Compile Data Set for Download or QSAR
Report error Found 42 Enz. Inhib. hit(s) with Target = 'Isoform TrkA-I of High affinity nerve growth factor receptor (TrkAI)'
LigandPNGBDBM204852(US9242977, 85-226)
Affinity DataIC50: 1nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204849(US9242977, 85-184)
Affinity DataIC50: 2nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204848(US9242977, 85-117)
Affinity DataIC50: 2nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204842(US9242977, 71)
Affinity DataIC50: 2nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204837(US9242977, 65-1)
Affinity DataIC50: 2nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204835(US9242977, 57)
Affinity DataIC50: 3nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204830(US9242977, 23)
Affinity DataIC50: 4nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204850(US9242977, 85-209)
Affinity DataIC50: 4nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204851(US9242977, 85-225)
Affinity DataIC50: 4nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204838(US9242977, 66-19)
Affinity DataIC50: 4nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204834(US9242977, 54)
Affinity DataIC50: 4nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204831(US9242977, 34)
Affinity DataIC50: 6nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204839(US9242977, 66-27)
Affinity DataIC50: 10nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204832(US9242977, 48)
Affinity DataIC50: 10nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204843(US9242977, 72-1)
Affinity DataIC50: 11nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204833(US9242977, 50)
Affinity DataIC50: 12nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204840(US9242977, 66-28)
Affinity DataIC50: 14nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204844(US9242977, 72-3)
Affinity DataIC50: 18nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204848(US9242977, 85-117)
Affinity DataIC50: 20nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204838(US9242977, 66-19)
Affinity DataIC50: 20nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204835(US9242977, 57)
Affinity DataIC50: 30nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204845(US9242977, 72-7)
Affinity DataIC50: 30nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204842(US9242977, 71)
Affinity DataIC50: 30nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204841(US9242977, 66-72)
Affinity DataIC50: 32nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204845(US9242977, 72-7)
Affinity DataIC50: 33nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204834(US9242977, 54)
Affinity DataIC50: 40nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204833(US9242977, 50)
Affinity DataIC50: 40nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204841(US9242977, 66-72)
Affinity DataIC50: 50nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204843(US9242977, 72-1)
Affinity DataIC50: 50nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204844(US9242977, 72-3)
Affinity DataIC50: 60nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204836(US9242977, 59)
Affinity DataIC50: 70nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204846(US9242977, 80-2)
Affinity DataIC50: 70nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204837(US9242977, 65-1)
Affinity DataIC50: 80nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204840(US9242977, 66-28)
Affinity DataIC50: 80nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204847(US9242977, 84-41)
Affinity DataIC50: 90nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204830(US9242977, 23)
Affinity DataIC50: 90nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204829(US9242977, 9)
Affinity DataIC50: 93nMAssay Description:TrkA kinase-inhibiting activity in cell systems was measured using CHO-K1 cells expressing human TrkA and NFAT-bla (CellSenser TrkA-NFAT-bla CHO-K1 c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204832(US9242977, 48)
Affinity DataIC50: 120nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204839(US9242977, 66-27)
Affinity DataIC50: 130nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204829(US9242977, 9)
Affinity DataIC50: 160nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204831(US9242977, 34)
Affinity DataIC50: 180nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
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LigandPNGBDBM204836(US9242977, 59)
Affinity DataIC50: 190nMpH: 7.5Assay Description:TrkA-inhibiting activity was measured according to the following method using LanthaScreen kinase assay reagents (Invitrogen; Fluorescein-Poly GT, La...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2016
Entry Details
Go to US Patent