Compile Data Set for Download or QSAR
Report error Found 1730 Enz. Inhib. hit(s) with Target = 'Alpha-2C adrenergic receptor'
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50218115((R)-2-[1-(3'-nitrobiphenyl-2-yloxy)ethyl]-4,5-dihy...)
Affinity DataEC50:  10nMAssay Description:Agonistic potency at human adrenergic Alpha-2C receptor expressed in CHO cells assessed as forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50055832((1H-Imidazol-2-yl)-(5-methyl-2,3-dihydro-benzo[1,4...)
Affinity DataEC50:  6.60nMAssay Description:Effective concentration at Alpha-2C adrenergic receptor from CHO-C4 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50055835((4-tert-Butyl-3-methoxy-2,6-dimethyl-phenyl)-(1H-i...)
Affinity DataEC50: >5.00E+3nMAssay Description:Effective concentration at Alpha-2C adrenergic receptor from CHO-C4 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM34572(UK 14,304 | SMR000058355 | CHEMBL844 | cid_2435 | ...)
Affinity DataEC50:  3.40nMAssay Description:Effective concentration at Alpha-2C adrenergic receptor from CHO-C4 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50055830((1H-Imidazol-2-yl)-(5-methyl-3,4-dihydro-2H-benzo[...)
Affinity DataEC50:  110nMAssay Description:Effective concentration at Alpha-2C adrenergic receptor from CHO-C4 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50029051(4-[(1R)-2-amino-1-hydroxyethyl]benzene-1,2-diol | ...)
Affinity DataEC50:  794nMAssay Description:Agonistic potency at human adrenergic Alpha-2C receptor expressed in CHO cells assessed as forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50002903(CHEMBL223836)
Affinity DataEC50:  60nMAssay Description:Agonistic potency at human adrenergic Alpha-2C receptor expressed in CHO cells assessed as forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50412250(CHEMBL128168)
Affinity DataEC50:  58nMAssay Description:Agonistic potency at human adrenergic Alpha-2C receptor expressed in CHO cells assessed as forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50417341(CHEMBL397753)
Affinity DataEC50:  741nMAssay Description:Agonistic potency at human adrenergic Alpha-2C receptor expressed in CHO cells assessed as forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50417354(CHEMBL396013)
Affinity DataEC50:  19nMAssay Description:Agonistic potency at human adrenergic Alpha-2C receptor expressed in CHO cells assessed as forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50417353(CHEMBL242265)
Affinity DataEC50:  112nMAssay Description:Agonistic potency at human adrenergic Alpha-2C receptor expressed in CHO cells assessed as forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50002905(CHEMBL373535)
Affinity DataEC50:  50nMAssay Description:Agonistic potency at human adrenergic Alpha-2C receptor expressed in CHO cells assessed as forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50002904(CHEMBL222928)
Affinity DataEC50:  100nMAssay Description:Agonistic potency at human adrenergic Alpha-2C receptor expressed in CHO cells assessed as forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50417350(CHEMBL374584)
Affinity DataEC50:  47nMAssay Description:Agonistic potency at human adrenergic Alpha-2C receptor expressed in CHO cells assessed as forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50180251(1-((S)-2-aminopropyl)-1H-indazol-6-ol | CHEMBL3713...)
Affinity DataEC50:  1.00E+4nMAssay Description:Activity at adrenergic Alpha-2C receptor expressed in rat-mouse hybrid NH108-15 cell by adenylyl cyclase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50415141(CHEMBL576819)
Affinity DataEC50:  2.88E+3nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50415138(CHEMBL576078)
Affinity DataEC50:  25nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50415140(CHEMBL569933)
Affinity DataEC50:  155nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50415139(CHEMBL576623)
Affinity DataEC50:  40nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50415137(CHEMBL570863)
Affinity DataEC50:  63nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50412245(CHEMBL495095)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50417342(CHEMBL1276139)
Affinity DataEC50:  186nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50417344(CHEMBL1276218)
Affinity DataEC50:  40nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50417345(CHEMBL1276219)
Affinity DataEC50:  126nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50218115((R)-2-[1-(3'-nitrobiphenyl-2-yloxy)ethyl]-4,5-dihy...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50417352(CHEMBL1278085)
Affinity DataEC50:  2.51E+3nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50417351(CHEMBL1278084)
Affinity DataEC50:  25nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50417347(CHEMBL385310)
Affinity DataEC50:  93nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50412246(CHEMBL495097)
Affinity DataEC50:  3.55E+3nMAssay Description:Agonist activity at human recombinant adrenergic Alpha-2C receptor expressed in CHO cells assessed as stimulation of extracellular acidificationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50412245(CHEMBL495095)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human recombinant adrenergic Alpha-2C receptor expressed in CHO cells assessed as stimulation of extracellular acidificationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50412244(CHEMBL495096)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human recombinant adrenergic Alpha-2C receptor expressed in CHO cells assessed as stimulation of extracellular acidificationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50412258(CHEMBL451229)
Affinity DataEC50:  21nMAssay Description:Agonist activity at human recombinant adrenergic Alpha-2C receptor expressed in CHO cells assessed as stimulation of extracellular acidificationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50412247(CHEMBL492639)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human recombinant adrenergic Alpha-2C receptor expressed in CHO cells assessed as stimulation of extracellular acidificationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50412248(CHEMBL442815)
Affinity DataEC50:  501nMAssay Description:Agonist activity at human recombinant adrenergic Alpha-2C receptor expressed in CHO cells assessed as stimulation of extracellular acidificationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50412249(CHEMBL493675)
Affinity DataEC50:  126nMAssay Description:Agonist activity at human recombinant adrenergic Alpha-2C receptor expressed in CHO cells assessed as stimulation of extracellular acidificationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50412250(CHEMBL128168)
Affinity DataEC50:  58nMAssay Description:Agonist activity at human recombinant adrenergic Alpha-2C receptor expressed in CHO cells assessed as stimulation of extracellular acidificationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50019646(CHEMBL17860 | lofexidine | 2-(alpha-(2,6-Dichlorop...)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at human adrenoceptor aplha 2C expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50419878(CHEMBL1956195)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human adrenoceptor aplha 2C expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50419879(CHEMBL1956196)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human adrenoceptor aplha 2C expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50419875(CHEMBL1956193)
Affinity DataEC50:  794nMAssay Description:Agonist activity at human adrenoceptor aplha 2C expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50419877(CHEMBL1956194)
Affinity DataEC50:  115nMAssay Description:Agonist activity at human adrenoceptor aplha 2C expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50419881(CHEMBL1956199)
Affinity DataEC50:  9.77E+3nMAssay Description:Agonist activity at human adrenoceptor aplha 2C expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50419882(CHEMBL1956200)
Affinity DataEC50:  316nMAssay Description:Agonist activity at human adrenoceptor aplha 2C expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50419880(CHEMBL1956197)
Affinity DataEC50:  48nMAssay Description:Agonist activity at human adrenoceptor aplha 2C expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50419876(CHEMBL266613)
Affinity DataEC50:  398nMAssay Description:Agonist activity at human adrenoceptor aplha 2C expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50419888(CHEMBL1956202)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human adrenoceptor aplha 2C expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50419873(CHEMBL1956203)
Affinity DataEC50:  79nMAssay Description:Agonist activity at human adrenoceptor aplha 2C expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50419883(CHEMBL1956201)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human adrenoceptor aplha 2C expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50419884(CHEMBL157955)
Affinity DataEC50:  28nMAssay Description:Agonist activity at human adrenoceptor aplha 2C expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2C adrenergic receptor(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50419889(CHEMBL155866)
Affinity DataEC50:  28nMAssay Description:Agonist activity at human adrenoceptor aplha 2C expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
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