BDBM292437 (2-(5-phenylpyrazolo[1,5-a]pyrimidin-3-yl)pyridin-4-yl)((R)-2-((S)-pyrrolidin-2-yl)piperidin-1-yl)methanone::US10100058, Example 93

SMILES O=C(N1CCCC[C@@H]1[C@@H]1CCCN1)c1ccnc(c1)-c1cnn2ccc(nc12)-c1ccccc1

InChI Key InChIKey=YDVLFOTYEFCKOA-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 292437   

LigandChemical structure of BindingDB Monomer ID 292437BDBM292437(US10100058, Example 93 | (2-(5-phenylpyrazolo[1,5-...)
Affinity DataIC50: 27.8nMAssay Description:The biochemical activity of recombinant CaMKIIδ was measured by monitoring the phosphorylation of a target peptide using Homogenous Time Resolve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2019
Entry Details
US Patent