BDBM50210161 CHEMBL1363184::LY-303511

SMILES O=c1cc(oc2c(cccc12)-c1ccccc1)N1CCNCC1

InChI Key InChIKey=NGAGMBNBKCDCDJ-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50210161   

TargetBromodomain-containing protein 4(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50210161(LY-303511 | CHEMBL1363184)
Affinity DataIC50: 9.05E+3nMAssay Description:Inhibition of immobilized N-LY294002 bead binding to C-terminal Flag-tagged BRD4 (unknown origin) expressed in HEK293T cell nuclear extract incubated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details Article
PubMed
TargetBromodomain-containing protein 2(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50210161(LY-303511 | CHEMBL1363184)
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of immobilized N-LY294002 bead binding to BRD2 (unknown origin) expressed in HEK293T cell nuclear extract incubated for 1 hr by LC-MS/MS a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details Article
PubMed
TargetBromodomain-containing protein 3(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50210161(LY-303511 | CHEMBL1363184)
Affinity DataIC50: 1.15E+4nMAssay Description:Inhibition of immobilized N-LY294002 bead binding to BRD3 (unknown origin) expressed in HEK293T cell nuclear extract incubated for 1 hr by LC-MS/MS a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details Article
PubMed