Report error Found 109 Enz. Inhib. hit(s) with Target = 'Gamma-aminobutyric acid receptor subunit rho-1'
Affinity DataEC50: 440nMAssay Description:Partial agonist activity against human rho-1 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 6.80E+4nMAssay Description:Full agonist activity against human rho-1 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 270nMAssay Description:Agonist activity at human GABAA rho1 expressed in tsA-201cells by FLIPR membrane potential blue assayMore data for this Ligand-Target Pair
Affinity DataEC50: 700nMAssay Description:Agonist activity at human GABAA rho1 expressed in tsA-201cells by FLIPR membrane potential blue assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.90E+4nMAssay Description:Agonist activity at human GABAA rho1 expressed in tsA-201cells by FLIPR membrane potential blue assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human GABAA rho1 expressed in tsA-201cells by FLIPR membrane potential blue assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human GABAA rho1 expressed in tsA-201cells by FLIPR membrane potential blue assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human GABAA rho1 expressed in tsA-201cells by FLIPR membrane potential blue assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human GABAA rho1 expressed in tsA-201cells by FLIPR membrane potential blue assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.30E+3nMAssay Description:Agonist activity at human GABAA rho1 expressed in tsA-201cells by FLIPR membrane potential blue assayMore data for this Ligand-Target Pair
Affinity DataEC50: 8.10E+3nMAssay Description:Agonist activity at human GABAA rho1 expressed in tsA-201cells by FLIPR membrane potential blue assayMore data for this Ligand-Target Pair
Affinity DataEC50: 269nMAssay Description:Agonist activity at human GABAA rho1 expressed in tsA-201cells by FLIPR membrane potential blue assayMore data for this Ligand-Target Pair
Affinity DataEC50: 692nMAssay Description:Agonist activity at human GABAA rho1 expressed in tsA-201cells by FLIPR membrane potential blue assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.89E+4nMAssay Description:Agonist activity at human GABAA rho1 expressed in tsA-201cells by FLIPR membrane potential blue assayMore data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+6nMAssay Description:Agonist activity at human GABAA rho1 expressed in tsA-201cells by FLIPR membrane potential blue assayMore data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+6nMAssay Description:Agonist activity at human GABAA rho1 expressed in tsA-201cells by FLIPR membrane potential blue assayMore data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+6nMAssay Description:Agonist activity at human GABAA rho1 expressed in tsA-201cells by FLIPR membrane potential blue assayMore data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+6nMAssay Description:Agonist activity at human GABAA rho1 expressed in tsA-201cells by FLIPR membrane potential blue assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.30E+3nMAssay Description:Agonist activity at human GABAA rho1 expressed in tsA-201cells by FLIPR membrane potential blue assayMore data for this Ligand-Target Pair
Affinity DataEC50: 8.10E+3nMAssay Description:Agonist activity at human GABAA rho1 expressed in tsA-201cells by FLIPR membrane potential blue assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.00E+4nMAssay Description:Agonist activity at human GABAc Rho1 receptor expressed in Xenopus oocytes assessed as whole cell current production by two electrode voltage clamp m...More data for this Ligand-Target Pair
Affinity DataEC50: 400nMAssay Description:Agonist activity at human GABAc Rho1 receptor expressed in Xenopus oocytes assessed as whole cell current production by two electrode voltage clamp m...More data for this Ligand-Target Pair
Affinity DataEC50: 1.40E+3nMAssay Description:Agonist activity at human GABAc Rho1 receptor expressed in Xenopus oocytes assessed as whole cell current production by two electrode voltage clamp m...More data for this Ligand-Target Pair
Affinity DataEC50: 5.90E+4nMAssay Description:Agonist activity at human GABAc Rho1 receptor expressed in Xenopus oocytes assessed as whole cell current production by two electrode voltage clamp m...More data for this Ligand-Target Pair
Affinity DataEC50: 9.00E+3nMAssay Description:Agonist activity at human GABAc Rho1 receptor expressed in Xenopus oocytes assessed as whole cell current production by two electrode voltage clamp m...More data for this Ligand-Target Pair
Affinity DataEC50: 800nMAssay Description:Agonist activity at human GABAc Rho1 receptor expressed in Xenopus oocytes assessed as whole cell current production by two electrode voltage clamp m...More data for this Ligand-Target Pair
Affinity DataEC50: 7.40E+4nMAssay Description:Agonist activity at human GABAc Rho1 receptor expressed in Xenopus oocytes assessed as whole cell current production by two electrode voltage clamp m...More data for this Ligand-Target Pair
Affinity DataKd: 2.30E+3nMAssay Description:Partial agonist activity against human rho-1 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 600nMAssay Description:Partial agonist activity against homomeric rho-1 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+4nMAssay Description:Full agonist activity against human rho-1 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 2.43E+3nMAssay Description:Partial agonist activity against rho-1 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 1.60E+4nMAssay Description:Partial agonist activity against rho-1 subunit GABA-C receptor expressed in Xenopus oocytes, low intrinsic activity (Im 3%)More data for this Ligand-Target Pair
Affinity DataEC50: 4.60E+3nMAssay Description:Partial agonist activity against human rho-1 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 7.40E+4nMAssay Description:Partial agonist activity against human rho-1 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+5nMAssay Description:Agonist activity at human GABAA rho1 receptor expressed in TSA201 cells after 1 min by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+5nMAssay Description:Agonist activity at human GABAA rho1 receptor expressed in TSA201 cells after 1 min by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+5nMAssay Description:Agonist activity at human GABAA rho1 receptor expressed in TSA201 cells after 1 min by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+5nMAssay Description:Agonist activity at human GABAA rho1 receptor expressed in TSA201 cells after 1 min by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+5nMAssay Description:Agonist activity at human GABAA rho1 receptor expressed in TSA201 cells after 1 min by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+5nMAssay Description:Agonist activity at human GABAA rho1 receptor expressed in TSA201 cells after 1 min by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: >5.00E+5nMAssay Description:Agonist activity at human GABAA rho1 receptor expressed in TSA201 cells after 1 min by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.10E+3nMAssay Description:Agonist activity at human GABAA rho1 receptor expressed in TSA201 cells after 1 min by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 700nMAssay Description:Agonist activity at human GABAA rho1 receptor expressed in TSA201 cells after 1 min by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 270nMAssay Description:Agonist activity at human GABAA rho1 receptor expressed in TSA201 cells after 1 min by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.50E+4nMAssay Description:Agonist activity at human GABAA rho1 receptor expressed in HEK293 cells by patch clamp electrophysiology assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.30E+3nMAssay Description:Partial agonist activity at GABAC rho1 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 2.20E+4nMAssay Description:Agonist activity at GABAC rho1 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 3.97E+4nMAssay Description:Agonist activity at GABAC rho1 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Agonist activity at GABAC rho1 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 6.50E+4nMAssay Description:Agonist activity at human recombinant GABAc rho1 receptor expressed in Xenopus laevis oocytes at -60mV by two-electrode voltage clamp methodMore data for this Ligand-Target Pair



3D Structure (crystal)

























