Compile Data Set for Download or QSAR
Report error Found 116 Enz. Inhib. hit(s) with Target = 'Histone lysine demethylase PHF8'
TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276044BDBM276044(2-[1-[2-(2-chlorophenyl)ethyl]imidazol-4-yl]-4-(1H...)
Affinity DataIC50: 100nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276050BDBM276050(2-[1-(3,4-dihydro-2H-chromen-4-ylmethyl)imidazol-4...)
Affinity DataIC50: 100nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276067BDBM276067(2-[1-[(3-chloro-2-fluorophenyl)methyl]imidazol-4-y...)
Affinity DataIC50: 100nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 50155449BDBM50155449(CHEMBL3780958)
Affinity DataIC50: 250nMAssay Description:Inhibition of human PHF8 preincubated for 10 mins followed by substrate addition by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2017
Entry Details Article
PubMed
TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 50155505BDBM50155505(CHEMBL3781414)
Affinity DataIC50: 250nMAssay Description:Inhibition of human PHF8 preincubated for 10 mins followed by substrate addition by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2017
Entry Details Article
PubMed
TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 50155507BDBM50155507(CHEMBL3780904)
Affinity DataIC50: 250nMAssay Description:Inhibition of human PHF8 preincubated for 10 mins followed by substrate addition by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2017
Entry Details Article
PubMed
TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 50155450BDBM50155450(CHEMBL3779953)
Affinity DataIC50: 250nMAssay Description:Inhibition of human PHF8 preincubated for 10 mins followed by substrate addition by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2017
Entry Details Article
PubMed
TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 50155509BDBM50155509(CHEMBL3780689)
Affinity DataIC50: 250nMAssay Description:Inhibition of human PHF8 preincubated for 10 mins followed by substrate addition by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2017
Entry Details Article
PubMed
TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 50155508BDBM50155508(CHEMBL3780833)
Affinity DataIC50: 250nMAssay Description:Inhibition of human PHF8 preincubated for 10 mins followed by substrate addition by AlphaLISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/10/2017
Entry Details Article
PubMed
TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276058BDBM276058(2-[1-[(2,3-dichlorophenyl)methyl]imidazol-4-yl]-4-...)
Affinity DataIC50: 300nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 50395083BDBM50395083(CHEMBL2164246)
Affinity DataIC50: 480nMAssay Description:Inhibition of human PHF8 expressed in Escherichia coli using methyl lysine peptide substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276057BDBM276057(2-[1-[(2,3-dichlorophenyl)methyl]imidazol-4-yl]-4-...)
Affinity DataIC50: 550nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276059BDBM276059(2-[1-[(2,3-dichlorophenyl)methyl]imidazol-4-yl]-4-...)
Affinity DataIC50: 550nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276053BDBM276053(4-[2-[1-(1,2,3,4-tetrahydronaphthalen-1-ylmethyl)i...)
Affinity DataIC50: 550nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276082BDBM276082(1-benzyl-4-{1H-[1,2,3]triazolo[4,5-c]pyridin-6-yl}...)
Affinity DataIC50: 550nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276054BDBM276054(4-[2-[1-(2-naphthalen-1-ylethyl)imidazol-4-yl]pyri...)
Affinity DataIC50: 550nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276039BDBM276039(2-(1-methylimidazol-4-yl)-4-(1H-triazol-4-yl)pyrid...)
Affinity DataIC50: 550nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276093BDBM276093(2-(5-bromo-1-(2-chlorobenzyl)-1H-imidazol-4-yl)-4-...)
Affinity DataIC50: 550nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276060BDBM276060(2-[1-[[2-chloro-3-(trifluoromethyl)phenyl]methyl]i...)
Affinity DataIC50: 550nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276062BDBM276062(2-[5-(4-fluoro-3-methoxyphenyl)-1-methylimidazol-4...)
Affinity DataIC50: 550nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276061BDBM276061(2-[1-(2-naphthalen-1-ylethyl)imidazol-4-yl]-4-(1H-...)
Affinity DataIC50: 550nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276043BDBM276043(2-[1-(1-phenylethyl)imidazol-4-yl]-4-(1H-triazol-4...)
Affinity DataIC50: 550nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276070BDBM276070(2-[1-[2-(2-chlorophenyl)-2-methylpropyl]imidazol-4...)
Affinity DataIC50: 550nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 50395076BDBM50395076(CHEMBL2164243)
Affinity DataIC50: 550nMAssay Description:Inhibition of human PHF8 expressed in Escherichia coli using methyl lysine peptide substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276073BDBM276073(4-(5-fluoro-1H-triazol-4-yl)-2-[1-(2-naphthalen-1-...)
Affinity DataIC50: 550nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276072BDBM276072(4-(1H-triazol-4-yl)-2-[1-[2-[2-(trifluoromethoxy)p...)
Affinity DataIC50: 550nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276040BDBM276040(2-[1-[(2-chlorophenyl)methyl]imidazol-4-yl]-4-(1H-...)
Affinity DataIC50: 550nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276066BDBM276066(2-[1-[(2-fluoro-3-methylphenyl)methyl]imidazol-4-y...)
Affinity DataIC50: 550nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276069BDBM276069(4-(1H-triazol-4-yl)-2-[1-[2-[2-(trifluoromethyl)ph...)
Affinity DataIC50: 550nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276041BDBM276041(2-[5-(4-fluorophenyl)-1-methylimidazol-4-yl]-4-(1H...)
Affinity DataIC50: 550nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276068BDBM276068(2-[1-[(2-fluoro-3-methoxyphenyl)methyl]imidazol-4-...)
Affinity DataIC50: 550nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276049BDBM276049(2-[1-[2-[2-(cyclopropylmethoxy)phenyl]ethyl]imidaz...)
Affinity DataIC50: 550nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276048BDBM276048(4-(1H-triazol-4-yl)-2-[1-[2-[2-(2,2,2-trifluoroeth...)
Affinity DataIC50: 550nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276046BDBM276046(2-[1-(1,2,3,4-tetrahydronaphthalen-1-ylmethyl)imid...)
Affinity DataIC50: 550nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276045BDBM276045(2-[1-[2-(2-methoxyphenyl)ethyl]imidazol-4-yl]-4-(1...)
Affinity DataIC50: 550nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276047BDBM276047(2-[1-[2-(2-ethoxyphenyl)ethyl]imidazol-4-yl]-4-(1H...)
Affinity DataIC50: 550nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 50273472BDBM50273472(CHEMBL4126235)
Affinity DataIC50: 1.70E+3nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7B (PHD) (unknown origin) preincubated for 15 mins followed by p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2020
Entry Details Article
PubMed
TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 50129197BDBM50129197(N-Hydroxy-succinamic acid | 4-(Hydroxyamino)-4-oxo...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human PHF8 expressed in Escherichia coli using methyl lysine peptide substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 50197063BDBM50197063(succinylacetone | 4,6-dioxoheptanoic acid | CHEMBL...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of human PHF8 expressed in Escherichia coli using methyl lysine peptide substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 50395078BDBM50395078(CHEMBL2164245)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of human PHF8 expressed in Escherichia coli using methyl lysine peptide substrate by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 293660BDBM293660(3-({[(1S)-6-[methyl(phenyl)amino]-1,2,3,4-tetrahyd...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of PHF8 (unknown origin) using biotinylated H3K9me1 peptide and alpha-ketoglutarate as substrate measured after 20 mins by LANCE TR-FRET a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 50483927BDBM50483927(CHEMBL3183531)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of PHF8 (1 to 1024 residues)(unknown origin) by Alphalisa assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276085BDBM276085(1-[(4-chlorophenyl)methyl]-4-{1H-[1,2,3]triazolo[4...)
Affinity DataIC50: 5.50E+3nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276071BDBM276071(2-[1-(1-phenylpropan-2-yl)imidazol-4-yl]-4-(1H-tri...)
Affinity DataIC50: 5.50E+3nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276056BDBM276056(2-[1-[2-(2-phenoxyphenyl)ethyl]imidazol-4-yl]-4-(1...)
Affinity DataIC50: 5.50E+3nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276086BDBM276086(1-[(3,4-dichlorophenyl)methyl]-4-{1H-[1,2,3]triazo...)
Affinity DataIC50: 5.50E+3nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276052BDBM276052(4-[2-[1-[(2,3-dichlorophenyl)methyl]imidazol-4-yl]...)
Affinity DataIC50: 5.50E+3nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276084BDBM276084(1-[(3-chlorophenyl)methyl]-4-{1H-[1,2,3]triazolo[4...)
Affinity DataIC50: 5.50E+3nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276042BDBM276042(2-[5-[2-(cyclopropylmethoxy)-4-fluorophenyl]-1-met...)
Affinity DataIC50: 5.50E+3nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

TargetHistone lysine demethylase PHF8(Human)
Celgene Quanticel Research

US Patent
LigandChemical structure of BindingDB Monomer ID 276055BDBM276055(2-[1-[2-(2-phenylmethoxyphenyl)ethyl]imidazol-4-yl...)
Affinity DataIC50: 5.50E+3nMAssay Description:PHF8 Assay: The ability of test compounds to inhibit the activity of PHF8 was determined in 384-well plate format under the following reaction condit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2020
Entry Details
US Patent

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