Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with Target = 'Histone acetyltransferase type B catalytic subunit'
TargetHistone acetyltransferase type B catalytic subunit(Homo sapiens)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50632831(CHEMBL5406943)
Affinity DataKd:  5.20E+3nMAssay Description:Binding affinity to CM5 sensor chip immobilized C-terminal FLAG tagged full length human HAT1/Rbap46 assessed as dissociation constant by SPR analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetHistone acetyltransferase type B catalytic subunit(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50562210(CHEMBL4754158)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of HAT1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetHistone acetyltransferase type B catalytic subunit(Homo sapiens)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50632831(CHEMBL5406943)
Affinity DataIC50: 1.48E+4nMAssay Description:Inhibition of C-terminal FLAG tagged full length human HAT1/Rbap46 transfected in HEK293F cells using histone H4 peptide as substrate and 4-pentynoyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetHistone acetyltransferase type B catalytic subunit(Homo sapiens)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50632830(CHEMBL1325863)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of C-terminal FLAG tagged full length human HAT1/Rbap46 transfected in HEK293F cells using histone H4 peptide as substrate and 4-pentynoyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetHistone acetyltransferase type B catalytic subunit(Homo sapiens)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50632831(CHEMBL5406943)
Affinity DataIC50: 1.91E+4nMAssay Description:Inhibition of C-terminal FLAG tagged full length human HAT1/Rbap46 transfected in HEK293F cells using histone H4 peptide as substrate and acetyl-CoA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetHistone acetyltransferase type B catalytic subunit(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50506380(CHEMBL4587968 | US20240122941, Compound 15)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of HAT1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetHistone acetyltransferase type B catalytic subunit(Homo sapiens)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50362895(Lactoflavin | RIBOFLAVIN)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of C-terminal FLAG tagged full length human HAT1/Rbap46 transfected in HEK293F cells using histone H4 peptide as substrate and 4-pentynoyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed