Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with Target = 'Cytochrome P450 4F12'
TargetCytochrome P450 4F12(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106737(N-(4-butyl-2-methylphenyl)-N'-hydroxyimidoformamid...)
Affinity DataIC50: 155nMAssay Description:Inhibition of human recombinant CYP4F12 using Luciferin ME EGE as substrate incubated for 30 mins in presence of NADPH by luminescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetCytochrome P450 4F12(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50609596(CHEMBL5272822)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human recombinant CYP4F12 using Luciferin ME EGE as substrate incubated for 30 mins in presence of NADPH by luminescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetCytochrome P450 4F12(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50527963(CHEMBL4557940)
Affinity DataIC50: 5.70E+4nMAssay Description:Inhibition of recombinant human CYP4F12 expressed in baculovirus infected insect cells using Luc-BE as substrate preincubated with NADPH for 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetCytochrome P450 4F12(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50527963(CHEMBL4557940)
Affinity DataIC50: 1.67E+5nMAssay Description:Inhibition of recombinant human CYP4F12 expressed in baculovirus infected insect cells using Luc-BE as substrate after 10 mins in presence of NADPH b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetCytochrome P450 4F12(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50527962(CHEMBL4442292)
Affinity DataIC50: 7.78E+5nMAssay Description:Inhibition of recombinant human CYP4F12 expressed in baculovirus infected insect cells using Luc-BE as substrate preincubated with NADPH for 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetCytochrome P450 4F12(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50527962(CHEMBL4442292)
Affinity DataIC50: 1.18E+6nMAssay Description:Inhibition of recombinant human CYP4F12 expressed in baculovirus infected insect cells using Luc-BE as substrate after 10 mins in presence of NADPH b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed