Report error Found 174 Enz. Inhib. hit(s) with Target = 'NAD-dependent protein deacylase sirtuin-6'
Affinity DataKd: 2.90E+4nMAssay Description:Binding affinity to recombinant human full length SIRT6 (1 to 355 residues) expressed in Escherichia coli M15 after 20 mins in presence of ADP-ribose...More data for this Ligand-Target Pair
Affinity DataKd: 3.30E+4nMAssay Description:Binding affinity to recombinant human full length SIRT6 (1 to 355 residues) expressed in Escherichia coli M15 after 20 mins in presence of ADP-ribose...More data for this Ligand-Target Pair
Affinity DataKd: 2.27E+5nMAssay Description:Binding affinity to recombinant human full length SIRT6 (1 to 355 residues) expressed in Escherichia coli M15 after 20 mins by fluorescence-based SDS...More data for this Ligand-Target Pair
Affinity DataKd: 4.45E+5nMAssay Description:Binding affinity to recombinant human full length SIRT6 (1 to 355 residues) expressed in Escherichia coli M15 after 20 mins in presence of NAM by flu...More data for this Ligand-Target Pair
Affinity DataEC50: 2.18E+5nMAssay Description:Inhibition of SIRT6 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 5.70E+3nMAssay Description:Inhibition of SIRT6 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 1.74E+5nMAssay Description:Inhibition of SIRT6 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 1.03E+4nMAssay Description:Inhibition of SIRT6 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 3.80E+4nMAssay Description:Inhibition of sirtuin 6 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 9.76E+3nMAssay Description:Binding affinity to SIRT6 (unknown origin) by surface plasmon resonance assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.00E+4nMAssay Description:Binding affinity to SIRT6 (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataEC50: 1.03E+4nMAssay Description:Allosteric activation of SIRT6 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 3.80E+4nMAssay Description:Activation of SIRT6 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 5.35E+3nMAssay Description:Activation of N-terminal his-tagged human SIRT6 expressed in Escherichia coli M15 [pREP4] assessed as increase in peptide demyristoylation incubated ...More data for this Ligand-Target Pair
Affinity DataEC50: 8.91E+3nMAssay Description:Activation of N-terminal his-tagged human SIRT6 expressed in Escherichia coli M15 [pREP4] assessed as increase in deacetylation activity incubated fo...More data for this Ligand-Target Pair
Affinity DataEC50: 5.49E+3nMAssay Description:Activation of N-terminal his-tagged human SIRT6 expressed in Escherichia coli M15 [pREP4] assessed as increase in deacetylation activity incubated fo...More data for this Ligand-Target Pair
Affinity DataKd: 8.85E+3nMAssay Description:Binding affinity to N-terminal his-tagged human SIRT6 expressed in Escherichia coli M15 [pREP4] by ITC assayMore data for this Ligand-Target Pair
Affinity DataKd: 5.52E+3nMAssay Description:Binding affinity to N-terminal his-tagged human SIRT6 expressed in Escherichia coli M15 [pREP4] by SPR assayMore data for this Ligand-Target Pair
Affinity DataKd: 9.51E+3nMAssay Description:Binding affinity to N-terminal his-tagged human SIRT6 expressed in Escherichia coli M15 [pREP4] by SPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 7.10E+3nMAssay Description:Activation of recombinant SIRT6 (unknown origin) using fluoro substrate peptide incubated for 1 hr in presence of NAD by Fluor de Lys assay based flu...More data for this Ligand-Target Pair
Affinity DataEC50: >2.50E+5nMAssay Description:Activation of N-terminal His-tagged human SIRT6 (1 to 355 residues) expressed in Escherichia coli M15(pREP4) assessed as increase in deacetylation ac...More data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+4nMAssay Description:Activation of wild type full length human SIRT6 expressed in Escherichia coli BL21(DE3) using RHKK-ac-AMC as substrate incubated for 2 hrs in presenc...More data for this Ligand-Target Pair
Affinity DataEC50: 3.80E+4nMAssay Description:Activation of human SIRT6 using acetylated histone H3K9 as peptide substrateMore data for this Ligand-Target Pair
Affinity DataEC50: 5.70E+3nMAssay Description:Activation of wild type human N-terminal full length SIRT6 deacetylation (8 to 533 residues) expressed in Escherichia coli BL21 (DE3) expression syst...More data for this Ligand-Target Pair
Affinity DataEC50: 2.46E+5nMAssay Description:Activation of SIRT6 (unknown origin) deacetylase activity using H3K9Ac peptide substrate by reversed-phase HPLCMore data for this Ligand-Target Pair
Affinity DataEC50: 3.10E+3nMAssay Description:Activation of his6-tagged SIRT6 (unknown origin) using H3K9Ac peptide substrate incubated for 30 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 4.60E+5nMAssay Description:Activation of human SIRT6 deacetylase activity by FDL assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.03E+4nMAssay Description:Activation of SIRT6 (unknown origin) deacetylase activityMore data for this Ligand-Target Pair
Affinity DataEC50: 5.30E+3nMAssay Description:Activation of SIRT6 (unknown origin) deacetylase activityMore data for this Ligand-Target Pair
Affinity DataEC50: 3.80E+4nMAssay Description:Activation of SIRT6 (unknown origin) deacetylase activityMore data for this Ligand-Target Pair
Affinity DataEC50: 6.47E+4nMAssay Description:Activation of recombinant SIRT6 (unknown origin) deacetylase activity using fluoro peptide as substrate by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataEC50: 3.88E+4nMAssay Description:Activation of recombinant SIRT6 (unknown origin) deacetylase activity using fluoro peptide as substrate by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataEC50: 4.88E+4nMAssay Description:Activation of recombinant SIRT6 (unknown origin) deacetylase activity using fluoro peptide as substrate by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataEC50: 5.80E+4nMAssay Description:Activation of recombinant SIRT6 (unknown origin) deacetylase activity using fluoro peptide as substrate by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataEC50: 4.86E+4nMAssay Description:Activation of recombinant SIRT6 (unknown origin) deacetylase activity using fluoro peptide as substrate by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataEC50: 5.25E+4nMAssay Description:Activation of recombinant SIRT6 (unknown origin) deacetylase activity using fluoro peptide as substrate by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataEC50: 4.60E+5nMAssay Description:Activation of GST-tagged SIRT6 (unknown origin) deacetylase activity using H3K9Ac peptide substrate by HPLCMore data for this Ligand-Target Pair
Affinity DataEC50: 4.04E+5nMAssay Description:Activation of GST-tagged SIRT6 (unknown origin) deacetylase activity using H3K9Ac peptide substrate by HPLCMore data for this Ligand-Target Pair
Affinity DataEC50: 7.60E+5nMAssay Description:Activation of GST-tagged SIRT6 (unknown origin) deacetylase activity using H3K9Ac peptide substrate by HPLCMore data for this Ligand-Target Pair
Affinity DataEC50: 3.10E+3nMAssay Description:Activation of human SIRT6 deacetylase activity expressed in Escherichia coli BL21(DE3) expressed in Escherichia coli using H3K9Ac peptide substrateMore data for this Ligand-Target Pair
Affinity DataEC50: 8.90E+4nMAssay Description:Activation of human SIRT6 deacetylase activity expressed in Escherichia coli BL21(DE3) expressed in Escherichia coli using H3K9Ac peptide substrateMore data for this Ligand-Target Pair
Affinity DataEC50: 2.30E+5nMAssay Description:Activation of human SIRT6 deacetylase activity expressed in Escherichia coli BL21(DE3) expressed in Escherichia coli using H3K9Ac peptide substrateMore data for this Ligand-Target Pair
Affinity DataEC50: 2.70E+5nMAssay Description:Activation of human SIRT6 deacetylase activity expressed in Escherichia coli BL21(DE3) expressed in Escherichia coli using H3K9Ac peptide substrateMore data for this Ligand-Target Pair
Affinity DataEC50: 9.90E+5nMAssay Description:Activation of human SIRT6 deacetylase activity expressed in Escherichia coli BL21(DE3) expressed in Escherichia coli using H3K9Ac peptide substrateMore data for this Ligand-Target Pair
Affinity DataEC50: 2.46E+5nMAssay Description:Activation of recombinant His-tagged SIRT6 (unknown origin) deacetylase activity expressed in Escherichia coli using H3K9Ac peptide substrateMore data for this Ligand-Target Pair
Affinity DataEC50: 9.00E+4nMAssay Description:Activation of recombinant His-tagged SIRT6 (unknown origin) deacetylase activity expressed in Escherichia coli using H3K9Ac peptide substrateMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+5nMAssay Description:Activation of recombinant His-tagged SIRT6 (unknown origin) deacetylase activity expressed in Escherichia coli using H3K9Ac peptide substrateMore data for this Ligand-Target Pair
Affinity DataEC50: 3.10E+3nMAssay Description:Activation of recombinant His-tagged SIRT6 (unknown origin) deacetylase activity expressed in Escherichia coli using H3K9Ac peptide substrateMore data for this Ligand-Target Pair
Affinity DataEC50: 7.50E+3nMAssay Description:Activation of recombinant His-tagged SIRT6 (unknown origin) deacetylase activity expressed in Escherichia coli using H3K9Ac peptide substrateMore data for this Ligand-Target Pair
Affinity DataEC50: 3.80E+4nMAssay Description:Activation of SIRT6 (unknown origin) deacetylase activityMore data for this Ligand-Target Pair
