Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with Target = 'Histone deacetylase 6 [60-420]'
TargetHistone deacetylase 6 [60-420](Zebrafish)
University of Pennsylvania

LigandPNGBDBM198125(fl-SAHA)
Affinity DataKd:  1.60E+3nMT: 2°CAssay Description:The fluorescence anisotropy assay was performed with fluorescein-labeled SAHA (fl-SAHA, gift of C. Fierke, University of Michigan) and measured using...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2016
Entry Details Article
PubMed
TargetHistone deacetylase 6 [60-420](Zebrafish)
University of Pennsylvania

LigandPNGBDBM198120(TSA)
Affinity DataKi:  4.80nM ΔG°:  -47.5kJ/mole IC50: 7nMT: 2°CAssay Description:The fluorescence anisotropy assay was performed with fluorescein-labeled SAHA (fl-SAHA, gift of C. Fierke, University of Michigan) and measured using...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2016
Entry Details Article
PubMed