Compile Data Set for Download or QSAR
Report error Found 116 Enz. Inhib. hit(s) with Target = 'G protein-activated inward rectifier potassium channel 1/4'
TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM50437968(CHEMBL2409134)
Affinity DataEC50:  3.50E+3nMAssay Description:Activation of GIRK1/4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585716(US11530213, Example 37 | 8-chloro-1-(2,6-dichlorop...)
Affinity DataIC50: 6nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585717(US11530213, Example 38 | 8-chloro-1-(2,6-dichlorop...)
Affinity DataIC50: 8nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585715(US11530213, Example 36 | N-(2-((8-chloro-1-(2,6- d...)
Affinity DataIC50: 9nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585727(US11530213, Example 48 | 8-chloro-1-(2,6-dichlorop...)
Affinity DataIC50: 9nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585729(US11530213, Example 50 | 8-chloro-1-(2,6-dichlorop...)
Affinity DataIC50: 11nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585719(US11530213, Example 40 | 8-chloro-1-(2,6-chlorophe...)
Affinity DataIC50: 13nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585741(US11530213, Example 62)
Affinity DataIC50: 13nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585738(US11530213, Example 59)
Affinity DataIC50: 14nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585718(US11530213, Example 39 | (S)-8-chloro-1-(2,6- dich...)
Affinity DataIC50: 15nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585721(US11530213, Example 42 | 8-chloro-1-(2,6-dichlorop...)
Affinity DataIC50: 15nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585742(US11530213, Example 63)
Affinity DataIC50: 16nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585737(US11530213, Example 58)
Affinity DataIC50: 17nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585764(US11530213, Example 85)
Affinity DataIC50: 19nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585760(US11530213, Example 81)
Affinity DataIC50: 23nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
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TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585768(US11530213, Example 89)
Affinity DataIC50: 24nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585694(US11530213, Example 15 | 5-(2,5,8,11,14,17- hexaox...)
Affinity DataIC50: 25nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585709(US11530213, Example 30 | 8-chloro-1-(2,6-dichlorop...)
Affinity DataIC50: 25nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585722(US11530213, Example 43 | 3,5-dichloro-4-(8-chloro-...)
Affinity DataIC50: 26nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585720(US11530213, Example 41 | 8-chloro-1-(2,6-dichlorop...)
Affinity DataIC50: 28nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585732(US11530213, Example 53 | 8-chloro-1-(2,6-dichlorop...)
Affinity DataIC50: 28nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585733(US11530213, Example 54 | 8-chloro-1-(2,6-dichlorop...)
Affinity DataIC50: 29nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM695823(US12084442, Example 16 | 3-((8-Chloro-1-(2,6-dichl...)
Affinity DataIC50: 30nMAssay Description:The GIRK1/4 activity of a compound according to the present invention was assessed by the following in vitro method.Buffers:a. External buffer: 10 mM...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
1/6/2025
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM695825(US12084442, Example 18 | 3-((8-Chloro-1-(2,6-dichl...)
Affinity DataIC50: 30nMAssay Description:The GIRK1/4 activity of a compound according to the present invention was assessed by the following in vitro method.Buffers:a. External buffer: 10 mM...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
1/6/2025
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585705(US11530213, Example 26 | 8-chloro-1-(2,6-dichlorop...)
Affinity DataIC50: 31nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585736(US11530213, Example 57 | 8-chloro-1-(2,6-dichlorop...)
Affinity DataIC50: 32nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585711(US11530213, Example 32 | 8-chloro-1-(2,6-dichloro-...)
Affinity DataIC50: 33nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585745(US11530213, Example 66)
Affinity DataIC50: 34nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585714(US11530213, Example 35 | 5-((2-(1H-imidazol-4- yl)...)
Affinity DataIC50: 35nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585691(US11530213, Example 12 | 8-chloro-1-(2,6-dichlorop...)
Affinity DataIC50: 36nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585765(US11530213, Example 86)
Affinity DataIC50: 37nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585707(US11530213, Example 28 | 8-chloro-1-(2,6-dichlorop...)
Affinity DataIC50: 39nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585770(US11530213, Example 91)
Affinity DataIC50: 40nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585730(US11530213, Example 51 | 8-chloro-1-(2,6-dichlorop...)
Affinity DataIC50: 41nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585728(US11530213, Example 49 | 8-chloro-1-(2,6-dichlorop...)
Affinity DataIC50: 42nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585772(US11530213, Example 93)
Affinity DataIC50: 46nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585771(US11530213, Example 92)
Affinity DataIC50: 47nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM695826(US12084442, Example 19 | N-(3-(8-Chloro-1-(2,6-dic...)
Affinity DataIC50: 50nMAssay Description:The GIRK1/4 activity of a compound according to the present invention was assessed by the following in vitro method.Buffers:a. External buffer: 10 mM...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
1/6/2025
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM695827(US12084442, Example 20 | 8-Chloro-1-(2,6-dichloro-...)
Affinity DataIC50: 50nMAssay Description:The GIRK1/4 activity of a compound according to the present invention was assessed by the following in vitro method.Buffers:a. External buffer: 10 mM...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
1/6/2025
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585693(US11530213, Example 14 | 8-chloro-1-(2,6-dichlorop...)
Affinity DataIC50: 52nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
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TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585734(US11530213, Example 55 | 3-chloro-2-(8-chloro-2- c...)
Affinity DataIC50: 54nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585723(US11530213, Example 44 | 3,5-dichloro-4-(8-chloro-...)
Affinity DataIC50: 56nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585726(US11530213, Example 47 | 8-chloro-1-(2,6-dichlorop...)
Affinity DataIC50: 59nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585696(US11530213, Example 17 | 3-((8-chloro-1-(2,6- dich...)
Affinity DataIC50: 60nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
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TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM695812(US12084442, Example 5 | 2-((8-Chloro-1-(2,6-dichlo...)
Affinity DataIC50: 60nMAssay Description:The GIRK1/4 activity of a compound according to the present invention was assessed by the following in vitro method.Buffers:a. External buffer: 10 mM...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
1/6/2025
Entry Details
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TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM695820(US12084442, Example 13 | (S)-3-((8-Chloro-1-(2,6-d...)
Affinity DataIC50: 60nMAssay Description:The GIRK1/4 activity of a compound according to the present invention was assessed by the following in vitro method.Buffers:a. External buffer: 10 mM...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
1/6/2025
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585740(US11530213, Example 61)
Affinity DataIC50: 68nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
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TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM585753(US11530213, Example 74)
Affinity DataIC50: 69nMAssay Description:Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2023
Entry Details
Go to US Patent

TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM695814(US12084442, Example 7 | (R)-3-((8-Chloro-1-(2,6-di...)
Affinity DataIC50: 70nMAssay Description:The GIRK1/4 activity of a compound according to the present invention was assessed by the following in vitro method.Buffers:a. External buffer: 10 mM...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
1/6/2025
Entry Details
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TargetG protein-activated inward rectifier potassium channel 1/4(Human)
Northwest Agriculture & Forestry University

Curated by ChEMBL
LigandPNGBDBM695815(US12084442, Example 8 | (S)-3-((8-Chloro-1-(2,6-di...)
Affinity DataIC50: 70nMAssay Description:The GIRK1/4 activity of a compound according to the present invention was assessed by the following in vitro method.Buffers:a. External buffer: 10 mM...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
1/6/2025
Entry Details
Go to US Patent

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