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Report error Found 39 Enz. Inhib. hit(s) with Target = 'Baculoviral IAP repeat-containing protein 5'
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209181(3-(3-bromophenyl)quinoline | CHEMBL397092)
Affinity DataKd:  1.00E+4nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209185(6-(5-chloro-2-hydroxyphenyl)-4-(2-chloro-5-(triflu...)
Affinity DataKd:  520nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM26673(CHEMBL391586 | 6-(5-bromo-2-hydroxyphenyl)-2-oxo-4...)
Affinity DataKd:  5.00E+3nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209197(6-(5-cyclohexyl-2-hydroxyphenyl)-4-(2,5-dichloroph...)
Affinity DataKd:  2.98E+3nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209204(N-(5-chloro-3-(4-(2-chloro-5-(trifluoromethyl)phen...)
Affinity DataKd:  76nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209180(6-(5-bromo-2-hydroxyphenyl)-4-(2-chloro-5-(trifluo...)
Affinity DataKd:  490nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209201(N-(5-chloro-3-(4-(2-chloro-5-(trifluoromethyl)phen...)
Affinity DataKd:  48nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209187(N-(5-chloro-3-(4-(2-chloro-5-(trifluoromethyl)phen...)
Affinity DataKd:  440nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209194(N-(5-chloro-3-(4-(2-chloro-5-(trifluoromethyl)phen...)
Affinity DataKd:  37nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209205(N-(4-methylpyridin-2-yl)piperidine-4-carboxamide |...)
Affinity DataKd:  1.30E+5nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209184(4-(2,5-dichlorophenyl)-6-(2-hydroxy-5-isobutylphen...)
Affinity DataKd:  7.56E+3nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209199(6-(5-bromo-2-hydroxyphenyl)-4-(2,4-dimethylphenyl)...)
Affinity DataKd:  700nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209206((2-ethylbenzofuran-3-yl)(4-hydroxy-3,5-diiodopheny...)
Affinity DataKd:  8.00E+3nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM26673(CHEMBL391586 | 6-(5-bromo-2-hydroxyphenyl)-2-oxo-4...)
Affinity DataKd:  5.70E+3nMAssay Description:Inhibition of survivinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209209(6-(5-bromo-2-hydroxyphenyl)-4-(2,5-dichlorophenyl)...)
Affinity DataKd:  800nMAssay Description:Inhibition of survivinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50550143(CHEMBL4793552)
Affinity DataKd:  34nMAssay Description:Binding affinity to recombinant full length N-terminal GST-tagged human survivin expressed in Escherichia coli BL21 incubated for 1 hr under shaking ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209194(N-(5-chloro-3-(4-(2-chloro-5-(trifluoromethyl)phen...)
Affinity DataKd:  44nMAssay Description:Binding affinity to recombinant full length N-terminal GST-tagged human survivin expressed in Escherichia coli BL21 incubated for 1 hr under shaking ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50573761(CHEMBL4862376)
Affinity DataKd:  4.27E+3nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 assessed as dissociation constant measured by Surface plasmon resonanceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50631616(CHEMBL4637348)
Affinity DataKd:  240nMAssay Description:Binding affinity to Survivin (unknown origin) assessed as dissociation constant by fluorogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209188(6-(2-hydroxyphenyl)-2-oxo-4-phenyl-1,2-dihydropyri...)
Affinity DataKd:  7.50E+4nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209208(N-(5-chloro-3-(4-(2-chloro-5-(trifluoromethyl)phen...)
Affinity DataKd:  86nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209190(N-(5-chloro-3-(4-(2-chloro-5-(trifluoromethyl)phen...)
Affinity DataKd:  60nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209202(N-(5-chloro-3-(4-(2-chloro-5-(trifluoromethyl)phen...)
Affinity DataKd:  880nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209193(N-(5-chloro-3-(4-(2-chloro-5-(trifluoromethyl)phen...)
Affinity DataKd:  64nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209203(N-(5-chloro-3-(4-(2-chloro-5-(trifluoromethyl)phen...)
Affinity DataKd:  620nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209192(6-(5-bromo-2-hydroxyphenyl)-4-(2,5-dimethylphenyl)...)
Affinity DataKd:  1.17E+3nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209196(6-(5-bromo-2-hydroxy-phenyl)-4-(4-chloro-biphenyl-...)
Affinity DataKd: >4.30E+3nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209191(6-(5-cyclopentyl-2-hydroxyphenyl)-4-(2,5-dichlorop...)
Affinity DataKd:  510nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209182(N-(5-chloro-3-(4-(2-chloro-5-(trifluoromethyl)phen...)
Affinity DataKd:  100nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209210(N-(5-chloro-3-(4-(2-chloro-5-(trifluoromethyl)phen...)
Affinity DataKd:  530nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209195(4-(2,5-dichloro-phenyl)-6-(4-hydroxy-biphenyl-3-yl...)
Affinity DataKd:  700nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209207(tert-butyl 4-((5-chloro-3-(4-(2-chloro-5-(trifluor...)
Affinity DataKd:  260nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209209(6-(5-bromo-2-hydroxyphenyl)-4-(2,5-dichlorophenyl)...)
Affinity DataKd:  810nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209198(N-(5-chloro-3-(4-(2-chloro-5-(trifluoromethyl)phen...)
Affinity DataKd:  200nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209183(N-(5-chloro-3-(4-(2-chloro-5-(trifluoromethyl)phen...)
Affinity DataKd:  220nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50024762(CHEMBL395633)
Affinity DataKd: <1.00E+4nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50024761(CHEMBL232200)
Affinity DataKd: <1.00E+4nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50209186(1-(4-chlorophenyl)-1H-indole | CHEMBL233218)
Affinity DataKd:  5.00E+3nMAssay Description:Binding affinity to human survivin expressed in Escherichia coli BL21 cells after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBaculoviral IAP repeat-containing protein 5(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50442671(CHEMBL2442083)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of survivin (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed