Compile Data Set for Download or QSAR
Report error Found 1016 Enz. Inhib. hit(s) with Target = 'Menin'
TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM50366388(NEOMYCIN A | NEOMYCIN)
Affinity DataKd:  1.56E+4nMAssay Description:Binding affinity to menin (unknown origin) by isothermal titration calorimetry analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2015
Entry Details Article
PubMed
TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM50156121(CHEMBL3780497)
Affinity DataKd:  24nMAssay Description:Binding affinity to menin (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM50156122(CHEMBL3781030)
Affinity DataKd:  6.5nMAssay Description:Binding affinity to menin (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM50455873(CHEMBL4216801)
Affinity DataKd:  9nMAssay Description:Binding affinity to human C-terminal Avi-tagged menin expressed in Escherichia coli BL21 (DE3) cells by bio-layer interferometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM50455876(CHEMBL4217916)
Affinity DataKd:  24nMAssay Description:Binding affinity to human C-terminal Avi-tagged menin expressed in Escherichia coli BL21 (DE3) cells by bio-layer interferometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM152235(US8993552, 70)
Affinity DataKd:  158nMAssay Description:Binding affinity to menin (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM50454122(CHEMBL4206413)
Affinity DataKd:  22nMAssay Description:Binding affinity to menin (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM50454124(CHEMBL3780822)
Affinity DataKd:  9.30nMAssay Description:Binding affinity to menin (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM50496327(CHEMBL3126198)
Affinity DataKd:  85nMAssay Description:Binding affinity to human menin by isothermal titration calorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM50496328(CHEMBL3126187)
Affinity DataKd:  285nMAssay Description:Binding affinity to human menin by isothermal titration calorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM50496340(CHEMBL3124953)
Affinity DataKd:  952nMAssay Description:Binding affinity to human menin by isothermal titration calorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM50489222(CHEMBL2314822)
Affinity DataKd:  1.40nMAssay Description:Binding affinity to menin (unknown origin) after 60 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM50489223(CHEMBL2314821)
Affinity DataKd:  16nMAssay Description:Binding affinity to menin (unknown origin) after 60 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM50454124(CHEMBL3780822)
Affinity DataKd:  10nMAssay Description:Binding affinity to human Menin expressed in Escherichia coli Rosetta2 (DE3) cells by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM50156122(CHEMBL3781030)
Affinity DataKd:  10nMAssay Description:Binding affinity to human Menin expressed in Escherichia coli Rosetta2 (DE3) cells by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM50455873(CHEMBL4216801)
Affinity DataKd:  10nMAssay Description:Binding affinity to human Menin expressed in Escherichia coli Rosetta2 (DE3) cells by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM50496346(CHEMBL3126196)
Affinity DataKd:  1.10E+5nMAssay Description:Binding affinity to biotinylated Menin (unknown origin) by biolayer interferometry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM50516582(CHEMBL4449381)
Affinity DataKd:  1.40E+3nMAssay Description:Binding affinity to biotinylated Menin (unknown origin) by biolayer interferometry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM50455859(CHEMBL3780895)
Affinity DataKd:  10nMAssay Description:Binding affinity to human Menin expressed in Escherichia coli Rosetta2 (DE3) cells by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM50540837(CHEMBL4647785)
Affinity DataKd:  82nMAssay Description:Binding affinity to human Menin expressed in Escherichia coli BL21 (DE3) assessed as inhibition of Menin/MLL1 protein-protein at 20 degree C by isoth...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM742411(4-methyl-1-[(2S)-5- oxomorpholin-2- (trifluorometh...)
Affinity DataEC50: <75nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM742412(4-methyl-1-[(3-oxo- 1,4-oxazepan-7- yl)methyl]-5- ...)
Affinity DataEC50: <75nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM742413(4-methyl-1-[2-(2- oxoimidazolidin- 1-yl)ethyl]- 5-...)
Affinity DataEC50: <75nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM742414(4-methyl-1-[(2- oxohexahydro- pyrimidin-5- yl)meth...)
Affinity DataEC50: <75nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM742415(4-methyl-1-[(7- oxoazepan-4-yl) methyl]-5-[[2- [6-...)
Affinity DataEC50: <75nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM742416(4-methyl-1-[(2- oxoimidazolidin- 4-yl)methyl]- 5-[...)
Affinity DataEC50:  3.00E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM742417(4-methyl-1-[(6-methyl- 5-oxo-morpholin-2- yl)methy...)
Affinity DataEC50: <75nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM742418(4-methyl-1- [(4-methyl- sulfonylmorpholin-2- yl)me...)
Affinity DataEC50:  288nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM742419(5-[[2-[5-fluoro- 6-(2,2,2- trifluoroethyl) quinazo...)
Affinity DataEC50: <75nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM742420(4-methyl-1- [1-methyl-3-(4- methylsulfonyl- pipera...)
Affinity DataEC50: <75nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM742421(4-methyl-1-[(6- oxo-1H-pyridin-3- yl)methyl]- 5-[[...)
Affinity DataEC50: <75nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM742422(4-methyl-1-[(4- methyl-5-oxo- morpholin-2- yl)meth...)
Affinity DataEC50: <75nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM742423(4-methyl-1-[(4- methyl-3,3-dioxo-1,3,4- oxathiazin...)
Affinity DataEC50: <75nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM742424(1-[2-(4-butyl- sulfonyl- piperazin-1- yl)propyl]-4...)
Affinity DataEC50: <75nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM742425(1-[2-(4-cyclopropyl- sulfonylpiperazin-1- yl)propy...)
Affinity DataEC50: <75nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM742426(6-methoxy-1- [2-(4-methyl- sulfonylpiperazin-1- yl...)
Affinity DataEC50: <75nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM742427(1-[(3,3-dioxo-1,3,4- oxathiazinan- 6-yl)methyl]- 4...)
Affinity DataEC50: <75nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM742428(4-methyl-1-[(2-oxo-4- piperidyl) methyl]-5-[[2- [6...)
Affinity DataEC50: <75nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM742429(4-methyl-1-[(1R)- 1-methyl-2-(4- methylsulfonyl- p...)
Affinity DataEC50: <75nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM742430(4-methyl-1-[(1S)- 1-methyl-2-(4- methylsulfonyl- p...)
Affinity DataEC50: <75nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM742431(1-[(2R)-2-[(3S)-4- ethylsulfonyl-3-methyl- piperaz...)
Affinity DataEC50: <75nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM742432(1-[(2S)-2-[(3S)-4- ethylsulfonyl-3-methyl- piperaz...)
Affinity DataEC50: <75nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM742433(4-methyl-1-[(2R)-2- [(3S)-3-methyl-4- methylsulfon...)
Affinity DataEC50: <75nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM742434(4-methyl-1-[(2S)-2- [(3S)-3-methyl-4- methylsulfon...)
Affinity DataEC50: <75nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM742435(4-methyl-1-[2-(4-methyl- sulfonyl-1,4-diazepan- 1-...)
Affinity DataEC50: <75nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM742436(5-[[2-[7-fluoro- 6-(2,2,2- trifluoroethyl) quinazo...)
Affinity DataEC50: <75nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM742437(1-[(4-isobutyl-5-oxo- morpholin-2-yl) methyl]- 4-m...)
Affinity DataEC50:  288nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM742438(N-(1R,4R)-[4-[2-cyano- 4-methyl-5-[[2-[6- (2,2,2-t...)
Affinity DataEC50: <75nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM742439(N-(1R,4R)- [4-[[2-cyano- 4-methyl-5-[[2-[6- (2,2,2...)
Affinity DataEC50:  288nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetMenin(Human)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM742440(4-methyl-1- [2-(4-methyl- sulfonylpiperazin-1- yl)...)
Affinity DataEC50: <75nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

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