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Report error Found 150 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2'
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544625(CHEMBL4632373)
Affinity DataEC50:  24nMAssay Description:Positive modulator activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544624(CHEMBL4643961)
Affinity DataEC50:  31nMAssay Description:Positive modulator activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544623(CHEMBL4635729)
Affinity DataEC50:  32nMAssay Description:Positive modulator activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544622(CHEMBL4645305)
Affinity DataEC50:  43nMAssay Description:Positive modulator activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544621(CHEMBL4646555)
Affinity DataEC50:  19nMAssay Description:Positive modulator activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50267632(4-(3-Hydroxy-2-methoxy-benzoyl)-1-(2-p-fluoropheny...)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mobilization i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544628(CHEMBL4638006)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mobilization i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544627(CHEMBL4636980)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mobilization i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401395(CHEMBL2206440)
Affinity DataEC50:  210nMAssay Description:Agonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mobilization i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544626(CHEMBL4646835)
Affinity DataEC50:  170nMAssay Description:Agonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mobilization i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544625(CHEMBL4632373)
Affinity DataEC50:  210nMAssay Description:Agonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mobilization i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544624(CHEMBL4643961)
Affinity DataEC50:  120nMAssay Description:Agonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mobilization i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544623(CHEMBL4635729)
Affinity DataEC50:  280nMAssay Description:Agonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mobilization i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544622(CHEMBL4645305)
Affinity DataEC50:  260nMAssay Description:Agonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mobilization i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544621(CHEMBL4646555)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mobilization i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544620(CHEMBL4642761)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mobilization i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544619(CHEMBL4639821)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mobilization i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544618(CHEMBL4635373)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mobilization i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544617(CHEMBL4638687)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mobilization i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544631(CHEMBL4645193)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mobilization i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544630(CHEMBL4641860)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mobilization i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544629(CHEMBL4635960)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mobilization i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50267632(4-(3-Hydroxy-2-methoxy-benzoyl)-1-(2-p-fluoropheny...)
Affinity DataEC50: <5.01E+4nMAssay Description:Agonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mobilization i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544628(CHEMBL4638006)
Affinity DataEC50: <5.01E+4nMAssay Description:Agonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mobilization i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544627(CHEMBL4636980)
Affinity DataEC50: <5.01E+4nMAssay Description:Agonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mobilization i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401395(CHEMBL2206440)
Affinity DataEC50:  209nMAssay Description:Agonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mobilization i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544626(CHEMBL4646835)
Affinity DataEC50:  174nMAssay Description:Agonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mobilization i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544625(CHEMBL4632373)
Affinity DataEC50:  209nMAssay Description:Agonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mobilization i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544624(CHEMBL4643961)
Affinity DataEC50:  120nMAssay Description:Agonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mobilization i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544623(CHEMBL4635729)
Affinity DataEC50:  282nMAssay Description:Agonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mobilization i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544622(CHEMBL4645305)
Affinity DataEC50:  263nMAssay Description:Agonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mobilization i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401395(CHEMBL2206440)
Affinity DataEC50:  19nMAssay Description:Positive modulator activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544626(CHEMBL4646835)
Affinity DataEC50:  25nMAssay Description:Positive modulator activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544625(CHEMBL4632373)
Affinity DataEC50:  24nMAssay Description:Positive modulator activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544624(CHEMBL4643961)
Affinity DataEC50:  31nMAssay Description:Positive modulator activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544623(CHEMBL4635729)
Affinity DataEC50:  32nMAssay Description:Positive modulator activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544622(CHEMBL4645305)
Affinity DataEC50:  43nMAssay Description:Positive modulator activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544621(CHEMBL4646555)
Affinity DataEC50:  19nMAssay Description:Positive modulator activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401395(CHEMBL2206440)
Affinity DataEC50:  19nMAssay Description:Positive modulator activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544626(CHEMBL4646835)
Affinity DataEC50:  25nMAssay Description:Positive modulator activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as increase in intracellular Ca2+ mob...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544628(CHEMBL4638006)
Affinity DataIC50: 5.40nMAssay Description:Antagonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as inhibition of 5HT-induced intracellular Ca...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544628(CHEMBL4638006)
Affinity DataIC50: 5.5nMAssay Description:Antagonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as inhibition of 5HT-induced intracellular Ca...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544628(CHEMBL4638006)
Affinity DataIC50: 6.20nMAssay Description:Antagonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells assessed as inhibition of 5HT-induced intracellular Ca2+ mobilization inc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544628(CHEMBL4638006)
Affinity DataIC50: 6.20nMAssay Description:Antagonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells assessed as inhibition of 5HT-induced intracellular Ca2+ mobilization inc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50267632(4-(3-Hydroxy-2-methoxy-benzoyl)-1-(2-p-fluoropheny...)
Affinity DataIC50: 9.10nMAssay Description:Antagonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells assessed as inhibition of 5HT-induced intracellular Ca2+ mobilization inc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50267632(4-(3-Hydroxy-2-methoxy-benzoyl)-1-(2-p-fluoropheny...)
Affinity DataIC50: 9.20nMAssay Description:Antagonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells assessed as inhibition of 5HT-induced intracellular Ca2+ mobilization inc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544627(CHEMBL4636980)
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells assessed as inhibition of 5HT-induced intracellular Ca2+ mobilization inc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50544627(CHEMBL4636980)
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells assessed as inhibition of 5HT-induced intracellular Ca2+ mobilization inc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50267632(4-(3-Hydroxy-2-methoxy-benzoyl)-1-(2-p-fluoropheny...)
Affinity DataIC50: 22nMAssay Description:Antagonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as inhibition of 5HT-induced intracellular Ca...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50267632(4-(3-Hydroxy-2-methoxy-benzoyl)-1-(2-p-fluoropheny...)
Affinity DataIC50: 22nMAssay Description:Antagonist activity at human 5HT2A/mGlu2 receptor expressed in HEK293 cells co-expressing Gqo5 assessed as inhibition of 5HT-induced intracellular Ca...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
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