Report error Found 2972 Enz. Inhib. hit(s) with Target = 'DNA topoisomerase'
Affinity DataEC50: 580nMAssay Description:In vitro activity against topoisomerase-1 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 430nMAssay Description:In vitro activity against topoisomerase-1 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 9.50E+3nMAssay Description:In vitro activity against topoisomerase-1 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 300nMAssay Description:In vitro activity against topoisomerase-1 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:In vitro activity against topoisomerase-1 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 580nMAssay Description:In vitro activity against topoisomerase-1 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:In vitro activity against topoisomerase-1 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 270nMAssay Description:In vitro activity against topoisomerase-1 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 700nMAssay Description:In vitro activity against topoisomerase-1 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 270nMAssay Description:In vitro activity against topoisomerase-1 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 1.20E+3nMAssay Description:In vitro activity against topoisomerase-1 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 350nMAssay Description:In vitro activity against topoisomerase-1 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 52nMAssay Description:In vitro activity against topoisomerase-1 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 3.00E+3nMAssay Description:In vitro activity against topoisomerase-1 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 170nMAssay Description:In vitro activity against topoisomerase-1 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 90nMAssay Description:In vitro activity against topoisomerase-1 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+3nMAssay Description:In vitro activity against topoisomerase-1 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 550nMAssay Description:In vitro activity against topoisomerase-1 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro activity against topoisomerase-1 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 160nMAssay Description:In vitro activity against topoisomerase-1 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 3.50E+3nMAssay Description:In vitro activity against topoisomerase-1 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 250nMAssay Description:In vitro activity against topoisomerase-1 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 2.80E+3nMAssay Description:In vitro activity against topoisomerase-1 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 70nMAssay Description:In vitro activity against topoisomerase-1 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 480nMAssay Description:In vitro activity against topoisomerase-1 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 360nMAssay Description:In vitro activity against topoisomerase-1 mediated cleavage of supercoiled pBR322 plasmid DNAMore data for this Ligand-Target Pair
Affinity DataEC50: 650nMAssay Description:In vitro inhibition of Topoisomerase I-mediated DNA cleavage using supercoiled pBR322 plasmid DNA.More data for this Ligand-Target Pair
Affinity DataEC50: 51nMAssay Description:In vitro inhibition of Topoisomerase I-mediated DNA cleavage using supercoiled pBR322 plasmid DNA.More data for this Ligand-Target Pair
Affinity DataEC50: 210nMAssay Description:In vitro inhibition of Topoisomerase I-mediated DNA cleavage using supercoiled pBR322 plasmid DNA.More data for this Ligand-Target Pair
TargetDNA topoisomerase 2-binding protein 1(Human)
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >5.00E+4nMAssay Description:In vitro inhibition of Topoisomerase II-mediated DNA cleavage using supercoiled pBR322 plasmid DNA.More data for this Ligand-Target Pair
TargetDNA topoisomerase 2-binding protein 1(Human)
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >5.00E+4nMAssay Description:In vitro inhibition of Topoisomerase II-mediated DNA cleavage using supercoiled pBR322 plasmid DNA.More data for this Ligand-Target Pair
Affinity DataEC50: 570nMAssay Description:In vitro inhibition of Topoisomerase I-mediated DNA cleavage using supercoiled pBR322 plasmid DNA.More data for this Ligand-Target Pair
Affinity DataEC50: 160nMAssay Description:In vitro inhibition of Topoisomerase I-mediated DNA cleavage using supercoiled pBR322 plasmid DNA.More data for this Ligand-Target Pair
TargetDNA topoisomerase 2-binding protein 1(Human)
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >5.00E+4nMAssay Description:In vitro inhibition of Topoisomerase II-mediated DNA cleavage using supercoiled pBR322 plasmid DNA.More data for this Ligand-Target Pair
TargetDNA topoisomerase 2-binding protein 1(Human)
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >5.00E+4nMAssay Description:In vitro inhibition of Topoisomerase II-mediated DNA cleavage using supercoiled pBR322 plasmid DNA.More data for this Ligand-Target Pair
Affinity DataEC50: 1.10E+3nMAssay Description:In vitro inhibition of Topoisomerase I-mediated DNA cleavage using supercoiled pBR322 plasmid DNA.More data for this Ligand-Target Pair
TargetDNA topoisomerase 2-binding protein 1(Human)
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >5.00E+4nMAssay Description:In vitro inhibition of Topoisomerase II-mediated DNA cleavage using supercoiled pBR322 plasmid DNA.More data for this Ligand-Target Pair
TargetDNA topoisomerase 2-binding protein 1(Human)
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >5.00E+4nMAssay Description:In vitro inhibition of Topoisomerase II-mediated DNA cleavage using supercoiled pBR322 plasmid DNA.More data for this Ligand-Target Pair
Affinity DataEC50: 230nMAssay Description:In vitro inhibition of Topoisomerase I-mediated DNA cleavage using supercoiled pBR322 plasmid DNA.More data for this Ligand-Target Pair
Affinity DataEC50: 490nMAssay Description:In vitro inhibition of Topoisomerase I-mediated DNA cleavage using supercoiled pBR322 plasmid DNA.More data for this Ligand-Target Pair
TargetDNA topoisomerase 2-binding protein 1(Human)
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >5.00E+4nMAssay Description:In vitro inhibition of Topoisomerase II-mediated DNA cleavage using supercoiled pBR322 plasmid DNA.More data for this Ligand-Target Pair
Affinity DataEC50: 510nMAssay Description:In vitro inhibition of Topoisomerase I-mediated DNA cleavage using supercoiled pBR322 plasmid DNA.More data for this Ligand-Target Pair
TargetDNA topoisomerase 2-binding protein 1(Human)
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >5.00E+4nMAssay Description:In vitro inhibition of Topoisomerase II-mediated DNA cleavage using supercoiled pBR322 plasmid DNA.More data for this Ligand-Target Pair
TargetDNA topoisomerase 2-binding protein 1(Human)
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >5.00E+4nMAssay Description:In vitro inhibition of Topoisomerase II-mediated DNA cleavage using supercoiled pBR322 plasmid DNA.More data for this Ligand-Target Pair
Affinity DataEC50: 90nMAssay Description:In vitro inhibition of Topoisomerase I-mediated DNA cleavage using supercoiled pBR322 plasmid DNA.More data for this Ligand-Target Pair
TargetDNA topoisomerase 2-binding protein 1(Human)
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >5.00E+4nMAssay Description:In vitro inhibition of Topoisomerase II-mediated DNA cleavage using supercoiled pBR322 plasmid DNA.More data for this Ligand-Target Pair
Affinity DataEC50: 1.90E+3nMAssay Description:In vitro inhibition of Topoisomerase I-mediated DNA cleavage using supercoiled pBR322 plasmid DNA.More data for this Ligand-Target Pair
TargetDNA topoisomerase 2-binding protein 1(Human)
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >5.00E+4nMAssay Description:In vitro inhibition of Topoisomerase II-mediated DNA cleavage using supercoiled pBR322 plasmid DNA.More data for this Ligand-Target Pair
TargetDNA topoisomerase 2-binding protein 1(Human)
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: >5.00E+4nMAssay Description:In vitro inhibition of Topoisomerase II-mediated DNA cleavage using supercoiled pBR322 plasmid DNA.More data for this Ligand-Target Pair
Affinity DataEC50: 55nMAssay Description:In vitro inhibition of Topoisomerase I-mediated DNA cleavage using supercoiled pBR322 plasmid DNA.More data for this Ligand-Target Pair








































