Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with Target = 'DNA-dependent protein kinase catalytic subunit/Serine/threonine-protein kinase mTOR'
LigandPNGBDBM36409(CID24905147 | 2-(4-amino-1-isopropyl-1H-pyrazolo[3...)
Affinity DataIC50: 410nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2011
Entry Details Article
PubMed
LigandPNGBDBM36410(CID24905148 | 1-cyclopentyl-3-(H-imidazo[1,2-a]pyr...)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2011
Entry Details Article
PubMed