Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with Target = 'Gonadotropin releasing hormone receptor'
TargetGonadotropin releasing hormone receptor(Crab-eating macaque)
Shanghai Hengrui Pharmaceutical

US Patent
LigandPNGBDBM405272(US10344034, Example 9 | 1-(4-(7-(2,6-difluorobenzy...)
Affinity DataIC50: 23.2nMAssay Description:Monkey: This assay was used to determine the inhibition effect of the present compounds on the activity of monkey GnRHr protein expressed by monkey G...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2020
Entry Details
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TargetGonadotropin releasing hormone receptor(Crab-eating macaque)
Shanghai Hengrui Pharmaceutical

US Patent
LigandPNGBDBM405274(US10344034, Example 11 | 1-(4-(7-(2,6-difluorobenz...)
Affinity DataIC50: 78.6nMAssay Description:Monkey: This assay was used to determine the inhibition effect of the present compounds on the activity of monkey GnRHr protein expressed by monkey G...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2020
Entry Details
Go to US Patent