Report error Found 11 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 3 [34-140]'
Affinity DataIC50: 35nMAssay Description:The bromodomain binding assays were performed by Reaction Biology Corp., Malvern, Pa., USA (www.reactionbiology.com). The BET binding assays were con...More data for this Ligand-Target Pair
Affinity DataKd: >3.00E+3nMAssay Description:T7 phage strains displaying bromodomains were grown in parallel in 24-well blocks in an E. coli host derived from the BL21 strain. E. coli were grown...More data for this Ligand-Target Pair
Affinity DataIC50: 2.97E+4nMAssay Description:The binding inhibitory effect of the compounds of the present invention on the BRD3 protein among the BET proteins was tested as follows and confirme...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 3.58E+4nMAssay Description:The binding inhibitory effect of the compounds of the present invention on the BRD3 protein among the BET proteins was tested as follows and confirme...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 4.90E+4nMAssay Description:The binding inhibitory effect of the compounds of the present invention on the BRD3 protein among the BET proteins was tested as follows and confirme...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 5.15E+4nMAssay Description:The binding inhibitory effect of the compounds of the present invention on the BRD3 protein among the BET proteins was tested as follows and confirme...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 6.11E+4nMAssay Description:The binding inhibitory effect of the compounds of the present invention on the BRD3 protein among the BET proteins was tested as follows and confirme...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 8.48E+4nMAssay Description:The binding inhibitory effect of the compounds of the present invention on the BRD3 protein among the BET proteins was tested as follows and confirme...More data for this Ligand-Target Pair
Affinity DataIC50: 9.87E+4nMAssay Description:The binding inhibitory effect of the compounds of the present invention on the BRD3 protein among the BET proteins was tested as follows and confirme...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.61E+5nMAssay Description:The binding inhibitory effect of the compounds of the present invention on the BRD3 protein among the BET proteins was tested as follows and confirme...More data for this Ligand-Target Pair
Affinity DataIC50: 2.34E+7nMAssay Description:The binding inhibitory effect of the compounds of the present invention on the BRD3 protein among the BET proteins was tested as follows and confirme...More data for this Ligand-Target Pair
