BDBM50359970 CHEMBL1927262

SMILES Cc1ccc(cc1c2c3c(c4c(n[nH]c4n2)N)CCCC3)F

InChI Key InChIKey=YPULTKAHHAYKOE-UHFFFAOYSA-N

Data  1 IC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50359970   

TargetEphrin type-A receptor 4(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50359970(CHEMBL1927262)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of his-tagged EPHA4-mediated poly(Glu,Tyr) phosphorylation after 75 mins using E4:Y1 as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)