Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with Target = 'Glutamine--fructose-6-phosphate aminotransferase [isomerizing]'
LigandPNGBDBM50356010(CHEMBL1911372)
Affinity DataIC50: 150nMAssay Description:Irreversible inhibition of GFATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
LigandPNGBDBM50356011(CHEMBL1911373)
Affinity DataIC50: 400nMAssay Description:Irreversible inhibition of GFATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
LigandPNGBDBM50356012(AAPTAMINE)
Affinity DataIC50: 1.20E+5nMAssay Description:Inhibition of GFAT using N-acetylglucosamine 6-phosphate as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetGlutamine--fructose-6-phosphate aminotransferase [isomerizing](Yeast)
Technical University of Gdansk

LigandPNGBDBM85319(GlcN-6-P synthase inhibitor, 12 (racemic mixture))
Affinity DataIC50: 5.00E+7nMpH: 6.85Assay Description:Two assays of GlcN-6-P synthase activity were used 1)determination of GlcN-6_P formation by the modified Elson-Morgan procedure and 2) continuous qua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2012
Entry Details

TargetGlutamine--fructose-6-phosphate aminotransferase [isomerizing](Yeast)
Technical University of Gdansk

LigandPNGBDBM85318(GlcN-6-P synthase inhibitor, 11 (racemic mixture))
Affinity DataIC50: 5.00E+7nMpH: 6.85Assay Description:Two assays of GlcN-6-P synthase activity were used 1)determination of GlcN-6_P formation by the modified Elson-Morgan procedure and 2) continuous qua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2012
Entry Details

TargetGlutamine--fructose-6-phosphate aminotransferase [isomerizing](Yeast)
Technical University of Gdansk

LigandPNGBDBM85317(GlcN-6-P synthase inhibitor, 10 (racemic mixture))
Affinity DataIC50: 5.00E+7nMpH: 6.85Assay Description:Two assays of GlcN-6-P synthase activity were used 1)determination of GlcN-6_P formation by the modified Elson-Morgan procedure and 2) continuous qua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2012
Entry Details

TargetGlutamine--fructose-6-phosphate aminotransferase [isomerizing](Yeast)
Technical University of Gdansk

LigandPNGBDBM85309(GlcN-6-P synthase inhibitor, 2 (racemic mixture))
Affinity DataIC50: 5.00E+7nMpH: 6.85Assay Description:Two assays of GlcN-6-P synthase activity were used 1)determination of GlcN-6_P formation by the modified Elson-Morgan procedure and 2) continuous qua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2012
Entry Details

TargetGlutamine--fructose-6-phosphate aminotransferase [isomerizing](Yeast)
Technical University of Gdansk

LigandPNGBDBM85310(GlcN-6-P synthase inhibitor, 3 (racemic mixture))
Affinity DataIC50: 5.00E+7nMpH: 6.85Assay Description:Two assays of GlcN-6-P synthase activity were used 1)determination of GlcN-6_P formation by the modified Elson-Morgan procedure and 2) continuous qua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2012
Entry Details

LigandPNGBDBM50356009(CHEMBL1911368)
Affinity DataKi:  300nMAssay Description:Competitive inhibition of GFAT in presence of glutamineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
LigandPNGBDBM50356009(CHEMBL1911368)
Affinity DataKi:  300nMAssay Description:Noncompetitive inhibition of GFAT in presence of fructose-6-phosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetGlutamine--fructose-6-phosphate aminotransferase [isomerizing](Escherichia coli (strain K12))
Enscp

LigandPNGBDBM100282((2S)-2-azaniumyl-3-[[(E)-4-methoxy-4-oxobut-2-enoy...)
Affinity DataKi:  350nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2013
Entry Details Article
PubMed
TargetGlutamine--fructose-6-phosphate aminotransferase [isomerizing](Escherichia coli (strain K12))
Enscp

LigandPNGBDBM100280((Z,5S)-5-amino-6-(carboxymethylamino)-1-diazonio-6...)
Affinity DataKi:  1.40E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2013
Entry Details Article
PubMed
TargetGlutamine--fructose-6-phosphate aminotransferase [isomerizing](Escherichia coli (strain K12))
Enscp

LigandPNGBDBM100281((E)-4-[[(2S)-2-azaniumyl-2-carboxylatoethyl]amino]...)
Affinity DataKi:  5.51E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2013
Entry Details Article
PubMed
TargetGlutamine--fructose-6-phosphate aminotransferase [isomerizing](Yeast)
Technical University of Gdansk

LigandPNGBDBM85322(GlcN-6-P synthase inhibitor, 15 (racemic mixture))
Affinity DataKi:  6.00E+5nM IC50: 1.60E+6nMpH: 6.85Assay Description:Two assays of GlcN-6-P synthase activity were used 1)determination of GlcN-6_P formation by the modified Elson-Morgan procedure and 2) continuous qua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2012
Entry Details

TargetGlutamine--fructose-6-phosphate aminotransferase [isomerizing](Yeast)
Technical University of Gdansk

LigandPNGBDBM85312(GlcN-6-P synthase inhibitor, 5 (racemic mixture))
Affinity DataKi:  9.00E+5nM IC50: 2.00E+6nMpH: 6.85Assay Description:Two assays of GlcN-6-P synthase activity were used 1)determination of GlcN-6_P formation by the modified Elson-Morgan procedure and 2) continuous qua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2012
Entry Details

TargetGlutamine--fructose-6-phosphate aminotransferase [isomerizing](Yeast)
Technical University of Gdansk

LigandPNGBDBM85316(GlcN-6-P synthase inhibitor, 9 (racemic mixture))
Affinity DataKi:  9.40E+5nM IC50: 3.60E+6nMpH: 6.85Assay Description:Two assays of GlcN-6-P synthase activity were used 1)determination of GlcN-6_P formation by the modified Elson-Morgan procedure and 2) continuous qua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2012
Entry Details

TargetGlutamine--fructose-6-phosphate aminotransferase [isomerizing](Yeast)
Technical University of Gdansk

LigandPNGBDBM85314(GlcN-6-P synthase inhibitor, 7 (racemic mixture))
Affinity DataKi:  4.40E+6nM IC50: 7.80E+6nMpH: 6.85Assay Description:Two assays of GlcN-6-P synthase activity were used 1)determination of GlcN-6_P formation by the modified Elson-Morgan procedure and 2) continuous qua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2012
Entry Details

TargetGlutamine--fructose-6-phosphate aminotransferase [isomerizing](Yeast)
Technical University of Gdansk

LigandPNGBDBM85321(GlcN-6-P synthase inhibitor, 14 (racemic mixture))
Affinity DataKi:  2.80E+6nM IC50: 5.50E+6nMpH: 6.85Assay Description:Two assays of GlcN-6-P synthase activity were used 1)determination of GlcN-6_P formation by the modified Elson-Morgan procedure and 2) continuous qua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2012
Entry Details

TargetGlutamine--fructose-6-phosphate aminotransferase [isomerizing](Yeast)
Technical University of Gdansk

LigandPNGBDBM85320(GlcN-6-P synthase inhibitor, 13 (racemic mixture))
Affinity DataKi:  1.50E+6nM IC50: 2.80E+6nMpH: 6.85Assay Description:Two assays of GlcN-6-P synthase activity were used 1)determination of GlcN-6_P formation by the modified Elson-Morgan procedure and 2) continuous qua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2012
Entry Details

TargetGlutamine--fructose-6-phosphate aminotransferase [isomerizing](Yeast)
Technical University of Gdansk

LigandPNGBDBM50004051(CHEMBL285843 | 2-Amino-4-phosphono-butyric acid | ...)
Affinity DataKi:  1.20E+7nM IC50: 2.60E+7nMpH: 6.85Assay Description:Two assays of GlcN-6-P synthase activity were used 1)determination of GlcN-6_P formation by the modified Elson-Morgan procedure and 2) continuous qua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2012
Entry Details

TargetGlutamine--fructose-6-phosphate aminotransferase [isomerizing](Yeast)
Technical University of Gdansk

LigandPNGBDBM85313(GlcN-6-P synthase inhibitor, 6 (racemic mixture))
Affinity DataKi:  1.10E+7nM IC50: 2.50E+7nMpH: 6.85Assay Description:Two assays of GlcN-6-P synthase activity were used 1)determination of GlcN-6_P formation by the modified Elson-Morgan procedure and 2) continuous qua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2012
Entry Details

TargetGlutamine--fructose-6-phosphate aminotransferase [isomerizing](Yeast)
Technical University of Gdansk

LigandPNGBDBM85311(GlcN-6-P synthase inhibitor, 4 (racemic mixture))
Affinity DataKi:  1.20E+6nM IC50: 2.60E+6nMpH: 6.85Assay Description:Two assays of GlcN-6-P synthase activity were used 1)determination of GlcN-6_P formation by the modified Elson-Morgan procedure and 2) continuous qua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2012
Entry Details

TargetGlutamine--fructose-6-phosphate aminotransferase [isomerizing](Yeast)
Technical University of Gdansk

LigandPNGBDBM85315(GlcN-6-P synthase inhibitor, 8 (racemic mixture))
Affinity DataKi:  1.30E+6nM IC50: 4.40E+6nMpH: 6.85Assay Description:Two assays of GlcN-6-P synthase activity were used 1)determination of GlcN-6_P formation by the modified Elson-Morgan procedure and 2) continuous qua...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2012
Entry Details