containing 40 mM HEPES (pH 7.0), 100 mM KCl, 5 mM MgCl2, 1 mM D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463453(2-phenyl-3-(4-(quinolin-2-yl)piperazin-1-yl)quinox...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified hPASK from insect cells (0.02 μg) is added to a 50 μL reaction mix containing 40 mM HEPES (pH 7.0), 100 mM KCl, 5 mM MgCl2, 1 mM D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463454(2-(Azepan-1-yl)-3-phenylquinoxaline-6-carboxylic a...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified hPASK from insect cells (0.02 μg) is added to a 50 μL reaction mix containing 40 mM HEPES (pH 7.0), 100 mM KCl, 5 mM MgCl2, 1 mM D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463455(3-Phenyl-2-(piperidin-1-yl)quinoxaline-6-carboxyli...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified hPASK from insect cells (0.02 μg) is added to a 50 μL reaction mix containing 40 mM HEPES (pH 7.0), 100 mM KCl, 5 mM MgCl2, 1 mM D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463456(2-(4-(4-Chlorophenyl)piperidin-1-yl)-3-(4-fluoroph...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified hPASK from insect cells (0.02 μg) is added to a 50 μL reaction mix containing 40 mM HEPES (pH 7.0), 100 mM KCl, 5 mM MgCl2, 1 mM D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463457(2-(4-(3-Chlorophenyl)piperidin-1-yl)-3-(4-fluoroph...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified hPASK from insect cells (0.02 μg) is added to a 50 μL reaction mix containing 40 mM HEPES (pH 7.0), 100 mM KCl, 5 mM MgCl2, 1 mM D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463458(3-(4-Fluorophenyl)-2-(4-(4-methoxyphenyl)piperidin...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified hPASK from insect cells (0.02 μg) is added to a 50 μL reaction mix containing 40 mM HEPES (pH 7.0), 100 mM KCl, 5 mM MgCl2, 1 mM D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463459(3-(4-Fluorophenyl)-2-(4-(pyridin-2-yl)piperazin-1-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified hPASK from insect cells (0.02 μg) is added to a 50 μL reaction mix containing 40 mM HEPES (pH 7.0), 100 mM KCl, 5 mM MgCl2, 1 mM D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
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TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463460(2-Phenyl-3-(4-(3-(trifluoromethyl)pyridin-2-yl)pip...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified hPASK from insect cells (0.02 μg) is added to a 50 μL reaction mix containing 40 mM HEPES (pH 7.0), 100 mM KCl, 5 mM MgCl2, 1 mM D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463461(3-(4-Fluorophenyl)-2-(4-(4-(trifluoromethyl)phenyl...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified hPASK from insect cells (0.02 μg) is added to a 50 μL reaction mix containing 40 mM HEPES (pH 7.0), 100 mM KCl, 5 mM MgCl2, 1 mM D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463462(2,3-Bis(4-phenylpiperidin-1-yl)quinoxaline-6-carbo...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified hPASK from insect cells (0.02 μg) is added to a 50 μL reaction mix containing 40 mM HEPES (pH 7.0), 100 mM KCl, 5 mM MgCl2, 1 mM D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463463(2,3-Bis(4-methoxyphenyl)-6-(1H-tetrazol-5-yl)quino...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified hPASK from insect cells (0.02 μg) is added to a 50 μL reaction mix containing 40 mM HEPES (pH 7.0), 100 mM KCl, 5 mM MgCl2, 1 mM D...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463464(2-Phenyl-3-(4-(4-(trifluoromethyl)phenyl)piperazin...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463465(2-Phenyl-3-(4-(pyridin-2-yl)piperazin-1-yl)quinoxa...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463466(3-(4-(3-Chlorophenyl)piperazin-1-yl)-2-phenylquino...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463467(3-(4-Methylpiperazin-1-yl)-2-phenylquinoxaline-6-c...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463468(2-Phenyl-3-(piperazin-1-yl)quinoxaline-6-carboxyli...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463469(2-Phenyl-3-(4-phenylpiperazin-1-yl)quinoxaline-6-c...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463470(2-Phenyl-3-(4-(4-(trifluoromethyl)phenyl)piperidin...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463471(3-(4-(4-Chlorophenyl)piperazin-1-yl)-2-phenylquino...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463472(3-(4-(4-Methoxyphenyl)piperazin-1-yl)-2-phenylquin...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
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TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463473(3-(4-(3-Chlorophenyl)piperidin-1-yl)-2-phenylquino...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463474(2-Phenyl-3-(piperidin-1-yl)quinoxaline-6-carboxyli...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463475(2-Phenyl-3-(4-phenylpiperidin-1-yl)quinoxaline-6-c...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463476(3-(Azepan-1-yl)-2-phenylquinoxaline-6-carboxylic a...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463477(3-(4-(4-Chlorophenyl)piperidin-1-yl)-2-phenylquino...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463448(3-Morpholino-2-phenylquinoxaline-6-carboxylic acid...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463449(3-(4-Methyl-1,4-diazepan-1-yl)-2-phenylquinoxaline...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463450(3-(Isopropylamino)-2-phenylquinoxaline-6-carboxyli...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463451(2-Phenyl-3-(4-(pyrimidin-2-yl)piperazin-1-yl)quino...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463452(2-Phenyl-3-(4-(5-(trifluoromethyl)pyridin-2-yl)pip...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463453(2-phenyl-3-(4-(quinolin-2-yl)piperazin-1-yl)quinox...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463456(2-(4-(4-Chlorophenyl)piperidin-1-yl)-3-(4-fluoroph...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463458(3-(4-Fluorophenyl)-2-(4-(4-methoxyphenyl)piperidin...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
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TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463460(2-Phenyl-3-(4-(3-(trifluoromethyl)pyridin-2-yl)pip...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463461(3-(4-Fluorophenyl)-2-(4-(4-(trifluoromethyl)phenyl...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463462(2,3-Bis(4-phenylpiperidin-1-yl)quinoxaline-6-carbo...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463463(2,3-Bis(4-methoxyphenyl)-6-(1H-tetrazol-5-yl)quino...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463478(3-(4-(N-Methylmethan-3-ylsulfonamido)piperidin-1-y...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463479(3-(3,4-Dihydroquinolin-1(2H)-yl)-2-phenylquinoxali...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463480(3-(Isopropyl(methyl)amino)-2-phenylquinoxaline-6-c...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM463481(3-(Cyclopropyl(methyl)amino)-2-phenylquinoxaline-6...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified PASK (UniProt # Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2021
Entry Details
Go to US Patent

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