Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with Target = 'AP-2 complex subunit sigma'
TargetAP-2 complex subunit sigma(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  24.2nMAssay Description:Displacement of [3H]-DTG from rat sigma2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetAP-2 complex subunit sigma(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50339687(4-(Dimethylamino)-N-(4-(4-(2-(2-fluoroethoxy)pheny...)
Affinity DataKi:  650nMAssay Description:Displacement of [3H]-DTG from rat sigma2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetAP-2 complex subunit sigma(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50339689(4-(2-Fluoroethoxy)-N-(4-(4-(2-methoxyphenyl)-piper...)
Affinity DataKi:  660nMAssay Description:Displacement of [3H]-DTG from rat sigma2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetAP-2 complex subunit sigma(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50339686(4-(2-Fluoroethoxy)-N-(4-(4-(2-(2-fluoroethoxy)phen...)
Affinity DataKi:  794nMAssay Description:Displacement of [3H]-DTG from rat sigma2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetAP-2 complex subunit sigma(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50339688(4-(2-(2-(2-Fluoroethoxy)ethoxy)ethoxy)-N-(4-(4-(2-...)
Affinity DataKi:  1.12E+3nMAssay Description:Displacement of [3H]-DTG from rat sigma2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetAP-2 complex subunit sigma(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50339683(4-(Thiophen-3-yl)-N-(4-(4-(2-(2-fluoroethoxy)pheny...)
Affinity DataKi:  1.32E+3nMAssay Description:Displacement of [3H]-DTG from rat sigma2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetAP-2 complex subunit sigma(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50339691(4-(dimethylamino)-N-(4-(4-(2-methoxyphenyl)piperaz...)
Affinity DataKi:  1.57E+3nMAssay Description:Displacement of [3H]-DTG from rat sigma2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetAP-2 complex subunit sigma(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50339684(4-(2-Fluoroethyl)-N-(4-(4-(2-(2-Fluoroethoxy)pheny...)
Affinity DataKi:  2.02E+3nMAssay Description:Displacement of [3H]-DTG from rat sigma2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetAP-2 complex subunit sigma(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50339690(4-(2-fluoroethyl)-N-(4-(4-(2-methoxyphenyl)piperaz...)
Affinity DataKi:  2.21E+3nMAssay Description:Displacement of [3H]-DTG from rat sigma2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetAP-2 complex subunit sigma(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50339685(4-(Thiophen-3-yl)-N-(4-(4-(2-(2-fluoroethoxy)pheny...)
Affinity DataKi:  5.96E+3nMAssay Description:Displacement of [3H]-DTG from rat sigma2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetAP-2 complex subunit sigma(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM26739(URB 597 | URB597 | CHEMBL184238 | 3-(3-carbamoylph...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetAP-2 complex subunit sigma(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM81790(NSC_2159 | CAS_71675-85-9 | Amisulpride | US101672...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2012
Entry Details Article
PubMed