Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with Target = 'N-methyl-D-aspartate receptor'
TargetN-methyl-D-aspartate receptor(Pig)
Zentrum FüR Pharmaforschung

Curated by ChEMBL
LigandPNGBDBM50089759((R)-1-(4-Chloro-phenyl)-2-[4-(4-fluoro-benzyl)-pip...)
Affinity DataIC50: 50nMAssay Description:Displacement of [3H]ifendropil from binding site of N-methyl-D-aspartate glutamate receptor was evaluated employing synaptosomal fraction of porcine ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetN-methyl-D-aspartate receptor(Pig)
Zentrum FüR Pharmaforschung

Curated by ChEMBL
LigandPNGBDBM50079387(CHEMBL28564 | 1-(4-Chloro-phenyl)-2-[4-(4-fluoro-b...)
Affinity DataIC50: 83nMAssay Description:Displacement of [3H]ifendropil from binding site of N-methyl-D-aspartate glutamate receptor was evaluated employing synaptosomal fraction of porcine ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetN-methyl-D-aspartate receptor(Pig)
Zentrum FüR Pharmaforschung

Curated by ChEMBL
LigandPNGBDBM50089759((R)-1-(4-Chloro-phenyl)-2-[4-(4-fluoro-benzyl)-pip...)
Affinity DataIC50: 213nMAssay Description:Compound was tested for inhibition of [3H]MK-801 binding to N-methyl-D-aspartate glutamate receptor at NR2B subunit in high affinity fraction of porc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetN-methyl-D-aspartate receptor(Pig)
Zentrum FüR Pharmaforschung

Curated by ChEMBL
LigandPNGBDBM50079387(CHEMBL28564 | 1-(4-Chloro-phenyl)-2-[4-(4-fluoro-b...)
Affinity DataIC50: 277nMAssay Description:Compound was tested for inhibition of [3H]MK-801 binding to N-methyl-D-aspartate glutamate receptor at NR2B subunit in high affinity fraction of porc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetN-methyl-D-aspartate receptor(Pig)
Zentrum FüR Pharmaforschung

Curated by ChEMBL
LigandPNGBDBM50089760((S)-1-(4-Chloro-phenyl)-2-[4-(4-fluoro-benzyl)-pip...)
Affinity DataIC50: 545nMAssay Description:Displacement of [3H]ifendropil from binding site of N-methyl-D-aspartate glutamate receptor was evaluated employing synaptosomal fraction of porcine ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetN-methyl-D-aspartate receptor(Pig)
Zentrum FüR Pharmaforschung

Curated by ChEMBL
LigandPNGBDBM50089760((S)-1-(4-Chloro-phenyl)-2-[4-(4-fluoro-benzyl)-pip...)
Affinity DataIC50: 5.10E+3nMAssay Description:Compound was tested for inhibition of [3H]MK-801 binding to N-methyl-D-aspartate glutamate receptor lacking NR2B subunit in low affinity fraction of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetN-methyl-D-aspartate receptor(Pig)
Zentrum FüR Pharmaforschung

Curated by ChEMBL
LigandPNGBDBM50089760((S)-1-(4-Chloro-phenyl)-2-[4-(4-fluoro-benzyl)-pip...)
Affinity DataIC50: 5.10E+3nMAssay Description:Compound was tested for inhibition of [3H]MK-801 binding to N-methyl-D-aspartate glutamate receptor at NR2B subunit in high affinity fraction of porc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetN-methyl-D-aspartate receptor(Pig)
Zentrum FüR Pharmaforschung

Curated by ChEMBL
LigandPNGBDBM50079387(CHEMBL28564 | 1-(4-Chloro-phenyl)-2-[4-(4-fluoro-b...)
Affinity DataIC50: 1.13E+4nMAssay Description:Compound was tested for inhibition of [3H]MK-801 binding to N-methyl-D-aspartate glutamate receptor lacking NR2B subunit in low affinity fraction of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetN-methyl-D-aspartate receptor(Pig)
Zentrum FüR Pharmaforschung

Curated by ChEMBL
LigandPNGBDBM50089759((R)-1-(4-Chloro-phenyl)-2-[4-(4-fluoro-benzyl)-pip...)
Affinity DataIC50: 2.37E+4nMAssay Description:Compound was tested for inhibition of [3H]MK-801 binding to N-methyl-D-aspartate glutamate receptor lacking NR2B subunit in low affinity fraction of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed