BDBM50183472 5-(2,4-dimethoxyphenyl)-4-(furan-2-carbonyl)-3-hydroxy-1-(2-morpholinoethyl)-1H-pyrrol-2(5H)-one::CHEMBL381077::cid_2909444

SMILES COc1ccc(C2C(C(=O)c3ccco3)C(=O)C(=O)N2CCN2CCOCC2)c(OC)c1

InChI Key InChIKey=TYPCDWZKHSXFOG-UHFFFAOYSA-N

Data  2 KI  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50183472   

TargetN-formyl peptide receptor 2(Human)
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM50183472(cid_2909444 | CHEMBL381077 | 5-(2,4-dimethoxypheny...)
Affinity DataIC50: 6.67E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH 1R03MH076381-01 Assay for Formylpeptide Receptor Family Ligands PI: Bruce S. Edwards, Ph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2011
Entry Details
PCBioAssay
TargetfMet-Leu-Phe receptor(Human)
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM50183472(cid_2909444 | CHEMBL381077 | 5-(2,4-dimethoxypheny...)
Affinity DataIC50: 9.80E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH 1R03MH076381-01 Assay for Formylpeptide Receptor Family Ligands PI: Bruce S. Edwards, Ph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2011
Entry Details
PCBioAssay
TargetIntegrase(Human immunodeficiency virus type 1)
University of Houston

Curated by ChEMBL
LigandPNGBDBM50183472(cid_2909444 | CHEMBL381077 | 5-(2,4-dimethoxypheny...)
Affinity DataIC50: 3.95E+5nMAssay Description:Inhibition of strand transfer activity of HIV1 integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
University of Houston

Curated by ChEMBL
LigandPNGBDBM50183472(cid_2909444 | CHEMBL381077 | 5-(2,4-dimethoxypheny...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of 3'-processing activity of HIV1 integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetfMet-Leu-Phe receptor(Human)
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM50183472(cid_2909444 | CHEMBL381077 | 5-(2,4-dimethoxypheny...)
Affinity DataKi:  6.40E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH 1R03MH076381-01 Assay for Formylpeptide Receptor Family Ligands PI: Bruce S. Edwards, Ph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2011
Entry Details
PCBioAssay
TargetN-formyl peptide receptor 2(Human)
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM50183472(cid_2909444 | CHEMBL381077 | 5-(2,4-dimethoxypheny...)
Affinity DataKi: >4.03E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH 1R03MH076381-01 Assay for Formylpeptide Receptor Family Ligands PI: Bruce S. Edwards, Ph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2011
Entry Details
PCBioAssay