BDBM50319157 4-Cyano-8-methoxy-3-methyl-1-propyl-imidazo[1,5-a]pyrido-[3,2-e]pyrazine::CHEMBL1086265

SMILES CCCc1nc(c2n1c3c(ccc(n3)OC)nc2C#N)C

InChI Key InChIKey=GQYPTVVKCVYXLX-UHFFFAOYSA-N

Data  1 IC50

PDB links: 1 PDB ID matches this monomer.

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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50319157   

LigandPNGBDBM50319157(4-Cyano-8-methoxy-3-methyl-1-propyl-imidazo[1,5-a]...)
Affinity DataIC50: 11nMAssay Description:Inhibition of human recombinant PDE10A expressed in baculovirus-SF21 cell system assessed as hydrolysis of [3H]cAMP after 1 hr by liquid scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)