BDBM50094670 1-(4-Dipropylamino-1,3,4,5-tetrahydro-benzo[cd]indol-6-yl)-ethanone::CHEMBL276031::LY 293284::LY-293284::LY-293384

SMILES CCCN(CCC)C1Cc2c[nH]c3ccc(C(C)=O)c(C1)c23

InChI Key InChIKey=CKYZLYQSDNLGPT-UHFFFAOYSA-N

Data  15 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 16 hits for monomerid = 50094670   

Target5-hydroxytryptamine receptor 1A(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094670(LY-293384 | LY 293284 | LY-293284 | CHEMBL276031 |...)
Affinity DataEC50:  0.130nMAssay Description:EC50 for inhibition of 50 uM forskolin-stimulated cAMP accumulation against 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094670(LY-293384 | LY 293284 | LY-293284 | CHEMBL276031 |...)
Affinity DataKi:  0.0880nMAssay Description:Inhibition constant of 50 uM forskolin-stimulated cAMP accumulation against 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50094670(LY-293384 | LY 293284 | LY-293284 | CHEMBL276031 |...)
Affinity DataKi:  66.9nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details
PubMed
LigandPNGBDBM50094670(LY-293384 | LY 293284 | LY-293284 | CHEMBL276031 |...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details
PubMed
LigandPNGBDBM50094670(LY-293384 | LY 293284 | LY-293284 | CHEMBL276031 |...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details
PubMed
LigandPNGBDBM50094670(LY-293384 | LY 293284 | LY-293284 | CHEMBL276031 |...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details
PubMed
LigandPNGBDBM50094670(LY-293384 | LY 293284 | LY-293284 | CHEMBL276031 |...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details
PubMed
TargetAlpha-1A adrenergic receptor(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50094670(LY-293384 | LY 293284 | LY-293284 | CHEMBL276031 |...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details
PubMed
TargetAlpha-2C adrenergic receptor(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50094670(LY-293384 | LY 293284 | LY-293284 | CHEMBL276031 |...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details
PubMed
TargetBeta-2 adrenergic receptor(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50094670(LY-293384 | LY 293284 | LY-293284 | CHEMBL276031 |...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details
PubMed
LigandPNGBDBM50094670(LY-293384 | LY 293284 | LY-293284 | CHEMBL276031 |...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details
PubMed
TargetD(1A) dopamine receptor(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50094670(LY-293384 | LY 293284 | LY-293284 | CHEMBL276031 |...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details
PubMed
TargetD(2) dopamine receptor(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50094670(LY-293384 | LY 293284 | LY-293284 | CHEMBL276031 |...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details
PubMed
LigandPNGBDBM50094670(LY-293384 | LY 293284 | LY-293284 | CHEMBL276031 |...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details
PubMed
LigandPNGBDBM50094670(LY-293384 | LY 293284 | LY-293284 | CHEMBL276031 |...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details
PubMed
TargetHistamine H1 receptor(Rat)
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50094670(LY-293384 | LY 293284 | LY-293284 | CHEMBL276031 |...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2011
Entry Details
PubMed