Compile Data Set for Download or QSAR
Report error Found 271 Enz. Inhib. hit(s) with Target = 'Estrogen receptor [D538G]'
TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263225(US9708370, DBG-145p)
Affinity DataEC50:  809nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263226(US9708370, DBG-168-8p)
Affinity DataEC50:  514nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263222(US9708370, DBG-175p)
Affinity DataEC50:  8.53E+3nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50394994(CHEMBL2163484 | US9708370, DBG-178p)
Affinity DataEC50:  1.57E+4nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50395003(CHEMBL2163476 | US9708370, DBG-188p)
Affinity DataEC50:  808nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50395001(CHEMBL2163478 | US9708370, DBG-253-1)
Affinity DataEC50:  2.77E+3nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50395000(CHEMBL2163479 | US9708370, DBG-253-2)
Affinity DataEC50:  1.95E+4nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50394999(CHEMBL2163480 | US9708370, DBG-253-3)
Affinity DataEC50:  1.34E+3nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM254027(US9708370, DBG-253-4)
Affinity DataEC50:  4.28E+3nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50394998(CHEMBL2163481 | US9708370, DBG-253-5)
Affinity DataEC50:  3.74E+3nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50394997(CHEMBL2163482 | US9708370, DBG-253-6)
Affinity DataEC50:  723nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50394996(CHEMBL2163348 | US9708370, DBG-253-7)
Affinity DataEC50:  771nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50394995(CHEMBL2163483 | US9708370, DBG-253-8)
Affinity DataEC50:  3.25E+3nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263216(US9708370, DBG-253-9)
Affinity DataEC50:  1.61E+4nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263217(US9708370, DBG-253-10)
Affinity DataEC50:  465nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263218(US9708370, DBG-253-11)
Affinity DataEC50:  729nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263219(US9708370, DBG-253-12)
Affinity DataEC50:  1.64E+3nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263220(US9708370, DBG-253-13)
Affinity DataEC50:  5.49E+3nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50395002(CHEMBL2163477 | US9708370, DBG-201-A)
Affinity DataEC50:  1.20E+3nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263227(US9708370, GHRP-6)
Affinity DataEC50:  3.65nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263669(5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...)
Affinity DataIC50: 4nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263674(US9714221, Example 11)
Affinity DataIC50: 4nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263692(US9714221, Example 29)
Affinity DataIC50: 4nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263673(6-(2-fluoro- 4-hydroxy- phenyl)-5- [4-[(3S)-1- (3-...)
Affinity DataIC50: 5nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263691(6- (benzofuran- 5-yl)-5- [4-[(3S)-1- (3- fluoropro...)
Affinity DataIC50: 5nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263892(5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...)
Affinity DataIC50: 6nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50370294(Examorelin | HEXARELIN | US9708370, Hexareline)
Affinity DataIC50: 6.08nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2018
Entry Details
Go to US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263719(6-(1,3- benzoxazol- 5-yl)-5-[4- [(3S)-1-(3- fluoro...)
Affinity DataIC50: 8nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263686(6-(2- chloro-4- methyl- phenyl)-5- [4-[(3S)-1- (3-...)
Affinity DataIC50: 9nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263690(6-(4- ethoxy-2- methyl- phenyl)-5- [4-[(3S)-1- (3-...)
Affinity DataIC50: 10nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263712(6-(2,3- dihydro- 1,4- benzodioxin-6-yl)-5- [4-[(3S...)
Affinity DataIC50: 11nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263683(5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...)
Affinity DataIC50: 12nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263755(6-(2- chloro-4- methoxy- phenyl)-5- [4-[(3S)-1- (3...)
Affinity DataIC50: 12nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263706(6-(2- chloro-4- ethoxy- phenyl)-5- [4-[(3S)-1- (3-...)
Affinity DataIC50: 14nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263671(6-(2- chloro-3- fluoro- phenyl)-5- [4-[(3S)-1- (3-...)
Affinity DataIC50: 15nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263677(5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...)
Affinity DataIC50: 15nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
Go to US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263707(5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...)
Affinity DataIC50: 16nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
Go to US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263675(5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...)
Affinity DataIC50: 18nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263697(6-(6- ethoxy-3- pyridyl)-5- [4-[(3S)-1- (3- fluoro...)
Affinity DataIC50: 18nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263764(6-(2,2- dimethyl- 3H- benzo- furan-5-yl)-5- [4-[(3...)
Affinity DataIC50: 18nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263893(5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...)
Affinity DataIC50: 18nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
Go to US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263676(6-(4- chloro-3- methyl- phenyl)-5- [4-[(3S)-1- (3-...)
Affinity DataIC50: 19nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263694(6-(2,3- dimethyl- phenyl)-5-[4- [(3S)-1-(3- fluoro...)
Affinity DataIC50: 19nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263743(5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...)
Affinity DataIC50: 19nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263672(US9714221, Example 36 | US9714221, Example 9)
Affinity DataIC50: 20nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263693(5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...)
Affinity DataIC50: 20nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263847(6-(2,2-dimethylindolin-5-yl)-5-[4-[(3S)-1-(3-fluor...)
Affinity DataIC50: 20nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263668(6-(2- chloro-4- fluoro- phenyl)-5- [4-[(3S)-1- (3-...)
Affinity DataIC50: 21nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
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TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263709(6-(4- ethoxy-2- methyl- phenyl)-1- fluoro-5-[4- [(...)
Affinity DataIC50: 21nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
Go to US Patent

TargetEstrogen receptor [D538G](Human)
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM263900(6-[2,3- difluoro-4- (1-piperidyl)- phenyl]-5- [4-[...)
Affinity DataIC50: 21nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
Go to US Patent

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