BDBM50280251 4-Methyl-N-[2-(3-oxo-1-phenyl-1,3-dihydro-isobenzofuran-1-ylamino)-ethyl]-benzenesulfonamide::CHEMBL38243::UK-73093

SMILES Cc1ccc(cc1)S(=O)(=O)NCCNC1(OC(=O)c2ccccc12)c1ccccc1

InChI Key InChIKey=DAJOKVSLVAAJLL-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50280251   

TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50280251(UK-73093 | 4-Methyl-N-[2-(3-oxo-1-phenyl-1,3-dihyd...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibitory concentration required for the displacement of [3H]NT from neurotensin receptor in mouse; value ranges from 4-6 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeurotensin receptor type 1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50280251(UK-73093 | 4-Methyl-N-[2-(3-oxo-1-phenyl-1,3-dihyd...)
Affinity DataIC50: 4.90E+4nMAssay Description:Inhibitory concentration required for the displacement of [3H]NT from neurotensin receptor in ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeurotensin receptor type 1/2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280251(UK-73093 | 4-Methyl-N-[2-(3-oxo-1-phenyl-1,3-dihyd...)
Affinity DataIC50: 5.50E+3nMAssay Description:Compound was evaluated for its ability to displace [3H]NT from the neurotensin receptor of bovine brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article