BDBM204923 phosphonoacetohydroxamate (PhAH)

SMILES C(C(=O)NO)P(=O)(O)O

InChI Key InChIKey=LDKRAXXVBWHMRH-UHFFFAOYSA-N

Data  3 IC50

PDB links: 6 PDB IDs match this monomer.

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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 204923   

TargetAlpha-enolase(Human)
University of Texas M. D. Anderson Cancer Center

LigandPNGBDBM204923(phosphonoacetohydroxamate (PhAH))
Affinity DataIC50: 53.2nMpH: 7.4Assay Description:Enolase activity was measured by two different methods: a fluorometric NADH-linked assay or adirect spectrophotometric assay via formation of PEP. In...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details Article
PubMed
TargetGamma-enolase(Human)
University of Texas M. D. Anderson Cancer Center

LigandPNGBDBM204923(phosphonoacetohydroxamate (PhAH))
Affinity DataIC50: 62.3nMpH: 7.4Assay Description:Enolase activity was measured by two different methods: a fluorometric NADH-linked assay or adirect spectrophotometric assay via formation of PEP. In...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAlpha-enolase(Human)
University of Texas M. D. Anderson Cancer Center

LigandPNGBDBM204923(phosphonoacetohydroxamate (PhAH))
Affinity DataIC50: 51nMAssay Description:Inhibition of ENO1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed