Compile Data Set for Download or QSAR
Report error Found 130 Enz. Inhib. hit(s) with Target = 'Disks large homolog 4'
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252827(N-Cyclohexylethyl-ETAV | CHEMBL493688)
Affinity DataKi:  450nMAssay Description:Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252827(N-Cyclohexylethyl-ETAV | CHEMBL493688)
Affinity DataKi:  630nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339567((2S,5S,8S,11S)-11-(2-carboxyethyl)-14-cyclohexyl-8...)
Affinity DataKi:  630nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339545((4S,7S,10S,13S)-4-(2-carboxyethyl)-10-(carboxymeth...)
Affinity DataKi:  750nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252827(N-Cyclohexylethyl-ETAV | CHEMBL493688)
Affinity DataKi:  940nMAssay Description:Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252828(N-(Naphthalene-2-yl)ethyl-ETAV | CHEMBL493689)
Affinity DataKi:  950nMAssay Description:Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252754(N-(3,4-Difluorophenyl)propyl-ETAV | CHEMBL538410)
Affinity DataKi:  980nMAssay Description:Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252828(N-(Naphthalene-2-yl)ethyl-ETAV | CHEMBL493689)
Affinity DataKi:  1.00E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252826(N-Cyclohexylmethyl-ETAV | CHEMBL494486)
Affinity DataKi:  1.00E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252754(N-(3,4-Difluorophenyl)propyl-ETAV | CHEMBL538410)
Affinity DataKi:  1.00E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339569((2S,5S,8S,11S)-11-(2-carboxyethyl)-14-(3,4-dichlor...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252753(N-(3,4-Dichlorophenyl)propyl-ETAV | CHEMBL495100)
Affinity DataKi:  1.10E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339568((2S,5S,8S,11S)-11-(2-carboxyethyl)-8-((R)-1-hydrox...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339548((2S,5S,8S,11S)-11-(2-carboxyethyl)-5-(carboxymethy...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339555((2S,5S,8S,11S)-11-(2-carboxyethyl)-14-cycloheptyl-...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252826(N-Cyclohexylmethyl-ETAV | CHEMBL494486)
Affinity DataKi:  1.30E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339552((3S,6S,9S,12S)-1-(bicyclo[2.2.1]heptan-2-yl)-3-(2-...)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339554((3S,6S,9S,12S)-3-(2-carboxyethyl)-1-cycloheptyl-6-...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339553((2S,5S,8S,11S)-14-(bicyclo[2.2.1]heptan-2-yl)-11-(...)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252715(N-Phenylethyl-ETAV | CHEMBL494895)
Affinity DataKi:  1.60E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339547((2S,5S,8S,11S)-11-(2-carboxyethyl)-5-(carboxymethy...)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339556((2S,5S,8S,11S)-11-(2-carboxyethyl)-8-((R)-1-hydrox...)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252752(N-Phenylpropyl-ETAV | CHEMBL495099)
Affinity DataKi:  2.10E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50253144(KSG-LDTKNYKQTSV | CHEMBL505051)
Affinity DataKi:  2.10E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ3 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339551((S)-2-[(S)-2-((2S,3R)-2-{(S)-2-[(Adamantan-1-ylmet...)
Affinity DataKi:  2.10E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252713(FETAV | CHEMBL492642)
Affinity DataKi:  2.30E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252753(N-(3,4-Dichlorophenyl)propyl-ETAV | CHEMBL495100)
Affinity DataKi:  2.40E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252752(N-Phenylpropyl-ETAV | CHEMBL495099)
Affinity DataKi:  3.10E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339539((4S,7S,10S,13S)-10-(carboxymethyl)-1-cyclohexyl-7-...)
Affinity DataKi:  3.60E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252825(N-Butyl-ETAV | CHEMBL494485)
Affinity DataKi:  4.00E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50253143(KSG-YEKLSSIESDV | CHEMBL445253)
Affinity DataKi:  4.10E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252824(N-Propyl-ETAV | CHEMBL494287)
Affinity DataKi:  4.20E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339557((2S,5S,8S,11S)-11-(2-carboxyethyl)-8-((R)-1-hydrox...)
Affinity DataKi:  4.20E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252715(N-Phenylethyl-ETAV | CHEMBL494895)
Affinity DataKi:  4.40E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50253145(YGRKKRRQRRR-KLSSIESDV | CHEMBL502630)
Affinity DataKi:  4.40E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339546((4S,7S,10S,13S)-4-(3-amino-3-oxopropyl)-10-(carbox...)
Affinity DataKi:  4.40E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50253145(YGRKKRRQRRR-KLSSIESDV | CHEMBL502630)
Affinity DataKi:  4.40E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339558((2S,5S,8S,11S)-11-(2-carboxyethyl)-8-((R)-1-hydrox...)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252714(N-Benzyl-ETAV | CHEMBL492643)
Affinity DataKi:  5.20E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252713(FETAV | CHEMBL492642)
Affinity DataKi:  6.30E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252753(N-(3,4-Dichlorophenyl)propyl-ETAV | CHEMBL495100)
Affinity DataKi:  6.70E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ3 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339551((S)-2-[(S)-2-((2S,3R)-2-{(S)-2-[(Adamantan-1-ylmet...)
Affinity DataKi:  6.70E+3nMAssay Description:Inhibition of PSD-95 PDZ3 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252824(N-Propyl-ETAV | CHEMBL494287)
Affinity DataKi:  7.00E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50253143(KSG-YEKLSSIESDV | CHEMBL445253)
Affinity DataKi:  7.00E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ1-2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252714(N-Benzyl-ETAV | CHEMBL492643)
Affinity DataKi:  7.20E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252754(N-(3,4-Difluorophenyl)propyl-ETAV | CHEMBL538410)
Affinity DataKi:  7.80E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ3 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339538((4S,7S,10S,13S)-1-cyclohexyl-7-((R)-1-hydroxyethyl...)
Affinity DataKi:  8.10E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339569((2S,5S,8S,11S)-11-(2-carboxyethyl)-14-(3,4-dichlor...)
Affinity DataKi:  8.30E+3nMAssay Description:Inhibition of PSD-95 PDZ3 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252825(N-Butyl-ETAV | CHEMBL494485)
Affinity DataKi:  8.40E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDisks large homolog 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339556((2S,5S,8S,11S)-11-(2-carboxyethyl)-8-((R)-1-hydrox...)
Affinity DataKi:  8.80E+3nMAssay Description:Inhibition of PSD-95 PDZ3 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
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