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Report error Found 10 Enz. Inhib. hit(s) with Target = 'Bifunctional peptidase and (3S)-lysyl hydroxylase JMJD7'
TargetBifunctional peptidase and (3S)-lysyl hydroxylase JMJD7(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50571209(CHEMBL4846929)
Affinity DataKd:  1.18E+3nMAssay Description:Binding affinity to N-terminal His-tagged human JMJD7 (1 to 316 residues) expressed in Escherichia coli BL21 (DE3) measured by MST assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBifunctional peptidase and (3S)-lysyl hydroxylase JMJD7(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50571209(CHEMBL4846929)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of N-terminal His-tagged human JMJD7 (1 to 316 residues) expressed in Escherichia coli BL21 (DE3) using peptide substrate DRG (16 to 30) m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBifunctional peptidase and (3S)-lysyl hydroxylase JMJD7(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50571209(CHEMBL4846929)
Affinity DataIC50: 6.62E+3nMAssay Description:Inhibition of N-terminal His-tagged human JMJD7 (1 to 316 residues) expressed in Escherichia coli BL21 (DE3) luciferase based succinate-gloTM JmjC de...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBifunctional peptidase and (3S)-lysyl hydroxylase JMJD7(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM16111(2-{[2-fluoro-4-(3-methoxyphenyl)phenyl]carbamoyl}c...)
Affinity DataIC50: 7.16E+3nMAssay Description:Inhibition of N-terminal His-tagged human JMJD7 (1 to 316 residues) expressed in Escherichia coli BL21 (DE3) luciferase based succinate-gloTM JmjC de...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBifunctional peptidase and (3S)-lysyl hydroxylase JMJD7(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM40249(5-(1,3-benzothiazol-2-yl)-N-propylthiophene-2-carb...)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of N-terminal His-tagged human JMJD7 (1 to 316 residues) expressed in Escherichia coli BL21 (DE3) luciferase based succinate-gloTM JmjC de...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBifunctional peptidase and (3S)-lysyl hydroxylase JMJD7(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50571208(CHEMBL4862698)
Affinity DataIC50: 2.62E+4nMAssay Description:Inhibition of N-terminal His-tagged human JMJD7 (1 to 316 residues) expressed in Escherichia coli BL21 (DE3) luciferase based succinate-gloTM JmjC de...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBifunctional peptidase and (3S)-lysyl hydroxylase JMJD7(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50339142(rac-7-(phenyl(pyridin-2-ylamino)methyl)quinolin-8-...)
Affinity DataIC50: 3.16E+4nMAssay Description:Inhibition of N-terminal His-tagged human JMJD7 (1 to 316 residues) expressed in Escherichia coli BL21 (DE3) luciferase based succinate-gloTM JmjC de...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBifunctional peptidase and (3S)-lysyl hydroxylase JMJD7(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50571207(CHEMBL1081780)
Affinity DataIC50: 3.32E+4nMAssay Description:Inhibition of N-terminal His-tagged human JMJD7 (1 to 316 residues) expressed in Escherichia coli BL21 (DE3) luciferase based succinate-gloTM JmjC de...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBifunctional peptidase and (3S)-lysyl hydroxylase JMJD7(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM251460(US9452998, 9)
Affinity DataIC50: 5.01E+4nMAssay Description:Inhibition of N-terminal His-tagged human JMJD7 (1 to 316 residues) expressed in Escherichia coli BL21 (DE3) luciferase based succinate-gloTM JmjC de...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBifunctional peptidase and (3S)-lysyl hydroxylase JMJD7(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50576306(CHEMBL4849961)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of JMJD7 (unknown origin) by Succinate-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed