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Report error Found 1345 Enz. Inhib. hit(s) with Target = 'Methionine aminopeptidase 2'
LigandPNGBDBM17451(5-(4-methylphenyl)-1H-pyrazole | pyrazole analogue...)
Affinity DatapH: 7.5 T: 2°CAssay Description:MetAP2 activity was monitored by measuring the initial velocity of turnover of the artificial substrate Met-AMC. Assays were performed in 96-well mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2007
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Mouse)
Massachusetts Institute of Technology

LigandPNGBDBM36588(AGM-1470)
Affinity DataEC50:  0.0370nMpH: 7.5Assay Description:Proliferation assay using bovine aortic endothelial cell (BAEC) line.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2011
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Mouse)
Massachusetts Institute of Technology

LigandPNGBDBM36589(Ovalicin)
Affinity DataEC50:  0.0180nMpH: 7.5Assay Description:Proliferation assay using bovine aortic endothelial cell (BAEC) line.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2011
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Mouse)
Massachusetts Institute of Technology

LigandPNGBDBM36590(FOS-72)
Affinity DataEC50:  0.0130nMpH: 7.5Assay Description:Proliferation assay using bovine aortic endothelial cell (BAEC) line.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2011
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Mouse)
Massachusetts Institute of Technology

LigandPNGBDBM36595(FOS-68)
Affinity DataEC50:  0.460nMpH: 7.5Assay Description:Proliferation assay using bovine aortic endothelial cell (BAEC) line.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2011
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Mouse)
Massachusetts Institute of Technology

LigandPNGBDBM36597(FOS-69)
Affinity DataEC50:  0.310nMpH: 7.5Assay Description:Proliferation assay using bovine aortic endothelial cell (BAEC) line.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2011
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Mouse)
Massachusetts Institute of Technology

LigandPNGBDBM36592(FOS-70)
Affinity DataEC50:  0.120nMpH: 7.5Assay Description:Proliferation assay using bovine aortic endothelial cell (BAEC) line.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2011
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Mouse)
Massachusetts Institute of Technology

LigandPNGBDBM36591(FOS-37)
Affinity DataEC50:  9.5nMpH: 7.5Assay Description:Proliferation assay using bovine aortic endothelial cell (BAEC) line.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2011
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Mouse)
Massachusetts Institute of Technology

LigandPNGBDBM36596(FOS-34)
Affinity DataEC50:  2.20nMpH: 7.5Assay Description:Proliferation assay using bovine aortic endothelial cell (BAEC) line.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2011
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Mouse)
Massachusetts Institute of Technology

LigandPNGBDBM36593(FOS-64)
Affinity DataEC50:  110nMpH: 7.5Assay Description:Proliferation assay using bovine aortic endothelial cell (BAEC) line.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2011
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Mouse)
Massachusetts Institute of Technology

LigandPNGBDBM36598(FOS-67)
Affinity DataEC50:  40nMpH: 7.5Assay Description:Proliferation assay using bovine aortic endothelial cell (BAEC) line.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2011
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Mouse)
Massachusetts Institute of Technology

LigandPNGBDBM36599(FOS-201)
Affinity DataEC50:  56nMpH: 7.5Assay Description:Proliferation assay using bovine aortic endothelial cell (BAEC) line.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2011
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Mouse)
Massachusetts Institute of Technology

LigandPNGBDBM36594(FOS-202)
Affinity DataEC50:  2.80E+3nMpH: 7.5Assay Description:Proliferation assay using bovine aortic endothelial cell (BAEC) line.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2011
Entry Details Article
PubMed
LigandPNGBDBM50433373(CHEMBL2375609)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of human methionine aminopeptidase 2 in presence of Mn2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
LigandPNGBDBM50433374(CHEMBL2375610)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of human methionine aminopeptidase 2 in presence of Mn2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
LigandPNGBDBM50433378(CHEMBL2375629)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of human methionine aminopeptidase 2 in presence of Mn2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
LigandPNGBDBM47468(N-(2-phenylethyl)-2-(2-pyridinyl)-4-quinazolinamin...)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of human methionine aminopeptidase 2 in presence of Mn2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
LigandPNGBDBM50433379(CHEMBL2375611)
Affinity DataEC50: >3.00E+5nMAssay Description:Inhibition of human methionine aminopeptidase 2 in presence of Mn2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
LigandPNGBDBM50433380(CHEMBL2375612)
Affinity DataEC50: >3.00E+5nMAssay Description:Inhibition of human methionine aminopeptidase 2 in presence of Mn2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
LigandPNGBDBM50433381(CHEMBL2375613)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of human methionine aminopeptidase 2 in presence of Mn2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
LigandPNGBDBM50433382(CHEMBL1329554)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of human methionine aminopeptidase 2 in presence of Mn2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
LigandPNGBDBM50433383(CHEMBL2375614)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of human methionine aminopeptidase 2 in presence of Mn2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
LigandPNGBDBM50433384(CHEMBL45721)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of human methionine aminopeptidase 2 in presence of Mn2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
LigandPNGBDBM50433385(CHEMBL49678)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of human methionine aminopeptidase 2 in presence of Mn2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
LigandPNGBDBM50433386(CHEMBL2375615)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of human methionine aminopeptidase 2 in presence of Mn2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
LigandPNGBDBM50433387(CHEMBL2375616)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of human methionine aminopeptidase 2 in presence of Mn2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
LigandPNGBDBM50433388(CHEMBL2375617)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of human methionine aminopeptidase 2 in presence of Mn2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
LigandPNGBDBM50433389(CHEMBL2375618)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of human methionine aminopeptidase 2 in presence of Mn2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
LigandPNGBDBM50433390(CHEMBL2375619)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of human methionine aminopeptidase 2 in presence of Mn2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
LigandPNGBDBM50433391(CHEMBL2375620)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of human methionine aminopeptidase 2 in presence of Mn2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
LigandPNGBDBM50433392(CHEMBL2375621)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of human methionine aminopeptidase 2 in presence of Mn2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
LigandPNGBDBM50433393(CHEMBL2375622)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of human methionine aminopeptidase 2 in presence of Mn2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
LigandPNGBDBM50433394(CHEMBL2375623)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of human methionine aminopeptidase 2 in presence of Mn2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
LigandPNGBDBM50433395(CHEMBL2375624)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of human methionine aminopeptidase 2 in presence of Mn2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
LigandPNGBDBM50433396(CHEMBL2375625)
Affinity DataEC50: >2.00E+5nMAssay Description:Inhibition of human methionine aminopeptidase 2 in presence of Mn2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
LigandPNGBDBM50433397(CHEMBL2375626)
Affinity DataEC50: >2.00E+5nMAssay Description:Inhibition of human methionine aminopeptidase 2 in presence of Mn2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
LigandPNGBDBM50433398(CHEMBL2375607)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of human methionine aminopeptidase 2 in presence of Mn2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
LigandPNGBDBM50433399(CHEMBL2375608)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of human methionine aminopeptidase 2 in presence of Mn2+More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
LigandPNGBDBM401307(US10005756, Compound A78)
Affinity DataKd:  0.880nMAssay Description:Inhibition of 5-[(S)-3-(3-Chloro-5-fluoro-benzylcarbamoyl)-3-hydroxy-2-oxopyrrolidin-1-yl]-1H-indole-2-carboxylic Acid (3-Amino-propyl)-amide-Dy647 b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
LigandPNGBDBM401307(US10005756, Compound A78)
Affinity DataKd:  0.880nMAssay Description:Inhibition of 5-[(S)-3-(3-Chloro-5-fluoro-benzylcarbamoyl)-3-hydroxy-2-oxopyrrolidin-1-yl]-1H-indole-2-carboxylic Acid (3-Amino-propyl)-amide-Dy647 b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
LigandPNGBDBM50531163(CHEMBL4464946)
Affinity DataKd:  2.10nMAssay Description:Inhibition of 5-[(S)-3-(3-Chloro-5-fluoro-benzylcarbamoyl)-3-hydroxy-2-oxopyrrolidin-1-yl]-1H-indole-2-carboxylic Acid (3-Amino-propyl)-amide-Dy647 b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
LigandPNGBDBM50531161(CHEMBL4448724)
Affinity DataKd:  1.10nMAssay Description:Inhibition of 5-[(S)-3-(3-Chloro-5-fluoro-benzylcarbamoyl)-3-hydroxy-2-oxopyrrolidin-1-yl]-1H-indole-2-carboxylic Acid (3-Amino-propyl)-amide-Dy647 b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
LigandPNGBDBM50531163(CHEMBL4464946)
Affinity DataKd:  2.10nMAssay Description:Inhibition of 5-[(S)-3-(3-Chloro-5-fluoro-benzylcarbamoyl)-3-hydroxy-2-oxopyrrolidin-1-yl]-1H-indole-2-carboxylic Acid (3-Amino-propyl)-amide-Dy647 b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
LigandPNGBDBM50531161(CHEMBL4448724)
Affinity DataKd:  1.10nMAssay Description:Inhibition of 5-[(S)-3-(3-Chloro-5-fluoro-benzylcarbamoyl)-3-hydroxy-2-oxopyrrolidin-1-yl]-1H-indole-2-carboxylic Acid (3-Amino-propyl)-amide-Dy647 b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
LigandPNGBDBM36597(FOS-69)
Affinity DataIC50: 0.100nMpH: 7.35 T: 2°CAssay Description:Enzymatic assay using recombinant human type 2 methionine aminopeptidase (MetAP2).More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2011
Entry Details Article
PubMed
LigandPNGBDBM50137405(Carbamic acid (3R,4S,5S,6R)-5-methoxy-4-[(2R,3R)-2...)
Affinity DataIC50: 0.390nMAssay Description:Inhibitory activity against Methionine aminopeptidase 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2012
Entry Details Article
PubMed
LigandPNGBDBM36589(Ovalicin)
Affinity DataIC50: 0.400nMpH: 7.35 T: 2°CAssay Description:Enzymatic assay using recombinant human type 2 methionine aminopeptidase (MetAP2).More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2011
Entry Details Article
PubMed
LigandPNGBDBM50295172(4-Hydroxy-5-methoxy-4-[(2S,3R)-2-methyl-3-(3-methy...)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of methionine aminopeptidase 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
LigandPNGBDBM50137403(Acetyl-carbamic acid (3R,4S,5S,6R)-5-methoxy-4-[(R...)
Affinity DataIC50: 0.430nMAssay Description:Inhibitory activity against Methionine aminopeptidase 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2012
Entry Details Article
PubMed
LigandPNGBDBM50137404(Acetic acid (3R,4S,5S,6R)-5-methoxy-4-[(2R,3R)-2-m...)
Affinity DataIC50: 0.510nMAssay Description:Inhibitory activity against Methionine aminopeptidase 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2012
Entry Details Article
PubMed
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