BDBM50475037 CHEMBL361383::TP-101

SMILES CC(C)[C@H](NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CC1CCCCC1)C(=O)NC(Cc1ccc(O)cc1)C=O

InChI Key InChIKey=PBHZSZHBJWAKIL-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50475037   

LigandPNGBDBM50475037(CHEMBL361383 | TP-101)
Affinity DataIC50: 330nMAssay Description:Inhibitory concentration to inhibit chymotrypsin-like activity of 20S proteasome prepared from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50475037(CHEMBL361383 | TP-101)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibitory concentration to inhibit trypsin-like activity of 20S proteasome from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
LigandPNGBDBM50475037(CHEMBL361383 | TP-101)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibitory concentration to inhibit the PGPH activity of 20S proteasome prepared from human leukemia HL-60 cells was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed