Compile Data Set for Download or QSAR
Report error Found 42 Enz. Inhib. hit(s) with Target = 'Opioid receptor delta 1'
TargetOpioid receptor delta 1(Guinea pig)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50268462(c[L-Phe-D-pro-L-Phe-L-trp] | CHEMBL506616)
Affinity DataIC50: 2.60E+3nMAssay Description:Displacement of [3H]DPDPE from delta-opioid receptor in guinea pig brain membranes after 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetOpioid receptor delta 1(Guinea pig)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50083926((cyclazocine)2-{4-[(2,4-Diamino-pteridin-6-ylmethy...)
Affinity DataKi:  0.580nMAssay Description:Displacement of [3H]Naltrindole from DOR in guinea pig brain membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetOpioid receptor delta 1(Bovine)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM85393(CAM | 14β-(p-chlorocinnamoylamino)-7,8-dihydr...)
Affinity DataKi:  0.75nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/6/2012
Entry Details
PubMed
TargetOpioid receptor delta 1(Guinea pig)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50018731(3-cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexa...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]Naltrindole from DOR in guinea pig brain membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetOpioid receptor delta 1(Bovine)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM82090(DALLE)
Affinity DataKi:  1.80nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details
PubMed
TargetOpioid receptor delta 1(Bovine)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM21025([D-Ala2-D-Leu5]enkephalin | (D-Ala2,D-Leu5)-Enkeph...)
Affinity DataKi:  1.80nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details
PubMed
TargetOpioid receptor delta 1(Guinea pig)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50007102(CHEMBL79470 | MR-2034 | 6,11-Dimethyl-3-(tetrahydr...)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]Naltrindole from DOR in guinea pig brain membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetOpioid receptor delta 1(Guinea pig)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50045114(EKC | CHEMBL55033 | 3-Cyclopropylmethyl-6-ethyl-8-...)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]Naltrindole from DOR in guinea pig brain membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetOpioid receptor delta 1(Rhesus macaque)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50458147(CHEMBL4204891)
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]naltrindole from DOR in monkey brain cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetOpioid receptor delta 1(Guinea pig)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50085020((3-Cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hex...)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]Naltrindole from DOR in guinea pig brain membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetOpioid receptor delta 1(Rhesus macaque)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50001031(SKF 10,047 (-) | CHEMBL330376 | SKF 10,047 (+) | S...)
Affinity DataKi:  5.5nMAssay Description:Displacement of [3H]naltrindole from DOR in monkey brain cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetOpioid receptor delta 1(Rhesus macaque)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50458145(CHEMBL4207341)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]naltrindole from DOR in monkey brain cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetOpioid receptor delta 1(Bovine)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM82090(DALLE)
Affinity DataKi:  7.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details
PubMed
TargetOpioid receptor delta 1(Guinea pig)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50101160(3-Cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexa...)
Affinity DataKi:  8.30nMAssay Description:Displacement of [3H]Naltrindole from DOR in guinea pig brain membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetOpioid receptor delta 1(Guinea pig)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50458137(CHEMBL4210742)
Affinity DataKi:  8.30nMAssay Description:Displacement of [3H]Naltrindole from DOR in guinea pig brain membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetOpioid receptor delta 1(Bovine)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM21025([D-Ala2-D-Leu5]enkephalin | (D-Ala2,D-Leu5)-Enkeph...)
Affinity DataKi:  9.70nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details
PubMed
TargetOpioid receptor delta 1(Guinea pig)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50458143(CHEMBL4215981)
Affinity DataKi:  9.80nMAssay Description:Displacement of [3H]Naltrindole from DOR in guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetOpioid receptor delta 1(Guinea pig)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50254563(3-Cyclopropylmethyl-6-ethyl-11-methyl-1-oxo-1,2,3,...)
Affinity DataKi:  9.80nMAssay Description:Displacement of [3H]Naltrindole from DOR in guinea pig brain membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetOpioid receptor delta 1(Rhesus macaque)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50458146(CHEMBL4209962)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]naltrindole from DOR in monkey brain cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetOpioid receptor delta 1(Bovine)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM85395(MC-CAM)
Affinity DataKi:  12nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/6/2012
Entry Details
PubMed
TargetOpioid receptor delta 1(Guinea pig)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50092176(3-Cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexa...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]Naltrindole from DOR in guinea pig brain membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetOpioid receptor delta 1(Bovine)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM81934(Beta-Endorphin)
Affinity DataKi:  14nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details
PubMed
TargetOpioid receptor delta 1(Bovine)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM85394(N-CPM-CACO)
Affinity DataKi:  16nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/6/2012
Entry Details
PubMed
TargetOpioid receptor delta 1(Bovine)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM50000788([17-(2,3-3H-2-propenyl)]-4, 5a -epoxy-3,14-dihydro...)
Affinity DataKi:  18.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details
PubMed
TargetOpioid receptor delta 1(Guinea pig)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50458152(CHEMBL4207167)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]Naltrindole from DOR in guinea pig brain membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetOpioid receptor delta 1(Rhesus macaque)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50458148(CHEMBL4214248)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]naltrindole from DOR in monkey brain cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetOpioid receptor delta 1(Bovine)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM50000788([17-(2,3-3H-2-propenyl)]-4, 5a -epoxy-3,14-dihydro...)
Affinity DataKi:  29.7nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details
PubMed
TargetOpioid receptor delta 1(Bovine)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM50021325(DIHYDROMORPHINE | CHEMBL1281 | 4-methyl-(1S,5R,13R...)
Affinity DataKi:  35.6nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details
PubMed
TargetOpioid receptor delta 1(Guinea pig)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50458141(CHEMBL4204304)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]Naltrindole from DOR in guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetOpioid receptor delta 1(Bovine)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM50021325(DIHYDROMORPHINE | CHEMBL1281 | 4-methyl-(1S,5R,13R...)
Affinity DataKi:  38.1nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details
PubMed
TargetOpioid receptor delta 1(Guinea pig)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50458142(CHEMBL4208635)
Affinity DataKi:  52nMAssay Description:Displacement of [3H]Naltrindole from DOR in guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetOpioid receptor delta 1(Bovine)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM81934(Beta-Endorphin)
Affinity DataKi:  58.1nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details
PubMed
TargetOpioid receptor delta 1(Bovine)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM50000092(Analog of 14-(Arylhydroxyamino)codeinone | 4-methy...)
Affinity DataKi:  63nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details
PubMed
TargetOpioid receptor delta 1(Bovine)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM50000092(Analog of 14-(Arylhydroxyamino)codeinone | 4-methy...)
Affinity DataKi:  73nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details
PubMed
TargetOpioid receptor delta 1(Bovine)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM50000092(Analog of 14-(Arylhydroxyamino)codeinone | 4-methy...)
Affinity DataKi:  147nMAssay Description: adrenals [23].More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2025
Entry Details
PubMed
TargetOpioid receptor delta 1(Bovine)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM86258(CAS_23552-18-3 | NSC_5980 | Morphine)
Affinity DataKi:  278nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2012
Entry Details Article
PubMed
TargetOpioid receptor delta 1(Bovine)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM50139013(CHEMBL333357 | (S)-N-((S)-1-((S)-1-amino-1-oxo-3-p...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in calf frontal cortex after 1 hr by gamma counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetOpioid receptor delta 1(Bovine)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM50106276(CHEMBL126243 | Endomorphin 2 | 1-[2-Amino-3-(4-hyd...)
Affinity DataKi:  500nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details
PubMed
TargetOpioid receptor delta 1(Bovine)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM86518(CAS_509-60-4 | NSC_273032 | DIHYDROMORPHINE)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2012
Entry Details Article
PubMed
TargetOpioid receptor delta 1(Bovine)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM86519(NSC_11221 | CAS_11221 | Dihydroheroin)
Affinity DataKi:  2.47E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2012
Entry Details Article
PubMed
TargetOpioid receptor delta 1(Bovine)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM86757(NSC_11603174 | CAS_0 | [11C]MMP)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2012
Entry Details Article
PubMed
TargetOpioid receptor delta 1(Bovine)
University of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM50308247(CHEMBL1215855 | ibogaine)
Affinity DataKi: >1.00E+5nMAssay Description:DPDPE cortex .More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2025
Entry Details
PubMed