Compile Data Set for Download or QSAR
Report error Found 3594 Enz. Inhib. hit(s) with Target = 'Glutaminase kidney isoform, mitochondrial'
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50232186(CHEMBL4092049)
Affinity DataKd:  4.95E+3nMAssay Description:Binding affinity to NT-647-NHS-labelled KGA (unknown origin) after 10 mins by microscale thermophoresis methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50400050(CHEMBL2177757 | US8604016, 1 | US9938267, Cmpd ID ...)
Affinity DataKd:  200nMAssay Description:Binding affinity to recombinant human C-terminal His-tagged GLS1 after 3 hrs in presence of glycine by GDH coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50512566(CHEMBL4444708)
Affinity DataKd:  142nMAssay Description:Binding affinity to human KGA assessed as dissociation constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50509184(CHEMBL4593229)
Affinity DataKd:  610nMAssay Description:Binding affinity to human GLS1 expressed in Escherichia coli strain BL21 (DE3)pLysS by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50509184(CHEMBL4593229)
Affinity DataKd:  450nMAssay Description:Binding affinity to human GLS1 expressed in Escherichia coli strain BL21 (DE3)pLysS by fluorescence polarization binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50509187(CHEMBL4526354)
Affinity DataKd:  350nMAssay Description:Binding affinity to human GLS1 expressed in Escherichia coli strain BL21 (DE3)pLysS by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50509188(CHEMBL4566446)
Affinity DataKd:  68nMAssay Description:Binding affinity to human GLS1 expressed in Escherichia coli strain BL21 (DE3)pLysS by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM109086(US8604016, 670 | US9938267, Cmpd ID 670 | US107935...)
Affinity DataKd:  92nMAssay Description:Binding affinity to human GLS1 expressed in Escherichia coli strain BL21 (DE3)pLysS by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50400050(CHEMBL2177757 | US8604016, 1 | US9938267, Cmpd ID ...)
Affinity DataKd:  4.30E+3nMAssay Description:Binding affinity to human GLS1 expressed in Escherichia coli strain BL21 (DE3)pLysS by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM109086(US8604016, 670 | US9938267, Cmpd ID 670 | US107935...)
Affinity DataKd:  1.5nMAssay Description:Binding affinity to wild type human KGA assessed as covalent bond formation by measuring dissociation constant by biomolecular interaction assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50574392(CHEMBL4849357)
Affinity DataKd:  24nMAssay Description:Binding affinity to human GLS1 expressed in Escherichia coli strain BL21 (DE3) assessed as dissociation constant by surface plasmon resonance analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50574392(CHEMBL4849357)
Affinity DataKoff:  2.09E+4s-1Assay Description:Binding affinity to human GLS1 expressed in Escherichia coli strain BL21 (DE3) assessed as association rate constant by surface plasmon resonance ana...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50574392(CHEMBL4849357)
Affinity DataKon:  0.00300M-1s-1Assay Description:Binding affinity to human GLS1 expressed in Escherichia coli strain BL21 (DE3) assessed as dissociation rate constant by surface plasmon resonance an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM109086(US8604016, 670 | US9938267, Cmpd ID 670 | US107935...)
Affinity DataKd:  105nMAssay Description:Binding affinity to human GLS1 expressed in Escherichia coli strain BL21 (DE3) by ITC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50574392(CHEMBL4849357)
Affinity DataKd:  37nMAssay Description:Binding affinity to human GLS1 expressed in Escherichia coli strain BL21 (DE3) by ITC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50593582(CHEMBL5179292)
Affinity DataEC50:  3.96E+3nMAssay Description:Inhibition of human recombinant GLS-1 by measuring glutamate production incubated for 1 hr by fluorescence based multimode plate reader methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM109086(US8604016, 670 | US9938267, Cmpd ID 670 | US107935...)
Affinity DataKd:  106nMAssay Description:Binding affinity to human GLS1 assessed as dissociation constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50605215(CHEMBL5178036)
Affinity DataKd:  81nMAssay Description:Binding affinity to human GLS1 assessed as dissociation constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50605217(CHEMBL5194638)
Affinity DataKd:  52nMAssay Description:Binding affinity to human GLS1 assessed as dissociation constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50652793(CHEMBL5653589)
Affinity DataKd:  3.02E+4nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50503299(CHEMBL4538736)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of kidney-type glutaminase in human BT20 cells assessed as reduction in glutamate levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50503300(CHEMBL4547874)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of kidney-type glutaminase in human BT20 cells assessed as reduction in glutamate levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50172241(CHEMBL3810168 | US10294221, Example 22(a))
Affinity DataIC50: 0.206nMAssay Description:Inhibition of GLS1 in human PC3 cells assessed as cellular glutamate depletion levels after 6 hrs by Glutamate Oxidase/ AmplexRed coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50172181(CHEMBL3810394 | US10040788, Example 3 | US10294221...)
Affinity DataIC50: 0.390nMAssay Description:Inhibition of GLS1 in human PC3 cells assessed as cellular glutamate depletion levels after 6 hrs by Glutamate Oxidase/ AmplexRed coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50172239(CHEMBL3809014 | US10040788, Example 11 | US1029422...)
Affinity DataIC50: 0.401nMAssay Description:Inhibition of GLS1 in human PC3 cells assessed as cellular glutamate depletion levels after 6 hrs by Glutamate Oxidase/ AmplexRed coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50503313(CHEMBL4454263)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of kidney-type glutaminase in human BT20 cells assessed as reduction in glutamate levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50517268(CHEMBL4475144)
Affinity DataIC50: 1nMAssay Description:Inhibition of human KGA preincubated for 15 to 30 mins followed by substrate addition and measured after 3 to 4 hrs by GDH-EZMTT reagent-based GDH co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50517275(CHEMBL4469040)
Affinity DataIC50: 1nMAssay Description:Inhibition of human KGA preincubated for 15 to 30 mins followed by substrate addition and measured after 3 to 4 hrs by GDH-EZMTT reagent-based GDH co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM47230(US8604016, 645 | US9938267, Cmpd ID 645)
Affinity DataIC50: 2nMAssay Description:Compounds were assessed for their ability to inhibit the enzymatic activity of a recombinant form of Glutaminase 1 (GAC) using a biochemical assay th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/12/2014
Entry Details
Go to US Patent

TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM108852(US8604016, 432 | US9938267, Cmpd ID 432)
Affinity DataIC50: 2nMAssay Description:Compounds were assessed for their ability to inhibit the enzymatic activity of a recombinant form of Glutaminase 1 (GAC) using a biochemical assay th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/12/2014
Entry Details
Go to US Patent

TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM108853(US8604016, 433 | US9938267, Cmpd ID 433)
Affinity DataIC50: 2nMAssay Description:Compounds were assessed for their ability to inhibit the enzymatic activity of a recombinant form of Glutaminase 1 (GAC) using a biochemical assay th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/12/2014
Entry Details
Go to US Patent

TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM108855(US8604016, 435 | US9938267, Cmpd ID 435)
Affinity DataIC50: 2nMAssay Description:Compounds were assessed for their ability to inhibit the enzymatic activity of a recombinant form of Glutaminase 1 (GAC) using a biochemical assay th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/12/2014
Entry Details
Go to US Patent

TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM108893(US8604016, 473 | US9938267, Cmpd ID 473)
Affinity DataIC50: 2nMAssay Description:Compounds were assessed for their ability to inhibit the enzymatic activity of a recombinant form of Glutaminase 1 (GAC) using a biochemical assay th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/12/2014
Entry Details
Go to US Patent

TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM108895(US8604016, 475 | US9938267, Cmpd ID 475)
Affinity DataIC50: 2nMAssay Description:Compounds were assessed for their ability to inhibit the enzymatic activity of a recombinant form of Glutaminase 1 (GAC) using a biochemical assay th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/12/2014
Entry Details
Go to US Patent

TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM108787(US8604016, 367 | US9938267, Cmpd ID 367)
Affinity DataIC50: 2nMAssay Description:Compounds were assessed for their ability to inhibit the enzymatic activity of a recombinant form of Glutaminase 1 (GAC) using a biochemical assay th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
Go to US Patent

TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM108852(US8604016, 432 | US9938267, Cmpd ID 432)
Affinity DataIC50: 2nMAssay Description:Compounds were assessed for their ability to inhibit the enzymatic activity of a recombinant form of Glutaminase 1 (GAC) using a biochemical assay th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
Go to US Patent

TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM108853(US8604016, 433 | US9938267, Cmpd ID 433)
Affinity DataIC50: 2nMAssay Description:Compounds were assessed for their ability to inhibit the enzymatic activity of a recombinant form of Glutaminase 1 (GAC) using a biochemical assay th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
Go to US Patent

TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM108855(US8604016, 435 | US9938267, Cmpd ID 435)
Affinity DataIC50: 2nMAssay Description:Compounds were assessed for their ability to inhibit the enzymatic activity of a recombinant form of Glutaminase 1 (GAC) using a biochemical assay th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
Go to US Patent

TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM108893(US8604016, 473 | US9938267, Cmpd ID 473)
Affinity DataIC50: 2nMAssay Description:Compounds were assessed for their ability to inhibit the enzymatic activity of a recombinant form of Glutaminase 1 (GAC) using a biochemical assay th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
Go to US Patent

TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM108895(US8604016, 475 | US9938267, Cmpd ID 475)
Affinity DataIC50: 2nMAssay Description:Compounds were assessed for their ability to inhibit the enzymatic activity of a recombinant form of Glutaminase 1 (GAC) using a biochemical assay th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
Go to US Patent

TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM47230(US8604016, 645 | US9938267, Cmpd ID 645)
Affinity DataIC50: 2nMAssay Description:Compounds were assessed for their ability to inhibit the enzymatic activity of a recombinant form of Glutaminase 1 (GAC) using a biochemical assay th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
Go to US Patent

TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM109086(US8604016, 670 | US9938267, Cmpd ID 670 | US107935...)
Affinity DataIC50: 2nMAssay Description:Inhibition of human KGA preincubated for 15 to 30 mins followed by substrate addition and measured after 3 to 4 hrs by GDH-EZMTT reagent-based GDH co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM109086(US8604016, 670 | US9938267, Cmpd ID 670 | US107935...)
Affinity DataIC50: 2nMAssay Description:Negative allosteric modulator activity at human wildtype KGA incubated for 5 hrs in presence of GDH and NADP by EZMTT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50503298(CHEMBL4462146)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of kidney-type glutaminase in human BT20 cells assessed as reduction in glutamate levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM108802(US8604016, 382 | US9938267, Cmpd ID 382)
Affinity DataIC50: 3nMAssay Description:Compounds were assessed for their ability to inhibit the enzymatic activity of a recombinant form of Glutaminase 1 (GAC) using a biochemical assay th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/12/2014
Entry Details
Go to US Patent

TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM108804(US8604016, 384 | US9938267, Cmpd ID 384)
Affinity DataIC50: 3nMAssay Description:Compounds were assessed for their ability to inhibit the enzymatic activity of a recombinant form of Glutaminase 1 (GAC) using a biochemical assay th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/12/2014
Entry Details
Go to US Patent

TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM108864(US8604016, 444 | US9938267, Cmpd ID 444)
Affinity DataIC50: 3nMAssay Description:Compounds were assessed for their ability to inhibit the enzymatic activity of a recombinant form of Glutaminase 1 (GAC) using a biochemical assay th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/12/2014
Entry Details
Go to US Patent

TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM108871(US8604016, 451 | US9938267, Cmpd ID 451)
Affinity DataIC50: 3nMAssay Description:Compounds were assessed for their ability to inhibit the enzymatic activity of a recombinant form of Glutaminase 1 (GAC) using a biochemical assay th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/12/2014
Entry Details
Go to US Patent

TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM108873(US8604016, 453 | US9938267, Cmpd ID 453)
Affinity DataIC50: 3nMAssay Description:Compounds were assessed for their ability to inhibit the enzymatic activity of a recombinant form of Glutaminase 1 (GAC) using a biochemical assay th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/12/2014
Entry Details
Go to US Patent

TargetGlutaminase kidney isoform, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM108875(US8604016, 455 | US9938267, Cmpd ID 455)
Affinity DataIC50: 3nMAssay Description:Compounds were assessed for their ability to inhibit the enzymatic activity of a recombinant form of Glutaminase 1 (GAC) using a biochemical assay th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/12/2014
Entry Details
Go to US Patent

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