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Report error Found 2090 Enz. Inhib. hit(s) with Target = 'Glucagon receptor'
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098571(His-Ser-Gln-Gly-Thr-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Ty...)
Affinity DataEC50:  8nMAssay Description:cAMP accumulation in rat hepatocytes in the presence rolipramMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059356([des-His1, Nle6, Glu9] glucagon-NH2 | CHEMBL236999...)
Affinity DataKd:  501nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059365([des-Phe6, Glu9] glucagon-NH2 | CHEMBL412352)
Affinity DataKd:  631nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059354([des-Phe6] glucagon-NH2 | CHEMBL438574)
Affinity DataKd:  501nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059360([des-His1, des-Phe6] glucagon-NH2 | CHEMBL429198)
Affinity DataKd:  562nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059351([des-His1, des-Phe6, Glu9] glucagon | [des-Phe6, G...)
Affinity DataKd:  794nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059355([des-Phe6] glucagon | CHEMBL409611)
Affinity DataKd:  562nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059361([des-His1, des-Phe6] glucagon | CHEMBL439271)
Affinity DataKd:  708nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059357([des-His1, Asp6, Glu9] glucagon-NH2 | CHEMBL438218)
Affinity DataKd:  501nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50301952((3S,6S,9S,12S,15S,21S)-21-(2-((S)-2-amino-3-(1H-im...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at glucagon receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50044849(CHEMBL3311308)
Affinity DataEC50: <5.01E+4nMAssay Description:Agonist activity at human glucagon receptor expressed in CHO cells by luciferase HTS/summary (Abse5) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50087844(c[ Lys12, Asp21] glucagon-NH2 | CHEMBL266411)
Affinity DataEC50:  794nMAssay Description:In vitro receptor binding affinity (95% CL) using rat liver plasma membrane bioassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098571(His-Ser-Gln-Gly-Thr-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Ty...)
Affinity DataEC50:  5nMAssay Description:In vitro receptor binding affinity (95% CL) using rat liver plasma membrane bioassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50087848(c[Asp15, Lys18,] glucagon-NH2 | CHEMBL427644)
Affinity DataEC50:  320nMAssay Description:In vitro receptor binding affinity (95% CL) using rat liver plasma membrane bioassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059362([des-His1, des-Phe6, Glu9] glucagon-NH2 | CHEMBL26...)
Affinity DataKd:  6.31nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059358([des-His1, Tyr6,Glu9] glucagon-NH2 | CHEMBL267885)
Affinity DataKd:  631nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059359([des-His1, des-Gly4, Glu9] glucagon-NH2 | CHEMBL41...)
Affinity DataKd:  891nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059363([des-His1,Ala6, Glu9] glucagon-NH2 | CHEMBL437095)
Affinity DataKd:  398nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059352([des-His1, Trp6, Glu9] glucagon-NH2 | CHEMBL442499)
Affinity DataKd:  562nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324711(CHEMBL1222085)
Affinity DataEC50:  0.0770nMAssay Description:Agonist activity at GCGR expressed in HEK293 cells assessed as stimulation of cAMP production by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324712(HSQGTFTSDYSKYLDEQAAKEFIAWLVKG | CHEMBL1222086)
Affinity DataEC50:  0.470nMAssay Description:Agonist activity at GCGR expressed in HEK293 cells assessed as stimulation of cAMP production by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324713(HSQGTFTSDYSKYLDEQAAKEFIAWLMNT | CHEMBL1222087)
Affinity DataEC50:  0.0680nMAssay Description:Agonist activity at GCGR expressed in HEK293 cells assessed as stimulation of cAMP production by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324714(CHEMBL1222088)
Affinity DataEC50:  0.0480nMAssay Description:Agonist activity at GCGR expressed in HEK293 cells assessed as stimulation of cAMP production by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324715(CHEMBL1222089)
Affinity DataEC50:  0.0870nMAssay Description:Agonist activity at GCGR expressed in HEK293 cells assessed as stimulation of cAMP production by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324716(CHEMBL1222090)
Affinity DataEC50:  0.0680nMAssay Description:Agonist activity at GCGR expressed in HEK293 cells assessed as stimulation of cAMP production by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324717(CHEMBL1222091)
Affinity DataEC50:  0.0730nMAssay Description:Agonist activity at GCGR expressed in HEK293 cells assessed as stimulation of cAMP production by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324718(CHEMBL1222092)
Affinity DataEC50:  0.0800nMAssay Description:Agonist activity at GCGR expressed in HEK293 cells assessed as stimulation of cAMP production by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324719(HAEGTFTSDVSSYLEERRAQDFVQWLMNT | CHEMBL1222093)
Affinity DataEC50:  50nMAssay Description:Agonist activity at GCGR expressed in HEK293 cells assessed as stimulation of cAMP production by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324720(CHEMBL1222094)
Affinity DataEC50:  3.70nMAssay Description:Agonist activity at GCGR expressed in HEK293 cells assessed as stimulation of cAMP production by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324721(CHEMBL1222095)
Affinity DataEC50:  2.40nMAssay Description:Agonist activity at GCGR expressed in HEK293 cells assessed as stimulation of cAMP production by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324722(CHEMBL1222096)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at GCGR expressed in HEK293 cells assessed as stimulation of cAMP production by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324723(CHEMBL1222097)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at GCGR expressed in HEK293 cells assessed as stimulation of cAMP production by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324724(CHEMBL1222098)
Affinity DataEC50:  0.0460nMAssay Description:Agonist activity at GCGR expressed in HEK293 cells assessed as stimulation of cAMP production by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324725(CHEMBL1222099)
Affinity DataEC50:  0.0580nMAssay Description:Agonist activity at GCGR expressed in HEK293 cells assessed as stimulation of cAMP production by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324726(CHEMBL1222100)
Affinity DataEC50:  0.0780nMAssay Description:Agonist activity at GCGR expressed in HEK293 cells assessed as stimulation of cAMP production by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324727(CHEMBL1222101)
Affinity DataEC50:  0.0760nMAssay Description:Agonist activity at GCGR expressed in HEK293 cells assessed as stimulation of cAMP production by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324728(CHEMBL1222102)
Affinity DataEC50:  0.590nMAssay Description:Agonist activity at GCGR expressed in HEK293 cells assessed as stimulation of cAMP production by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324729(CHEMBL1222174)
Affinity DataEC50:  0.0550nMAssay Description:Agonist activity at GCGR expressed in HEK293 cells assessed as stimulation of cAMP production by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50098571(His-Ser-Gln-Gly-Thr-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Ty...)
Affinity DataEC50:  0.0710nMAssay Description:Agonist activity at GCGR expressed in HEK293 cells assessed as stimulation of cAMP production by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324731(HAEGTFTSDVSSYLEGQAAKEFIAWLVKGR | CHEMBL1222074)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at GCGR expressed in HEK293 cells assessed as stimulation of cAMP production by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324732(CHEMBL1222075)
Affinity DataEC50:  0.150nMAssay Description:Agonist activity at GCGR expressed in HEK293 cells assessed as stimulation of cAMP production by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324702(CHEMBL1222076)
Affinity DataEC50:  0.0490nMAssay Description:Agonist activity at GCGR expressed in HEK293 cells assessed as stimulation of cAMP production by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324703(CHEMBL1222077)
Affinity DataEC50:  0.0530nMAssay Description:Agonist activity at GCGR expressed in HEK293 cells assessed as stimulation of cAMP production by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324704(CHEMBL1222078)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at GCGR expressed in HEK293 cells assessed as stimulation of cAMP production by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324705(CHEMBL1222079)
Affinity DataEC50:  0.0710nMAssay Description:Agonist activity at GCGR expressed in HEK293 cells assessed as stimulation of cAMP production by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324706(CHEMBL1222080)
Affinity DataEC50:  0.0540nMAssay Description:Agonist activity at GCGR expressed in HEK293 cells assessed as stimulation of cAMP production by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324707(CHEMBL1222081)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at GCGR expressed in HEK293 cells assessed as stimulation of cAMP production by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324708(CHEMBL1222082)
Affinity DataEC50:  0.0680nMAssay Description:Agonist activity at GCGR expressed in HEK293 cells assessed as stimulation of cAMP production by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324709(CHEMBL1222083)
Affinity DataEC50:  0.130nMAssay Description:Agonist activity at GCGR expressed in HEK293 cells assessed as stimulation of cAMP production by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50324710(CHEMBL1222084)
Affinity DataEC50:  0.130nMAssay Description:Agonist activity at GCGR expressed in HEK293 cells assessed as stimulation of cAMP production by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2013
Entry Details Article
PubMed
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