Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with Target = 'Diacylglycerol kinase 1'
TargetDiacylglycerol kinase 1(Fruit fly)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50206506(9-beta-D-arabinofuranosylguanosine | CHEMBL240933)
Affinity DataIC50: 1.33E+5nMAssay Description:Inhibition of Drosophila melanogaster dGK assessed as [methyl-3H]dThd phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2012
Entry Details Article
PubMed
TargetDiacylglycerol kinase 1(Fruit fly)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50206501(9-(2'-O-octanoyl-beta-D-arabinofuranosyl)guanine |...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of Drosophila melanogaster dGK assessed as [methyl-3H]dThd phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2012
Entry Details Article
PubMed
TargetDiacylglycerol kinase 1(Fruit fly)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50206500(N2-octanoyl-9-(2'-O-octanoyl-beta-D-arabinofuranos...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of Drosophila melanogaster dGK assessed as [methyl-3H]dThd phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2012
Entry Details Article
PubMed
TargetDiacylglycerol kinase 1(Fruit fly)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50206499(9-(2'-O-pentanoyl-beta-D-arabinofuranosyl)guanine ...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of Drosophila melanogaster dGK assessed as [methyl-3H]dThd phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2012
Entry Details Article
PubMed