Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with Target = 'Golgi-associated PDZ and coiled-coil motif-containing protein'
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50596828(CHEMBL4783570)
Affinity DataKd:  490nMAssay Description:Binding affinity to CAL PDZ domain (unknown origin) assessed as dissociation constant in presence of tris(carboxylethyl)phosphine by fluorescence ani...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50555259(CHEMBL4756359)
Affinity DataKd:  6nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr by fluorescence pola...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50555258(CHEMBL4789294)
Affinity DataKd:  87nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr by fluorescence pola...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50555257(CHEMBL4763464)
Affinity DataKd:  49nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr by fluorescence pola...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50555256(CHEMBL4756115)
Affinity DataKd:  113nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr by fluorescence pola...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50555255(CHEMBL4777388)
Affinity DataIC50: 20nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-22 probe b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50555248(CHEMBL4779439)
Affinity DataIC50: 150nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-22 probe b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50555247(CHEMBL4789394)
Affinity DataIC50: 150nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-22 probe b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50555251(CHEMBL4739952)
Affinity DataIC50: 170nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-22 probe b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50555254(CHEMBL4753496)
Affinity DataIC50: 240nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-22 probe b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50555252(CHEMBL4795173)
Affinity DataIC50: 270nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-22 probe b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50555249(CHEMBL4798520)
Affinity DataIC50: 370nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-22 probe b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50555253(CHEMBL4792301)
Affinity DataIC50: 380nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-22 probe b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50555250(CHEMBL4752826)
Affinity DataIC50: 400nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-22 probe b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50555246(CHEMBL4790861)
Affinity DataIC50: 680nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-22 probe b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50555245(CHEMBL4762047)
Affinity DataIC50: 1.50E+3nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-22 probe b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50555236(CHEMBL4759877)
Affinity DataIC50: 1.60E+3nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-ANSRWPTSII...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50555244(CHEMBL4764244)
Affinity DataIC50: 1.80E+3nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-22 probe b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50613394(CHEMBL5278465)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of CAL (unknown origin) by Ambit kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50613392(CHEMBL5270581)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of CAL (unknown origin) by Ambit kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50613393(CHEMBL5288565)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of CAL (unknown origin) by Ambit kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50555239(CHEMBL4794279)
Affinity DataIC50: 2.20E+3nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-ANSRWPTSII...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50555238(CHEMBL4763642)
Affinity DataIC50: 2.40E+3nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-ANSRWPTSII...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50555240(CHEMBL4800168)
Affinity DataIC50: 2.50E+3nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-ANSRWPTSII...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50555235(CHEMBL4791418)
Affinity DataIC50: 3.70E+3nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-ANSRWPTSII...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50555234(CHEMBL4792820)
Affinity DataIC50: 4.30E+3nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-ANSRWPTSII...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50555241(CHEMBL4757746)
Affinity DataIC50: 7.40E+3nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-ANSRWPTSII...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50555237(CHEMBL4792234)
Affinity DataIC50: 7.90E+3nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-ANSRWPTSII...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50555243(CHEMBL4764592)
Affinity DataIC50: 8.00E+3nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-ANSRWPTSII...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50555242(CHEMBL4758509)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal His6 tagged CAL PDZ domain (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr using FAM-ANSRWPTSII...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50596827(CHEMBL5177006)
Affinity DataKi:  2.30E+3nMAssay Description:Inhibition of CAL PDZ domain (unknown origin) assessed as inhibition constant by fluorescence polarization competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50596826(CHEMBL5202803)
Affinity DataKi:  2.26E+4nMAssay Description:Inhibition of CAL PDZ domain (unknown origin) assessed as inhibition constant by fluorescence polarization competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetGolgi-associated PDZ and coiled-coil motif-containing protein(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50596825(CHEMBL5196216)
Affinity DataKi:  3.90E+5nMAssay Description:Inhibition of wild type CAL PDZ domain (unknown origin) expressed in Escherichia coli Rosette 2 (DE3) assessed as inhibition constant incubated for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed