Compile Data Set for Download or QSAR
Report error Found 58 Enz. Inhib. hit(s) with Target = 'Hydroxycarboxylic acid receptor 1'
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539685(CHEMBL4649089)
Affinity DataEC50:  21nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539672(CHEMBL4640189)
Affinity DataEC50:  22nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539673(CHEMBL4635725)
Affinity DataEC50:  360nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539674(CHEMBL4636849)
Affinity DataEC50:  560nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539675(CHEMBL4636565)
Affinity DataEC50:  299nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539676(CHEMBL4639430)
Affinity DataEC50:  103nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539677(CHEMBL4641428)
Affinity DataEC50:  260nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539678(CHEMBL4633947)
Affinity DataEC50:  769nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50462127(CHEMBL4239086)
Affinity DataEC50:  120nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539679(CHEMBL4638731)
Affinity DataEC50:  719nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539680(CHEMBL4643496)
Affinity DataEC50:  895nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539681(CHEMBL4634029)
Affinity DataEC50:  166nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539682(CHEMBL4642413)
Affinity DataEC50: >1.60E+4nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539683(CHEMBL4635119)
Affinity DataEC50: >3.30E+4nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539684(CHEMBL4641120)
Affinity DataEC50: >3.30E+4nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539671(CHEMBL4641219)
Affinity DataEC50:  19nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539686(CHEMBL4644587)
Affinity DataEC50:  490nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539687(CHEMBL4635089)
Affinity DataEC50:  22nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539688(CHEMBL4638263)
Affinity DataEC50:  75nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539689(CHEMBL4642043)
Affinity DataEC50:  5nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539690(CHEMBL4645314)
Affinity DataEC50:  240nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539691(CHEMBL4642179)
Affinity DataEC50:  410nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539692(CHEMBL4638676)
Affinity DataEC50:  740nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539693(CHEMBL4646005)
Affinity DataEC50:  110nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539694(CHEMBL4633635)
Affinity DataEC50:  600nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539695(CHEMBL4649741)
Affinity DataEC50:  160nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539696(CHEMBL4641503)
Affinity DataEC50:  270nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539697(CHEMBL4636832)
Affinity DataEC50:  54nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539698(CHEMBL4641449)
Affinity DataEC50:  1.90E+3nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50391828(CHEMBL2146992)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50391823(CHEMBL2146902)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50336491(CHEMBL65369 | 3-Hydroxybenzoate, II | 3-hydroxyben...)
Affinity DataEC50:  1.84E+5nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50391824(CHEMBL2146903)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50391818(CHEMBL2146904)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50391819(CHEMBL2146905)
Affinity DataEC50:  4.20E+4nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50391817(CHEMBL2146485)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50391816(CHEMBL2146906)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50391821(CHEMBL2146907)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50391820(CHEMBL2146908)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50391815(CHEMBL2146909)
Affinity DataEC50:  1.29E+5nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50391825(CHEMBL2146910)
Affinity DataEC50:  1.60E+4nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50391822(CHEMBL2146989)
Affinity DataEC50:  3.80E+4nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50391826(CHEMBL2146990)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50391827(CHEMBL2146991)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50336490(3,5-dihydroxybenzoic acid | 3,5-dihydroxybenzoicac...)
Affinity DataEC50:  3.77E+5nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50391829(CHEMBL2146993)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at human recombinant GPR81 transfected in african green monkey COS-7 cells after 20 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM50391825(CHEMBL2146910)
Affinity DataEC50:  6.70E+4nMAssay Description:Agonist activity at dog GPR81More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50391825(CHEMBL2146910)
Affinity DataEC50:  2.20E+4nMAssay Description:Agonist activity at mouse GPR81More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539662(CHEMBL4641579)
Affinity DataEC50:  23nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetHydroxycarboxylic acid receptor 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50539663(CHEMBL4632411)
Affinity DataEC50:  74nMAssay Description:Agonist activity at human GPR81 overexpressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
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