BDBM50573191 CHEMBL4870218

SMILES CN1C(=O)C(=C(C=N1)Nc2ccc(cc2)CN(C)C)Cl

InChI Key InChIKey=NERLHNQOXJXDPS-UHFFFAOYSA-N

Data  1 IC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50573191   

TargetNucleosome-remodeling factor subunit BPTF(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50573191(CHEMBL4870218)
Affinity DataIC50: 310nMAssay Description:Inhibition of HIS9-tagged BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)