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Report error Found 92 Enz. Inhib. hit(s) with Target = 'ADP-ribosylation factor GTPase-activating protein 1'
TargetADP-ribosylation factor GTPase-activating protein 1(Homo sapiens)
National Clinical Research Center For Geriatrics

Curated by ChEMBL
LigandPNGBDBM50373058(CHEMBL259181)
Affinity DataEC50:  500nMAssay Description:Inhibition of ARFGAP1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94663((6Z)-6-[[5-(3-chlorophenyl)-2-furanyl]methylidene]...)
Affinity DataIC50: 2.03E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94657(5-azanyl-N-(5-chloranyl-2-methoxy-phenyl)-1-[2-[(3...)
Affinity DataIC50: 5.04E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM43208(SMR000018499 | MLS000101523 | cid_3404474 | N-[5-(...)
Affinity DataIC50: 7.92E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94686(cid_9593463 | SMR000283966 | MLS000687260 | N'-[(E...)
Affinity DataIC50: 1.03E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94655(MLS001234975 | SMR000810924 | 2-[2-(2,6-dimethylmo...)
Affinity DataIC50: 1.07E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94665(MLS001230224 | SMR000678732 | N-[(Z)-[4-methoxy-3-...)
Affinity DataIC50: 1.24E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM40968(N-(1,3-benzodioxol-5-ylmethyl)-7-methyl-furo[2,3-b...)
Affinity DataIC50: 1.67E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94683(N-[4-(aminocarbonyl)phenyl]-5-({2-nitro-4-methylph...)
Affinity DataIC50: 1.67E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94681(MLS000030984 | 1-(2,3-dihydro-1,4-benzodioxin-6-yl...)
Affinity DataIC50: 1.77E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95208(2-(5-azanyl-1,2,3,4-tetrazol-1-yl)-N-[(E)-[5-(2,5-...)
Affinity DataIC50: 1.78E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM41086(N-[3-chloranyl-4-(2-oxidanylidenechromen-3-yl)phen...)
Affinity DataIC50: 1.79E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95229(MLS001234985 | SMR000810925 | N-(3-chlorophenyl)-2...)
Affinity DataIC50: 1.83E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95242(MLS003123272 | SMR001291104 | cid_49786470 | N-[2-...)
Affinity DataIC50: 1.83E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM67822(SMR000142546 | 1-[2-(2,4-dichlorophenoxy)ethyl]-3-...)
Affinity DataIC50: 1.84E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95203(MLS000390717 | SMR000259755 | (E)-3-[3-(4-methylph...)
Affinity DataIC50: 2.03E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94694(MLS000723379 | [2-methoxy-4-[(Z)-[(6-methylpyridin...)
Affinity DataIC50: 2.10E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM41188(MLS000111800 | SMR000107719 | cid_2909321)
Affinity DataIC50: 2.31E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94689(cid_7256699 | SMR000808695 | 2-[[2-(1-azepanyl)-2-...)
Affinity DataIC50: 2.31E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM88864(2-(2,4-Dichloro-benzylsulfanyl)-6,7,8,9-tetrahydro...)
Affinity DataIC50: 2.38E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94700(cid_241318 | 1,3-bis[(2-methoxyphenyl)methylidenea...)
Affinity DataIC50: 2.56E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94705(SMR000808696 | cid_7256700 | 7-methyl-2-[2-(4-meth...)
Affinity DataIC50: 2.62E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94693(7-methyl-2-[[2-oxo-2-[4-(phenylmethyl)-1-piperidin...)
Affinity DataIC50: 2.69E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95200(2-[4-[(Z)-(2-amino-4-oxo-5-thiazolylidene)methyl]-...)
Affinity DataIC50: 2.83E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95236(1-methyl-3-indolecarboxylic acid [2-(3,5-dimethyl-...)
Affinity DataIC50: 2.84E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94697(2-(2-furyl)-6-[2-oxo-2-(1-piperidinyl)ethoxy]-4H-c...)
Affinity DataIC50: 2.85E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95211(cid_5168242 | N-(2,3-dimethylphenyl)-2-(4-oxo-[1]b...)
Affinity DataIC50: 2.87E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM55790(MLS000678964 | cid_5829079 | (E)-3-phenyl-N-(4-pyr...)
Affinity DataIC50: 2.88E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM54212(MLS000326804 | N-[[2,6-bis(chloranyl)phenyl]methox...)
Affinity DataIC50: 3.03E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95204([2-[2-(difluoromethoxy)anilino]-2-oxoethyl] 4-[(4-...)
Affinity DataIC50: 3.13E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94669(7-methyl-2-(2-oxo-2-piperidin-1-ylethyl)sulfanylpy...)
Affinity DataIC50: 3.20E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM67993(3-(1,3-diphenyl-1H-pyrazol-4-yl)-N-1,3-thiazol-2-y...)
Affinity DataIC50: 3.21E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM48131(MLS000058395 | cid_2084400 | SMR000064062 | 1H-ind...)
Affinity DataIC50: 3.24E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95241(N-[2-methoxy-4-[[2-(4-nitrophenoxy)-1-oxoethyl]ami...)
Affinity DataIC50: 3.36E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95224(SMR000646826 | MLS001146387 | N-[(E)-[3-[(4-bromop...)
Affinity DataIC50: 3.43E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95225(cid_24818752 | 1-(3,4-dimethylphenyl)-3-[[2-(4-nit...)
Affinity DataIC50: 3.45E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94673(5-bromo-N-(2-methoxy-5-nitrophenyl)thiophene-2-car...)
Affinity DataIC50: 3.56E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94668(SMR000385055 | MLS001010721 | 4-acetamido-N-[4-(3-...)
Affinity DataIC50: 3.66E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM28655(2-(5-butoxy-1-oxo-1,2-dihydroisoquinolin-2-yl)-N-(...)
Affinity DataIC50: 3.68E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM34388(N-[5-(4-chlorophenyl)-1,2,4-thiadiazol-3-yl]-2-[(1...)
Affinity DataIC50: 3.76E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94706(SMR000034292 | MLS000830253 | cid_658947)
Affinity DataIC50: 3.81E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95214(SMR000426956 | 3-(2-Pyridin-3-yl-quinazolin-4-ylam...)
Affinity DataIC50: 3.83E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95217(MLS001028814 | cid_20920416 | N-benzyl-1-[2-(4-met...)
Affinity DataIC50: 4.06E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95209(N-[4-[2-[[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1,2...)
Affinity DataIC50: 4.07E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95198(cid_1090038 | SMR000178542 | N-[4-(1H-benzimidazol...)
Affinity DataIC50: 4.20E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95215(cid_2112635 | 4-[[(2,5,6-trimethyl-4-thieno[2,3-d]...)
Affinity DataIC50: 4.25E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM43011(2-[(6-amino-3,5-dicyano-4-thiophen-2-yl-2-pyridiny...)
Affinity DataIC50: 4.32E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95201(3-(2-Chloro-6-fluoro-phenyl)-4,5-dihydro-isoxazole...)
Affinity DataIC50: 4.36E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM40512(2-({3-[2-(3,4-dimethoxyphenyl)ethyl]-4-oxo-3,4-dih...)
Affinity DataIC50: 4.40E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rat)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95230(cid_7256720 | MLS001234953 | SMR000810902 | N-(3-f...)
Affinity DataIC50: 4.49E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2013
Entry Details
PCBioAssay
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