BDBM50135884 (S)-1-(2,6-dimethylphenoxy)propan-2-amine::(S)-2-(2,6-Dimethyl-phenoxy)-1-methyl-ethylamine::CHEMBL146855::MEXILETINE

SMILES Cc1cccc(c1OC[C@H](C)N)C

InChI Key InChIKey=VLPIATFUUWWMKC-UHFFFAOYSA-N

Data  1 EC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50135884   

TargetSodium channel protein type 4 subunit alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50135884((S)-1-(2,6-dimethylphenoxy)propan-2-amine | (S)-2-...)
Affinity DataEC50:  2.69E+4nMAssay Description:Inhibition of Nav1.4 ion channel assessed as reduction in cumulative sodium currentMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed