BDBM50614163 CHEMBL5288779
SMILES c1ccc(cc1)CNc2c3c(cncn3)c4ccc(cc4n2)C(=O)O
InChI Key InChIKey=HEVVNKYNJCSHFA-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 15 hits for monomerid = 50614163
TargetCasein kinase II subunit alpha(Human)
University of North Carolina At Chapel Hill
Curated by ChEMBL
University of North Carolina At Chapel Hill
Curated by ChEMBL
Affinity DataIC50: 920nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K10 by NanoBR...More data for this Ligand-Target Pair
3D Structure (crystal)TargetCasein kinase II subunit alpha'(Human)
University of North Carolina At Chapel Hill
Curated by ChEMBL
University of North Carolina At Chapel Hill
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of C-terminal Nano-Luc fused human CK2alpha' expressed in HEK293 cells using NanoBRET NanoGlo substrate in presence of tracer K5 by NanoBR...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Human)
University of North Carolina At Chapel Hill
Curated by ChEMBL
University of North Carolina At Chapel Hill
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of wild type human CK2alpha in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha'(Human)
University of North Carolina At Chapel Hill
Curated by ChEMBL
University of North Carolina At Chapel Hill
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of wild type human CK2alpha' in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
TargetDeath-associated protein kinase 3(Human)
University of North Carolina At Chapel Hill
Curated by ChEMBL
University of North Carolina At Chapel Hill
Curated by ChEMBL
Affinity DataIC50: 1.50E+6nMAssay Description:Inhibition of wild type human DAPK3 in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
TargetHomeodomain-interacting protein kinase 1(Human)
University of North Carolina At Chapel Hill
Curated by ChEMBL
University of North Carolina At Chapel Hill
Curated by ChEMBL
Affinity DataIC50: 1.80E+6nMAssay Description:Inhibition of wild type human HIPK1 in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
TargetDeath-associated protein kinase 2(Human)
University of North Carolina At Chapel Hill
Curated by ChEMBL
University of North Carolina At Chapel Hill
Curated by ChEMBL
Affinity DataIC50: 1.50E+6nMAssay Description:Inhibition of wild type human DAPK2 in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
TargetHomeodomain-interacting protein kinase 3(Human)
University of North Carolina At Chapel Hill
Curated by ChEMBL
University of North Carolina At Chapel Hill
Curated by ChEMBL
Affinity DataIC50: 9.00E+5nMAssay Description:Inhibition of wild type human HIPK3 in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
TargetMyosin light chain kinase family member 4(Human)
University of North Carolina At Chapel Hill
Curated by ChEMBL
University of North Carolina At Chapel Hill
Curated by ChEMBL
Affinity DataIC50: 1.00E+7nMAssay Description:Inhibition of wild type human MYLK4 in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Human)
University of North Carolina At Chapel Hill
Curated by ChEMBL
University of North Carolina At Chapel Hill
Curated by ChEMBL
Affinity DataIC50: 5.30E+6nMAssay Description:Inhibition of wild type human PIK3CG in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 3-kinase C2 domain-containing subunit gamma(Human)
University of North Carolina At Chapel Hill
Curated by ChEMBL
University of North Carolina At Chapel Hill
Curated by ChEMBL
Affinity DataIC50: 4.50E+6nMAssay Description:Inhibition of wild type human PIK3C2G in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
University of North Carolina At Chapel Hill
Curated by ChEMBL
University of North Carolina At Chapel Hill
Curated by ChEMBL
Affinity DataIC50: 7.60E+5nMAssay Description:Inhibition of wild type human DYRK1A in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
TargetHomeodomain-interacting protein kinase 2(Human)
University of North Carolina At Chapel Hill
Curated by ChEMBL
University of North Carolina At Chapel Hill
Curated by ChEMBL
Affinity DataIC50: 6.00E+5nMAssay Description:Inhibition of wild type human HIPK2 in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 17B(Human)
University of North Carolina At Chapel Hill
Curated by ChEMBL
University of North Carolina At Chapel Hill
Curated by ChEMBL
Affinity DataIC50: 2.80E+6nMAssay Description:Inhibition of wild type human DRAK2 in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 19(Human)
University of North Carolina At Chapel Hill
Curated by ChEMBL
University of North Carolina At Chapel Hill
Curated by ChEMBL
Affinity DataIC50: 3.70E+6nMAssay Description:Inhibition of wild type human YSK4 in presence of ATP by radiometric kinase assayMore data for this Ligand-Target Pair